
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 1025 productos de "Receptor 5-HT"
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Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Forma y color:SolidPeso molecular:383.495-HT6/5-HT2A receptor ligand-1
CAS:Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.Fórmula:C21H19FN2O2Forma y color:SolidPeso molecular:350.39Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFórmula:C16H23ClN2O2Forma y color:SolidPeso molecular:310.82Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Fórmula:C23H32Cl2FN3Pureza:98%Forma y color:SolidPeso molecular:440.42EMD 56551
CAS:EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Forma y color:SolidPeso molecular:393.522Usmarapride
CAS:Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.Fórmula:C23H31N5O6Forma y color:SolidPeso molecular:473.53RS 64459-193
CAS:RS 64459-193 has a high affinity for the 5-HT1A binding site.Fórmula:C26H36Cl2N2O2Forma y color:SolidPeso molecular:479.48EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Fórmula:C15H22N2OPureza:97.66% - 99.78%Forma y color:SolidPeso molecular:246.35Ref: TM-T11183
1mg87,00€2mg118,00€5mg167,00€10mg202,00€25mg449,00€50mg652,00€100mg888,00€500mg1.783,00€1mL*10mM (DMSO)166,00€Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Fórmula:C18H19NForma y color:SolidPeso molecular:249.35SB 714786
CAS:SB 714786 is a selective antagonist of 5-HT1D.Fórmula:C26H28N4OPureza:98%Forma y color:SolidPeso molecular:412.53Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Fórmula:C21H25ClN2O4SPureza:99.57%Forma y color:SolidPeso molecular:436.95CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Fórmula:C19H28ClN5OPureza:99.72%Forma y color:SolidPeso molecular:377.91Ref: TM-T22671
1mg48,00€5mg101,00€10mg170,00€25mg270,00€50mg386,00€100mg520,00€1mL*10mM (DMSO)124,00€Trelanserin
CAS:Trelanserin (SL-650472) is an antagonist of the serotonin receptor.Fórmula:C24H24FN5O2SForma y color:SolidPeso molecular:465.54MHP 133
CAS:MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).Fórmula:C17H20ClN5O3Pureza:98%Forma y color:SolidPeso molecular:377.83Bopindolol
CAS:Bopindolol: oral β1/β2-ARs antagonist and partial agonist; prodrug of pindolol for hypertension research.Fórmula:C23H28N2O3Forma y color:SolidPeso molecular:380.48AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Fórmula:C20H19ClN2O3SPureza:98%Forma y color:SolidPeso molecular:402.89WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Fórmula:C14H18N2Pureza:98%Forma y color:SolidPeso molecular:214.31Iloperidone hydrochloride
CAS:Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.Fórmula:C24H28ClFN2O4Pureza:98%Forma y color:SolidPeso molecular:462.95Isamoltane hemifumarate
CAS:5-HT1B antagonistFórmula:C16H22N202C4H404Pureza:98%Forma y color:SolidPeso molecular:332.4Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Forma y color:SolidPeso molecular:328.38
