
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 645 productos de "Receptor adrenérgico"
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Butanserin
CAS:<p>Butanserin is a 5-hydroxytryptamine S2-antagonist.</p>Fórmula:C24H26FN3O3Pureza:98%Forma y color:SolidPeso molecular:423.48Methyldopa hydrochloride
CAS:<p>L-(-)-α-Methyldopa HCl: alpha-adrenergic agonist, antihypertensive, inhibits DOPA decarboxylase.</p>Fórmula:C10H14ClNO4Pureza:98%Forma y color:SolidPeso molecular:247.68Afurolol Hydrochloride
CAS:<p>Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.</p>Fórmula:C15H22ClNO4Pureza:98.86%Forma y color:SolidPeso molecular:315.79Ulimorelin
CAS:<p>Ulimorelin, ghrelin receptor agonist (EC50: 29 nM, Ki: 16 nM), is a prokinetic and vasorelaxant via α1-adrenoceptor antagonism.</p>Fórmula:C30H39FN4O4Pureza:98%Forma y color:SolidPeso molecular:538.65Ronactolol
CAS:<p>Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.</p>Fórmula:C20H26N2O4Forma y color:SolidPeso molecular:358.43Levobetaxolol
CAS:<p>Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.</p>Fórmula:C18H29NO3Pureza:98%Forma y color:SolidPeso molecular:307.43Guanfacine
CAS:<p>Guanfacine is a selective agonist of the α2A receptor.</p>Fórmula:C9H9Cl2N3OPureza:98%Forma y color:SolidPeso molecular:246.09Arnolol
CAS:<p>Arnolol, a beta blocker, slows heart rate, reduces force of beats, lowers blood pressure, and enhances blood flow.</p>Fórmula:C14H23NO3Forma y color:SolidPeso molecular:253.34Lubabegron
CAS:<p>Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.</p>Fórmula:C29H29N3O3SForma y color:SolidPeso molecular:499.62Zolertine HCl
CAS:<p>Zolertine HCl is an antagonist of alpha-Adrenoceptor.</p>Fórmula:C13H19ClN6Pureza:98%Forma y color:SolidPeso molecular:294.78Cirazoline (free base)
CAS:<p>Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.</p>Fórmula:C13H16N2OForma y color:SolidPeso molecular:216.28ZD 7114 hydrochloride
CAS:<p>β3-adrenoceptor agonist</p>Fórmula:C22H31ClN2O6Pureza:98%Forma y color:SolidPeso molecular:454.94Protokylol
CAS:<p>Protokylol is a β-adrenergic receptor agonist.</p>Fórmula:C18H21NO5Pureza:98%Forma y color:SolidPeso molecular:331.36Metazosin
CAS:<p>Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.</p>Fórmula:C18H25N5O4Pureza:98%Forma y color:SolidPeso molecular:375.42Piribedil dihydrochloride
CAS:<p>dopamine agonist</p>Fórmula:C16H20Cl2N4O2Pureza:98%Forma y color:SolidPeso molecular:371.26Todralazine
CAS:<p>Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.</p>Fórmula:C11H12N4O2Pureza:98%Forma y color:SolidPeso molecular:232.24BFE-55
CAS:<p>BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors</p>Fórmula:C14H19NO3Pureza:98%Forma y color:SolidPeso molecular:249.31(RS)-Butyryltimolol
CAS:<p>(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.</p>Fórmula:C17H30N4O4SPureza:98%Forma y color:SolidPeso molecular:386.51L-Alprenolol
CAS:<p>L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.</p>Fórmula:C15H23NO2Pureza:98%Forma y color:SolidPeso molecular:249.35Centanafadine
CAS:<p>Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).</p>Fórmula:C15H15NPureza:98%Forma y color:SolidPeso molecular:209.29S(-)-Bisoprolol
CAS:<p>S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.</p>Fórmula:C18H31NO4Forma y color:SolidPeso molecular:325.44Spirendolol
CAS:<p>Spirendolol is an antagonist of β adrenergic receptor.</p>Fórmula:C21H31NO3Pureza:98%Forma y color:SolidPeso molecular:345.48Epinephrine bitartrate
CAS:<p>L-Epinephrine Bitartrate is alpha- and beta-adrenergic receptor stimulator.</p>Fórmula:C13H19NO9Pureza:98.6% - 99.07%Forma y color:White SolidPeso molecular:333.3Epanolol
