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Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Se han encontrado 645 productos de "Receptor adrenérgico"

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  • AG-825

    CAS:
    <p>AG-825(Tyrphostin C15) is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (Tyrphostin</p>
    Fórmula:C19H15N3O3S2
    Pureza:98.43%
    Forma y color:Yellow Solid
    Peso molecular:397.47
  • Esprolol

    CAS:
    <p>Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.</p>
    Fórmula:C17H27NO4
    Pureza:71.58% - 99.16%
    Forma y color:Soild
    Peso molecular:309.4
  • Bromchlorbuterol hydrochloride

    CAS:
    <p>Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.</p>
    Fórmula:C12H19BrCl2N2O
    Forma y color:Solid
    Peso molecular:358.1
  • MK-761 TFA


    <p>MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.</p>
    Fórmula:C15H20F3N3O4
    Forma y color:Solid
    Peso molecular:363.332
  • Vanilpyruvic acid

    CAS:
    <p>Vanillylpyruvic acid is a phenylpyruvic acid derivative applicable in biochemical experiments and drug synthesis research.</p>
    Fórmula:C10H10O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:210.18
  • 4-Hydroxypropranolol-d7 hydrochloride

    CAS:
    <p>Deuterium-labeled 4-Hydroxypropranolol HCl, a Propranolol metabolite that blocks β1/β2 receptors.</p>
    Fórmula:C16H22ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:318.85
  • Diacetolol D7

    CAS:
    <p>Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.</p>
    Fórmula:C16H24N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:315.42
  • Apraclonidine hydrochloride

    CAS:
    <p>Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.</p>
    Fórmula:C9H11Cl3N4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:281.57
  • Benoxathian hydrochloride

    CAS:
    <p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>
    Fórmula:C19H24ClNO4S
    Forma y color:Solid
    Peso molecular:397.91
  • Nadolol-d9

    CAS:
    <p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>
    Fórmula:C17H27NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:318.46
  • Clencyclohexerol-d10

    CAS:
    <p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>
    Fórmula:C14H20Cl2N2O2
    Forma y color:Solid
    Peso molecular:329.29
  • Zilpaterol-d7

    CAS:
    <p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>
    Fórmula:C14H12D7N3O2
    Forma y color:Solid
    Peso molecular:268.36
  • Cimbuterol-d9

    CAS:
    <p>Cimbuterol-d9 is a deuterated compound of Cimbuterol.</p>
    Fórmula:C13H10D9N3O
    Pureza:99.22%
    Forma y color:Solid
    Peso molecular:242.37
  • 4-Hydroxyatomoxetine D3

    CAS:
    <p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>
    Fórmula:C17H21NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:274.37
  • Naphazoline nitrate

    CAS:
    <p>Naphazoline nitrate: α1-adrenergic agonist, induces autophagy, necrosis in cancer cells, inhibits differentiation, treats congestion and eye issues.</p>
    Fórmula:C14H15N3O3
    Pureza:98%
    Forma y color:White Crystalline Powder White Solid
    Peso molecular:273.29
  • Piribedil D8

    CAS:
    <p>Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.</p>
    Fórmula:C16H18N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:306.39
  • rac-Propranolol-d7

    CAS:
    <p>Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.</p>
    Fórmula:C16H14D7NO2
    Forma y color:Solid
    Peso molecular:266.39
  • Ivabradine-d6 hydrochloride

    CAS:
    <p>Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.</p>
    Fórmula:C27H37ClN2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:511.08
  • (+)-Penbutolol

    CAS:
    <p>(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.</p>
    Fórmula:C18H29NO2
    Forma y color:Solid
    Peso molecular:291.43
  • Brombuterol hydrochloride

    CAS:
    <p>Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.</p>
    Fórmula:C12H19Br2ClN2O
    Forma y color:Solid
    Peso molecular:402.56