
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 942 productos de "Receptor 5-HT"
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AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C21H25ClN2Pureza:99.61%Forma y color:SolidPeso molecular:340.89SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Forma y color:SolidPeso molecular:324.24Mosapride
CAS:<p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>Fórmula:C21H25ClFN3O3Pureza:99.56%Forma y color:White To Off-White Crystalline SolidPeso molecular:421.89Tianeptine sodium salt
CAS:<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Fórmula:C21H24ClN2NaO4SPureza:99.82%Forma y color:SolidPeso molecular:458.93Vilazodone Hydrochloride
CAS:<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Fórmula:C26H27N5O2·HClPureza:99.56% - >99.99%Forma y color:SolidPeso molecular:477.99Xaliproden hydrochloride
CAS:<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Fórmula:C24H23ClF3NPureza:99.99%Forma y color:SolidPeso molecular:417.89lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Forma y color:SolidPeso molecular:565.7Cerlapirdine
CAS:<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Fórmula:C22H23N3O3SPureza:98.77%Forma y color:SolidPeso molecular:409.5Cariprazine hydrochloride
CAS:<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Forma y color:SolidPeso molecular:463.87Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Forma y color:SolidPeso molecular:292.38Indophagolin
CAS:<p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>Fórmula:C19H15BrClF3N2O3SPureza:99.76%Forma y color:SolidPeso molecular:523.75Amperozide
CAS:<p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>Fórmula:C23H29F2N3OPureza:99.68%Forma y color:SolidPeso molecular:401.49Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Forma y color:SolidPeso molecular:354.27Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Fórmula:C12H17ClN2O2Pureza:99.35%Forma y color:SolidPeso molecular:256.73Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Fórmula:C18H22N2S·HBrPureza:98.85% - 99.98%Forma y color:SolidPeso molecular:379.36Azaphen dihydrochloride monohydrate
CAS:<p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C16H23Cl2N5O2Pureza:99.85%Forma y color:SolidPeso molecular:388.29RS-67333
CAS:<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Fórmula:C19H29ClN2O2Pureza:99.24%Forma y color:SolidPeso molecular:352.9LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Fórmula:C27H23ClF4N4O3Pureza:98%Forma y color:SolidPeso molecular:562.94Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Fórmula:C26H28FN3O9Pureza:99.68%Forma y color:SolidPeso molecular:545.51Tandospirone
CAS:<p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>Fórmula:C21H29N5O2Pureza:99.94%Forma y color:SolidPeso molecular:383.49