CAS:<p>Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.</p>Fórmula:C20H23N3O4Pureza:98%Forma y color:SolidPeso molecular:369.41Adrenaline sulfate
CAS:<p>Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.</p>Fórmula:C9H15NO7SForma y color:SolidPeso molecular:281.279Broxaterol
CAS:<p>Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.</p>Fórmula:C9H15BrN2O2Pureza:98%Forma y color:SolidPeso molecular:263.13B-HT 933 dihydrochloride
CAS:<p>Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.</p>Fórmula:C9H17Cl2N3OForma y color:SolidPeso molecular:254.16Levobunolol
CAS:<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Fórmula:C17H25NO3Forma y color:White To Pink PowderPeso molecular:291.39Bufetolol
CAS:<p>Bufetolol is an antagonist of beta-adrenoceptor.</p>Fórmula:C18H29NO4Pureza:98%Forma y color:SolidPeso molecular:323.43Alprenolol tartrate, (S)-
CAS:<p>Alprenolol tartrate, (S)- is an 5-HT1A antagonist.</p>Fórmula:C19H29NO8Pureza:98%Forma y color:SolidPeso molecular:399.44Guanoxabenz hydrochloride
CAS:<p>Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.</p>Fórmula:C8H9Cl3N4OForma y color:SolidPeso molecular:283.54Methyldopate hydrochloride
CAS:<p>Methyldopate HCl is an agent of antihypertensive.</p>Fórmula:C12H18ClNO4Forma y color:SolidPeso molecular:275.73UK 1745
CAS:<p>UK 1745 is a novel drug of cardiotonic.</p>Fórmula:C16H23ClN2O2Forma y color:SolidPeso molecular:310.82Guanethidine
CAS:<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Fórmula:C10H22N4Forma y color:SolidPeso molecular:198.31A 55453
CAS:<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Fórmula:C25H32N6O3Forma y color:SolidPeso molecular:464.56RS 79948 hydrochloride
CAS:<p>α2-adrenoreceptor antagonist</p>Fórmula:C19H29ClN2O3SPureza:98%Forma y color:SolidPeso molecular:400.96MK761
CAS:<p>MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.</p>Fórmula:C13H19N3O2Forma y color:SolidPeso molecular:249.31Napamezole
CAS:<p>Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.</p>Fórmula:C14H16N2Pureza:98%Forma y color:SolidPeso molecular:212.29Flestolol sulfate
CAS:<p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>Fórmula:C15H24FN3O8SForma y color:SolidPeso molecular:425.43BMS-466442
CAS:<p>BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.</p>Fórmula:C31H30N4O5Forma y color:SolidPeso molecular:538.59Mabuterol hydrochloride
CAS:<p>Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.</p>Fórmula:C13H19Cl2F3N2OForma y color:SolidPeso molecular:347.20Arbutamine hydrochloride
CAS:<p>Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.</p>Fórmula:C18H24ClNO4Forma y color:SolidPeso molecular:353.84Fenmetozole
CAS:<p>Fenmetozole is an antagonist of the actions of ethanol.</p>Fórmula:C10H10Cl2N2OForma y color:SolidPeso molecular:245.11CP 59430
CAS:<p>CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.</p>Fórmula:C21H22N8O3Forma y color:SolidPeso molecular:434.45Clencyclohexerol
CAS:<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Fórmula:C14H20Cl2N2O2Forma y color:SolidPeso molecular:319.23Dapiprazole
CAS:<p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>Fórmula:C19H27N5Pureza:98%Forma y color:SolidPeso molecular:325.45BRL 37344 sodium
CAS:<p>BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.</p>Fórmula:C19H22ClNNaO4Pureza:98%Forma y color:SolidPeso molecular:386.83Pronethalol hydrochloride
CAS:<p>β-adrenergic antagonist</p>Fórmula:C15H20ClNOPureza:98%Forma y color:SolidPeso molecular:265.78Naminterol
CAS:<p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>Fórmula:C19H26N2O3Pureza:98%Forma y color:SolidPeso molecular:330.42Zenidolol
CAS:<p>Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.</p>Fórmula:C17H27NO2Forma y color:SolidPeso molecular:277.4ONO-2952
