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Receptor 5-HT

Receptor 5-HT

Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.

Se han encontrado 1025 productos de "Receptor 5-HT"

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  • LY 344864 S-enantiomer

    CAS:
    LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.
    Fórmula:C21H22FN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:351.42

    Ref: TM-T11902

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • PRX-08066 Maleic acid

    CAS:
    PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.
    Fórmula:C23H21ClFN5O4S
    Pureza:97.59%
    Forma y color:Solid
    Peso molecular:517.96

    Ref: TM-T6959

    1mg
    84,00€
    5mg
    172,00€
    10mg
    233,00€
    25mg
    419,00€
    50mg
    620,00€
    100mg
    882,00€
    200mg
    1.198,00€
    1mL*10mM (DMSO)
    401,00€
  • Bopindolol fumarate

    CAS:
    Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.
    Fórmula:C27H32N2O7
    Forma y color:Solid
    Peso molecular:496.56

    Ref: TM-T63356

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • DR4485 hydrochloride

    CAS:
    5-HT7 antagonist
    Fórmula:C26H29Cl3N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:491.88

    Ref: TM-T22750

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • OSU 6162 hydrochloride

    CAS:
    Dopamine stabilizer
    Fórmula:C15H24ClNO2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:317.88

    Ref: TM-T23114

    50mg
    3.132,00€
  • S-15535

    CAS:
    S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.
    Fórmula:C21H24N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:336.43

    Ref: TM-T28642

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Etoperidone hydrochloride

    CAS:
    Etoperidone hydrochloride is an antidepressant agent.
    Fórmula:C19H29Cl2N5O
    Forma y color:Solid
    Peso molecular:414.37

    Ref: TM-T24048

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • SLV-310

    CAS:
    SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.
    Fórmula:C25H24FN3O2
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:417.48

    Ref: TM-T28809

    1mg
    279,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Lesopitron dihydrochloride

    CAS:
    Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.
    Fórmula:C15H23Cl3N6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:393.74

    Ref: TM-T11839

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Naronapride

    CAS:
    Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.
    Fórmula:C27H41ClN4O5
    Forma y color:Solid
    Peso molecular:537.09

    Ref: TM-T63785

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • Fonazine

    CAS:
    Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.
    Fórmula:C19H25N3O2S2
    Forma y color:Solid
    Peso molecular:391.55

    Ref: TM-T31844

    25mg
    1.586,00€
    50mg
    2.072,00€
    100mg
    2.660,00€
  • Bopindolol (malonate)

    CAS:
    Bopindolol is a non-selective β-adrenergic receptor antagonist.
    Fórmula:C26H32N2O7
    Forma y color:Solid
    Peso molecular:484.549

    Ref: TM-T35871

    100mg
    298,00€
    500mg
    1.035,00€
  • (R)-Viloxazine Hydrochloride

    CAS:
    (R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.
    Fórmula:C13H20ClNO3
    Pureza:99.88% - 99.94%
    Forma y color:Solid
    Peso molecular:273.76

    Ref: TM-T22413

    1mg
    52,00€
    5mg
    111,00€
    10mg
    162,00€
    25mg
    235,00€
    50mg
    330,00€
    100mg
    452,00€
    200mg
    607,00€
    1mL*10mM (DMSO)
    101,00€
  • LEK 8841

    CAS:
    LEK 8841 is an ergoline derivative that is a potential antipsychotic.
    Fórmula:C21H24BrN3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:494.4

    Ref: TM-T25657

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • AP-521 (Free base)

    CAS:
    AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.
    Fórmula:C20H18N2O3S
    Forma y color:Solid
    Peso molecular:366.43

    Ref: TM-T26640

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Trimipramine

    CAS:
    Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.
    Fórmula:C20H26N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:294.43

    Ref: TM-T21364

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • 5-HT2A receptor agonist-2

    CAS:
    Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.
    Fórmula:C20H21ClN2O3
    Forma y color:Solid
    Peso molecular:372.85

    Ref: TM-T61507

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Alniditan

    CAS:
    Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.
    Fórmula:C17H26N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.41

    Ref: TM-T14190

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • OPC-14523 hydrochloride

    CAS:
    OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.
    Fórmula:C23H29Cl2N3O2
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:450.4

    Ref: TM-T62711

    5mg
    873,00€
    10mg
    1.160,00€
    25mg
    1.458,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
    1mL*10mM (DMSO)
    925,00€
  • Lidanserin

    CAS:
    Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.
    Fórmula:C26H31FN2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.53

    Ref: TM-T15754

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€