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Receptor 5-HT

Receptor 5-HT

Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.

Se han encontrado 942 productos de "Receptor 5-HT"

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  • AVN-101

    CAS:
    <p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C21H25ClN2
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:340.89
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Forma y color:Solid
    Peso molecular:324.24
  • Mosapride

    CAS:
    <p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>
    Fórmula:C21H25ClFN3O3
    Pureza:99.56%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:421.89
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H24ClN2NaO4S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:458.93
  • Vilazodone Hydrochloride

    CAS:
    <p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>
    Fórmula:C26H27N5O2·HCl
    Pureza:99.56% - >99.99%
    Forma y color:Solid
    Peso molecular:477.99
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:417.89
  • lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Fórmula:C31H36FN3O4S
    Pureza:95.83% - 99.95%
    Forma y color:Solid
    Peso molecular:565.7
  • Cerlapirdine

    CAS:
    <p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>
    Fórmula:C22H23N3O3S
    Pureza:98.77%
    Forma y color:Solid
    Peso molecular:409.5
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Forma y color:Solid
    Peso molecular:463.87
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Fórmula:C18H20N4
    Pureza:99.15% - 99.82%
    Forma y color:Solid
    Peso molecular:292.38
  • Indophagolin

    CAS:
    <p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>
    Fórmula:C19H15BrClF3N2O3S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:523.75
  • Amperozide

    CAS:
    <p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>
    Fórmula:C23H29F2N3O
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:401.49
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Fórmula:C14H25Cl2N3O3
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:354.27
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:256.73
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Forma y color:Solid
    Peso molecular:379.36
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Fórmula:C16H23Cl2N5O2
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:388.29
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:352.9
  • LP-533401 hydrochloride

    CAS:
    LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.
    Fórmula:C27H23ClF4N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:562.94
  • Ketanserin tartrate

    CAS:
    Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.
    Fórmula:C26H28FN3O9
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:545.51
  • Tandospirone

    CAS:
    <p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>
    Fórmula:C21H29N5O2
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:383.49