CAS:<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Fórmula:C22H20ClFN2O2Pureza:98%Forma y color:SolidPeso molecular:398.86(-)-S-Timolol
CAS:<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Fórmula:C13H26N4O4SForma y color:SolidPeso molecular:334.44Trimazosin
CAS:<p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>Fórmula:C20H29N5O6Forma y color:SolidPeso molecular:435.47Primidolol
CAS:<p>Primidolol is a beta adrenergic receptor antagonist and antihypertensive agent.</p>Fórmula:C17H23N3O4Pureza:98%Forma y color:SolidPeso molecular:333.38Oxyfedrine
CAS:<p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>Fórmula:C19H23NO3Forma y color:SolidPeso molecular:313.39Ko-3290
CAS:<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Fórmula:C19H25N3O3Pureza:98%Forma y color:SolidPeso molecular:343.42Imiloxan hydrochloride
CAS:<p>Imiloxan hydrochloride is an α2-adrenoceptor antagonist.</p>Fórmula:C14H17ClN2O2Pureza:98%Forma y color:SolidPeso molecular:280.75Metrenperone
CAS:<p>Metrenperone is used as a S(2)-receptor blocker.</p>Fórmula:C24H26FN3O2Pureza:98%Forma y color:SolidPeso molecular:407.48Zinterol hydrochloride
CAS:<p>Zinterol HCl is a selective β2-adrenoceptor agonist.</p>Fórmula:C19H27ClN2O4SForma y color:SolidPeso molecular:414.95Hexoprenaline
CAS:<p>Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.</p>Fórmula:C22H32N2O6Forma y color:SolidPeso molecular:420.5Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Fórmula:C17H18Cl2N2O4SPureza:98%Forma y color:SolidPeso molecular:417.31Agroclavine
CAS:<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Fórmula:C16H18N2Forma y color:SolidPeso molecular:238.33ADRA1D receptor antagonist 1 free base
CAS:<p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>Fórmula:C15H13ClN4OForma y color:SolidPeso molecular:300.74(E)-Guanabenz
CAS:<p>(E)-Guanabenz is an oral α2-adrenoceptor agonist, antihypertensive, GADD34 inhibitor, and has neuroprotective properties.</p>Fórmula:C8H8Cl2N4Forma y color:SolidPeso molecular:231.08Ro 363 hydrochloride
CAS:<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Fórmula:C19H26ClNO6Forma y color:SolidPeso molecular:399.87Pargolol hydrochloride
CAS:<p>Pargolol hydrochloride is an antagonist of β adrenergic receptor.</p>Fórmula:C16H24ClNO3Pureza:98%Forma y color:SolidPeso molecular:313.82Edivoxetine
CAS:<p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>Fórmula:C18H26FNO4Forma y color:SolidPeso molecular:339.4Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Fórmula:C20H24N2O5Forma y color:SolidPeso molecular:372.42Povafonidine
CAS:<p>Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.</p>Fórmula:C11H13N5Forma y color:SolidPeso molecular:215.25MG 1
CAS:<p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>Fórmula:C17H25N3O2Pureza:98.98% - >99.99%Forma y color:SolidPeso molecular:303.4ZK-90055 hydrochloride
CAS:<p>ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.</p>Fórmula:C16H23ClN2O4Pureza:99.26%Forma y color:SolidPeso molecular:342.82Thioproperazine
CAS:<p>Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.</p>Fórmula:C22H30N4O2S2Pureza:99.45%Forma y color:SolidPeso molecular:446.63Guanadrel
CAS:<p>Guanadrel is an antihypertensive agent.</p>Fórmula:C10H19N3O2Pureza:98%Forma y color:SolidPeso molecular:213.28(E)-Alprenoxime
CAS:<p>(E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.</p>Fórmula:C15H22N2O2Pureza:98%Forma y color:SolidPeso molecular:262.35Dexnafenodone Hydrochloride
CAS:<p>Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.</p>Fórmula:C20H24ClNOForma y color:SolidPeso molecular:329.86LY 87130
CAS:<p>LY 87130 is a phenylethanolamine-N-methyltransferase inhibitor.</p>Fórmula:C12H13NPureza:98%Forma y color:SolidPeso molecular:171.24Talsupram hydrochloride
