
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 1025 productos de "Receptor 5-HT"
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LY 344864 S-enantiomer
CAS:LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.Fórmula:C21H22FN3OPureza:98%Forma y color:SolidPeso molecular:351.42PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Fórmula:C23H21ClFN5O4SPureza:97.59%Forma y color:SolidPeso molecular:517.96Ref: TM-T6959
1mg84,00€5mg172,00€10mg233,00€25mg419,00€50mg620,00€100mg882,00€200mg1.198,00€1mL*10mM (DMSO)401,00€Bopindolol fumarate
CAS:Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.Fórmula:C27H32N2O7Forma y color:SolidPeso molecular:496.56DR4485 hydrochloride
CAS:5-HT7 antagonistFórmula:C26H29Cl3N2OPureza:98%Forma y color:SolidPeso molecular:491.88OSU 6162 hydrochloride
CAS:Dopamine stabilizerFórmula:C15H24ClNO2SPureza:98%Forma y color:SolidPeso molecular:317.88S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Fórmula:C21H24N2O2Pureza:98%Forma y color:SolidPeso molecular:336.43Etoperidone hydrochloride
CAS:Etoperidone hydrochloride is an antidepressant agent.Fórmula:C19H29Cl2N5OForma y color:SolidPeso molecular:414.37SLV-310
CAS:SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Fórmula:C25H24FN3O2Pureza:99.39%Forma y color:SolidPeso molecular:417.48Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Fórmula:C15H23Cl3N6Pureza:98%Forma y color:SolidPeso molecular:393.74Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Fórmula:C27H41ClN4O5Forma y color:SolidPeso molecular:537.09Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Fórmula:C19H25N3O2S2Forma y color:SolidPeso molecular:391.55Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Fórmula:C26H32N2O7Forma y color:SolidPeso molecular:484.549(R)-Viloxazine Hydrochloride
CAS:(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.Fórmula:C13H20ClNO3Pureza:99.88% - 99.94%Forma y color:SolidPeso molecular:273.76Ref: TM-T22413
1mg52,00€5mg111,00€10mg162,00€25mg235,00€50mg330,00€100mg452,00€200mg607,00€1mL*10mM (DMSO)101,00€LEK 8841
CAS:LEK 8841 is an ergoline derivative that is a potential antipsychotic.Fórmula:C21H24BrN3O4SPureza:98%Forma y color:SolidPeso molecular:494.4AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Fórmula:C20H18N2O3SForma y color:SolidPeso molecular:366.43Trimipramine
CAS:Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.Fórmula:C20H26N2Pureza:98%Forma y color:SolidPeso molecular:294.435-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Fórmula:C20H21ClN2O3Forma y color:SolidPeso molecular:372.85Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Fórmula:C17H26N4OPureza:98%Forma y color:SolidPeso molecular:302.41OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Fórmula:C23H29Cl2N3O2Pureza:99.60%Forma y color:SolidPeso molecular:450.4Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Fórmula:C26H31FN2O4Pureza:98%Forma y color:SolidPeso molecular:454.53
