
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 645 productos de "Receptor adrenérgico"
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Fluparoxan HCl
CAS:<p>Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).</p>Fórmula:C10H11ClFNO2Forma y color:SolidPeso molecular:231.65Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Forma y color:White Or Almost White Crystalline PowderPeso molecular:236.74Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Forma y color:White SolidPeso molecular:238.24Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Fórmula:C19H23NO3·CH4O3SPureza:99.18% - 99.87%Forma y color:Tan Or Off-White Cyrstalline SolidPeso molecular:409.5Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Fórmula:C23H29NO5SPureza:98%Forma y color:SolidPeso molecular:431.55Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Fórmula:C14H22ClNO2Pureza:97.63%Forma y color:SolidPeso molecular:271.78Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Fórmula:C9H10Cl2N4Forma y color:SolidPeso molecular:245.11Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Forma y color:Appearance White Crystalline PowderPeso molecular:264.19Reboxetine
CAS:<p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>Fórmula:C19H23NO3Pureza:98%Forma y color:SolidPeso molecular:313.39Piribedil hydrochloride
CAS:<p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>Fórmula:C16H19ClN4O2Forma y color:SolidPeso molecular:334.8Solabegron HCl
CAS:<p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>Fórmula:C23H24Cl2N2O3Forma y color:SolidPeso molecular:447.35Guanabenz Acetate
CAS:<p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>Fórmula:C8H8Cl2N4·C2H4O2Pureza:99% - 99.66%Forma y color:White Solid From Acetonitrile White SolidPeso molecular:291.13L755507
CAS:<p>L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).</p>Fórmula:C30H40N4O6SPureza:99% - 99.75%Forma y color:SolidPeso molecular:584.73Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Forma y color:SolidPeso molecular:224.26Bunazosin
CAS:<p>Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].</p>Fórmula:C19H27N5O3Forma y color:SolidPeso molecular:373.45Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Forma y color:SolidPeso molecular:301.81Levalbuterol tartrate
CAS:<p>Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.</p>Fórmula:C17H27NO9Pureza:98.97% - 99.79%Forma y color:SolidPeso molecular:389.39Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Forma y color:White To Tan Powder SolidPeso molecular:383.4LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Forma y color:SolidPeso molecular:226.53Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Forma y color:SolidPeso molecular:240.69
