Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 942 productos de "Receptor 5-HT"
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Flibanserin-d4
CAS:<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Fórmula:C20H21F3N4OPureza:98%Forma y color:SolidPeso molecular:394.43Paliperidone Palmitate
CAS:<p>Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>Fórmula:C39H57FN4O4Pureza:98%Forma y color:SolidPeso molecular:664.89Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Fórmula:C22H25N3O3Pureza:99.94%Forma y color:SolidPeso molecular:379.45Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Fórmula:C17H17Cl2NOForma y color:SolidPeso molecular:322.23Dehydroaripiprazole
CAS:<p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>Fórmula:C23H25Cl2N3O2Pureza:98.7%Forma y color:SolidPeso molecular:446.37Clozapine-d8
CAS:<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Fórmula:C18H19ClN4Forma y color:SolidPeso molecular:334.875-HT3 antagonist 5
CAS:<p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>Fórmula:C16H13N3O2Pureza:99.84%Forma y color:SolidPeso molecular:279.29WAY-100635
CAS:<p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>Fórmula:C25H34N4O2Pureza:98.972%Forma y color:SolidPeso molecular:422.56Alosetron D3 Hydrochloride
CAS:<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Fórmula:C17H19ClN4OPureza:98%Forma y color:SolidPeso molecular:333.83Nefazodone
CAS:<p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>Fórmula:C25H32ClN5O2Pureza:99.85%Forma y color:White To Off-White Crystalline PowderPeso molecular:470.015-HT2B antagonist-1
CAS:<p>Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.</p>Fórmula:C11H14BrN5Pureza:99.965%Forma y color:SolidPeso molecular:296.17Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Fórmula:C21H26D6Cl2N4OPureza:98%Forma y color:SolidPeso molecular:433.45Ziprasidone amino acid
CAS:<p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>Fórmula:C21H23ClN4O2SForma y color:SolidPeso molecular:430.95Asenapine
CAS:<p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>Fórmula:C17H16ClNOPureza:99.64%Forma y color:CoaPeso molecular:285.77Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Fórmula:C26H27N5O2Pureza:98%Forma y color:SolidPeso molecular:449.573-Hydroxy agomelatine D3
CAS:<p>3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).</p>Fórmula:C15H17NO3Pureza:98%Forma y color:SolidPeso molecular:262.32Levomepromazine
CAS:Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.Fórmula:C19H24N2OSPureza:99.15%Forma y color:SolidPeso molecular:328.474,4-Diphenylbutylamine hydrochloride
CAS:<p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>Fórmula:C16H20ClNForma y color:SolidPeso molecular:261.79BW 723C86
CAS:<p>BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.</p>Fórmula:C16H19ClN2OSPureza:99.35%Forma y color:SolidPeso molecular:322.85LY310762
CAS:LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.Fórmula:C24H27FN2O2·HClPureza:99.8%Forma y color:SolidPeso molecular:430.94