CAS:<p>noradrenalin re-uptake inhibitor</p>Fórmula:C20H26ClNSPureza:98%Forma y color:SolidPeso molecular:347.95RS 52367
CAS:<p>RS 52367 is a beta-adrenergic antagonist.</p>Fórmula:C18H34ClN3O3SForma y color:SolidPeso molecular:408S 12024-2
CAS:<p>S 12024-2 (Dabelotine mesylate) is a new cognitive drug-enhancer.</p>Fórmula:C16H26N2O5SPureza:98%Forma y color:SolidPeso molecular:358.45Flerobuterol
CAS:<p>Flerobuterol is a potential antidepressant agent related to beta-adrenergic agonists.</p>Fórmula:C12H18FNOPureza:98%Forma y color:SolidPeso molecular:211.28Befunolol HCl
CAS:<p>Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.</p>Fórmula:C16H22ClNO4Forma y color:SolidPeso molecular:327.8Flutonidine
CAS:<p>Flutonidine is an agonist of alpha2-Adrenergic receptor.</p>Fórmula:C10H12FN3Pureza:98%Forma y color:SolidPeso molecular:193.22S-Nitroso-N-acetylcysteine
CAS:<p>S-Nitroso-N-acetylcysteine inhibits proliferation and survival of multiple MM cells. It acts by the S-nitrosylation-dependent inhibition of STAT3 and NF-κB.</p>Fórmula:C5H8N2O4SPureza:98%Forma y color:SolidPeso molecular:192.19Bremazocine
CAS:<p>Bremazocineis a potent opiate kappa-agonist and centrally acting analgesic.</p>Fórmula:C20H29NO2Pureza:98%Forma y color:SolidPeso molecular:315.45RS 15385-197
CAS:<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Fórmula:C18H26N2O3SForma y color:SolidPeso molecular:350.48Garomefrine HCl
CAS:<p>Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.</p>Fórmula:C9H14ClFN2O3SPureza:98%Forma y color:SolidPeso molecular:284.73Cafaminol
CAS:<p>Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.</p>Fórmula:C11H17N5O3Forma y color:SolidPeso molecular:267.28R 47243
CAS:<p>R 47243 is used as a racemic alpha 2 antagonist.</p>Fórmula:C22H25N3O2SPureza:98%Forma y color:SolidPeso molecular:395.52Burimamide
CAS:<p>Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.</p>Fórmula:C9H16N4SPureza:98%Forma y color:SolidPeso molecular:212.32BE 2254
CAS:<p>BE 2254 is an antagonist of central noradrenergic receptor.</p>Fórmula:C19H21NO2Forma y color:SolidPeso molecular:295.38Dabuzalgron HCl
CAS:<p>Dabuzalgron, an adrenoceptor agonist, is used potentially for the treatment of urinary incontinence.</p>Fórmula:C12H17Cl2N3O3SPureza:98%Forma y color:SolidPeso molecular:354.25Butidrine
CAS:<p>Butidrine has an Antiarrhythmic activities.</p>Fórmula:C16H25NOPureza:98%Forma y color:SolidPeso molecular:247.38Dipiproverine hydrochloride
CAS:<p>Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.</p>Fórmula:C20H32Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:403.39JTH-601 free base
CAS:<p>JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.</p>Fórmula:C24H35NO4Pureza:98%Forma y color:SolidPeso molecular:401.54JNJ-7925476 HCl
CAS:<p>JNJ-7925476 HCl inhibits DAT, NET, SERT; ED(50): DAT 2.4, NET 0.09, SERT 0.18 mg/kg in rats.</p>Fórmula:C20H20ClNForma y color:SolidPeso molecular:309.83L-748328
CAS:<p>L-748328 is a potent and selective antagonist of human beta(3)-adrenergic receptor.</p>Fórmula:C23H27N3O6S2Pureza:98%Forma y color:SolidPeso molecular:505.61SKF 86466 hydrochloride
CAS:<p>SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.</p>Fórmula:C11H15Cl2NPureza:98%Forma y color:SolidPeso molecular:232.15KUL-7211
CAS:<p>KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.</p>Fórmula:C19H23NO5Pureza:98%Forma y color:SolidPeso molecular:345.39Esprolol hydrochloride
CAS:<p>Esprolol is a β-adrenergic receptor antagonist.</p>Fórmula:C17H28ClNO4Pureza:98%Forma y color:SolidPeso molecular:345.86Dipiproverine
CAS:<p>Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.</p>Fórmula:C20H30N2O2Forma y color:SolidPeso molecular:330.46
