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Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Se han encontrado 645 productos de "Receptor adrenérgico"

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  • Dihydroalprenolol, (S)-

    CAS:
    <p>Dihydroalprenolol, (S)- is a hydrogenated alprenolol derivative. It acts as a beta-adrenergic blocker.</p>
    Fórmula:C15H25NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:251.36
  • Levomoprolol

    CAS:
    <p>Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.</p>
    Fórmula:C13H21NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:239.31
  • L-771688 dihydrochloride

    CAS:
    <p>L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.</p>
    Fórmula:C28H35Cl2F2N5O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:630.51
  • Levoprotiline

    CAS:
    <p>Levoprotiline, a fast-acting antidepressant, is the R-enantiomer of Oxaprotiline and successor to maprotiline.</p>
    Fórmula:C20H23NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:293.4
  • SNAP 5089

    CAS:
    <p>α1A-adrenoceptor antagonist</p>
    Fórmula:C36H40N4O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:608.73
  • Dilevalol

    CAS:
    <p>Dilevalol, an RR-stereoisomer of labetalol, is a beta-blocker with partial beta 2-agonism and minimal alpha 1-blockade.</p>
    Fórmula:C19H24N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:328.41
  • Delequamine HCl

    CAS:
    <p>Delequamine HCl: potent, selective alpha 2-adrenoceptor blocker; pKi 9.45 in rat cortex, pA2 9.72 in guinea-pig ileum.</p>
    Fórmula:C18H27ClN2O3S
    Forma y color:Solid
    Peso molecular:386.94
  • Oxaprotiline

    CAS:
    <p>Oxaprotiline: an antidepressant, norepinephrine inhibitor, and H1 blocker; studied in hospital depression but not marketed.</p>
    Fórmula:C20H23NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:293.4
  • Zometapine

    CAS:
    <p>Zometapine (CI 716) is an antidepressant compound that is a derivative of pyrazole and diazepine.</p>
    Fórmula:C14H15ClN4
    Pureza:98.87%
    Forma y color:Solid
    Peso molecular:274.75
  • Levoprotiline hydrochloride

    CAS:
    <p>Levoprotiline hydrochloride is an antidepressant.</p>
    Fórmula:C20H24ClNO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:329.86
  • FMS586

    CAS:
    <p>FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.</p>
    Fórmula:C24H30N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:390.52
  • Tilisolol HCl

    CAS:
    <p>Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.</p>
    Fórmula:C17H25ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:340.85
  • (S)-Viloxazine Hydrochloride

    CAS:
    <p>(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.</p>
    Fórmula:C13H20ClNO3
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:273.76
  • Tranterol hydrochloride

    CAS:
    <p>Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.</p>
    Fórmula:C13H19Cl2F3N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:347.2
  • Pamatolol

    CAS:
    <p>Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.</p>
    Fórmula:C16H26N2O4
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:310.39
  • Cicloprolol hydrochloride

    CAS:
    <p>Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.</p>
    Fórmula:C18H30ClNO4
    Pureza:97.26%
    Forma y color:Solid
    Peso molecular:359.89
  • L-771688

    CAS:
    <p>L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign</p>
    Fórmula:C28H33F2N5O5
    Pureza:94.15%
    Forma y color:Solid
    Peso molecular:557.59
  • Indanidine

    CAS:
    <p>Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the</p>
    Fórmula:C11H13N5
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:215.25
  • TD-5471 hydrochloride

    CAS:
    <p>TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (</p>
    Fórmula:C32H32ClN3O4
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:558.07
  • Napitane

    CAS:
    <p>napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the</p>
    Fórmula:C22H25NO2
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:335.44