
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 651 productos de "Receptor adrenérgico"
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Efaroxan hydrochloride
CAS:<p>Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.</p>Fórmula:C13H17ClN2OPureza:98%Forma y color:SolidPeso molecular:252.74Protokylol hydrochloride
CAS:<p>Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.</p>Fórmula:C18H22ClNO5Forma y color:SolidPeso molecular:367.83Clonidine
CAS:<p>Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.</p>Fórmula:C9H9Cl2N3Pureza:99.42% - 99.44%Forma y color:Crystals SolidPeso molecular:230.09BRL 44408 Maleate Salt
CAS:<p>BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.</p>Fórmula:C17H21N3O4Pureza:98.71%Forma y color:SolidPeso molecular:331.37Butaxamine
CAS:<p>Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.</p>Fórmula:C15H25NO3Pureza:98%Forma y color:SolidPeso molecular:267.36Lusaperidone
CAS:Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.Fórmula:C22H21N3O2Pureza:99.75%Forma y color:SolidPeso molecular:359.42IMTPPE
CAS:<p>IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.</p>Fórmula:C20H27N3O2SForma y color:SolidPeso molecular:373.51Abanoquil
CAS:Abanoquil is an antagonist of alpha-1 adrenoceptor.Fórmula:C22H25N3O4Forma y color:SolidPeso molecular:395.45Zinterol
CAS:<p>Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).</p>Fórmula:C19H26N2O4SPureza:98%Forma y color:SolidPeso molecular:378.49Metoprolol fumarate
CAS:<p>Metoprolol fumarate (CGP 2175C): selective β1-blocker with anti-inflammatory, antitumor, anti-angiogenic effects.</p>Fórmula:C34H54N2O10Forma y color:SolidPeso molecular:650.8Clenproperol
CAS:<p>Clenproperol is a β2-adrenergic agonist.</p>Fórmula:C11H16Cl2N2OForma y color:SolidPeso molecular:263.16Isoetharine
CAS:<p>Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.</p>Fórmula:C13H21NO3Forma y color:SolidPeso molecular:239.31Denopamine
CAS:<p>Denopamine is an agonist of 1-Adrenoceptor.</p>Fórmula:C18H23NO4Forma y color:SolidPeso molecular:317.38HEAT hydrochloride
CAS:<p>HEAT hydrochloride is an α1-adrenoceptor antagonist.</p>Fórmula:C19H22ClNO2Pureza:98%Forma y color:SolidPeso molecular:331.845-Methylurapidil
CAS:<p>5-Methylurapidil is an alpha1A-adrenoceptor antagonist.</p>Fórmula:C21H31N5O3Pureza:98%Forma y color:SolidPeso molecular:401.5Tiamenidine
CAS:<p>Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.</p>Fórmula:C8H10ClN3SPureza:98%Forma y color:SolidPeso molecular:215.7RWJ 52353
CAS:<p>α2D adrenergic receptor agonist</p>Fórmula:C11H10N2SPureza:98%Forma y color:SolidPeso molecular:202.28Bucumarol (HCl)
CAS:<p>Bucumarol is a beta-adrenergic blocking agent.</p>Fórmula:C17H24ClNO4Forma y color:SolidPeso molecular:341.83Tiodazosin
CAS:<p>Tiodazosin is a competitive antagonist of the postsynaptic alpha-adrenergic receptor.</p>Fórmula:C18H21N7O4SPureza:98%Forma y color:SolidPeso molecular:431.47A 61603
CAS:<p>Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.</p>Fórmula:C14H20BrN3O3SForma y color:SolidPeso molecular:390.3
