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Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Se han encontrado 645 productos de "Receptor adrenérgico"

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  • Benoxathian hydrochloride

    CAS:
    <p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>
    Fórmula:C19H24ClNO4S
    Forma y color:Solid
    Peso molecular:397.91
  • Zilpaterol-d7

    CAS:
    <p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>
    Fórmula:C14H12D7N3O2
    Forma y color:Solid
    Peso molecular:268.36
  • Clencyclohexerol-d10

    CAS:
    <p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>
    Fórmula:C14H20Cl2N2O2
    Forma y color:Solid
    Peso molecular:329.29
  • Doxazosin D8

    CAS:
    <p>Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.</p>
    Fórmula:C23H25N5O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:459.52
  • Propranolol-d7 hydrochloride

    CAS:
    <p>Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.</p>
    Fórmula:C16H22ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.85
  • Levosalbutamol Hydrochloride

    CAS:
    <p>Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.</p>
    Fórmula:C13H22ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:275.77
  • Cannabigerol

    CAS:
    <p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Forma y color:Solid
    Peso molecular:316.48
  • Phentolamine

    CAS:
    <p>Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist</p>
    Fórmula:C17H19N3O
    Pureza:99.86% - 99.94%
    Forma y color:Crystals Solid
    Peso molecular:281.35
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • ICI 89406

    CAS:
    <p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>
    Fórmula:C19H22N4O3
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:354.4
  • Olodaterol hydrochloride

    CAS:
    <p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>
    Fórmula:C21H27ClN2O5
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:422.9
  • Indacaterol

    CAS:
    <p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>
    Fórmula:C24H28N2O3
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:392.49
  • LUN42518 HCl 47142-51-8(free base)


    <p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>
    Fórmula:C17H20ClN3O
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:317.81
  • Carbazochrome

    CAS:
    <p>Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.</p>
    Fórmula:C10H12N4O3
    Pureza:98.36%
    Forma y color:Nacarat Crystalline Powder
    Peso molecular:236.23
  • Detomidine hydrochloride

    CAS:
    <p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>
    Fórmula:C12H14N2·HCl
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:222.71
  • Phosphorylcholine chloride

    CAS:
    <p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>
    Fórmula:C5H15ClNO4P
    Pureza:99.481% - 99.85%
    Forma y color:Solid
    Peso molecular:219.6
  • Nomifensine

    CAS:
    <p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:238.33
  • Eformoterol Hemifumarate

    CAS:
    <p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>
    Fórmula:C19H24N2O4C4H4O4
    Pureza:99.86% - >99.99%
    Forma y color:White Powder
    Peso molecular:402.4
  • Phentolamine hydrochloride

    CAS:
    <p>Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].</p>
    Fórmula:C17H20ClN3O
    Forma y color:Solid
    Peso molecular:317.82
  • Bevantolol

    CAS:
    <p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>
    Fórmula:C20H27NO4
    Forma y color:Solid
    Peso molecular:345.43
  • Yohimbine hydrochloride

    CAS:
    <p>Yohimbine hydrochloride (Antagonil) is a plant alkaloid with α-2-adrenergic blocking activity, used as a mydriatic and in the treatment of erectile dysfunction</p>
    Fórmula:C21H27ClN2O3
    Pureza:99.86% - >99.99%
    Forma y color:Very Slightly Yellow Needles
    Peso molecular:390.90
  • Clebopride malate

    CAS:
    <p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>
    Fórmula:C24H30ClN3O7
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:507.96
  • Romifidine hydrochloride

    CAS:
    <p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>
    Fórmula:C9H10BrClFN3
    Forma y color:Solid
    Peso molecular:294.55
  • Landiolol hydrochloride

    CAS:
    <p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>
    Fórmula:C25H40ClN3O8
    Pureza:99.91%
    Forma y color:White Crystalline Powder
    Peso molecular:546.05
  • Dronedarone

    CAS:
    <p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>
    Fórmula:C31H44N2O5S
    Pureza:98.85% - 99.58%
    Forma y color:Solid
    Peso molecular:556.76
  • Reboxetine

    CAS:
    <p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>
    Fórmula:C19H23NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:313.39
  • Bupranolol

    CAS:
    <p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>
    Fórmula:C14H22ClNO2
    Pureza:97.63%
    Forma y color:Solid
    Peso molecular:271.78
  • Parethoxycaine hydrochloride

    CAS:
    <p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>
    Fórmula:C15H24ClNO3
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:301.81
  • Atipamezole hydrochloride

    CAS:
    <p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>
    Fórmula:C14H16N2·HCl
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:248.75
  • Midaglizole

    CAS:
    <p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>
    Fórmula:C16H17N3
    Forma y color:Solid
    Peso molecular:251.33
  • Droxidopa hydrochloride

    CAS:
    <p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>
    Fórmula:C9H12ClNO5
    Forma y color:Solid
    Peso molecular:249.65
  • Synephrine hydrochloride

    CAS:
    <p>Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).</p>
    Fórmula:C9H14ClNO2
    Pureza:98.16% - 99.73%
    Forma y color:White Fine Powder
    Peso molecular:203.666
  • Arformoterol Tartrate

    CAS:
    <p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>
    Fórmula:C23H30N2O10
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:494.49
  • Brefonalol

    CAS:
    <p>Brefonalol is a vasodilating beta-adrenergic receptor blocker.</p>
    Fórmula:C22H28N2O2
    Forma y color:Solid
    Peso molecular:352.47
  • Solabegron HCl

    CAS:
    <p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>
    Fórmula:C23H24Cl2N2O3
    Forma y color:Solid
    Peso molecular:447.35
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Fórmula:C22H33Cl2N3O3
    Pureza:97.32% - 99.08%
    Forma y color:Solid
    Peso molecular:458.42
  • LY 78335

    CAS:
    <p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>
    Fórmula:C8H10Cl3N
    Pureza:99.30% - 99.81%
    Forma y color:Solid
    Peso molecular:226.53
  • Lofexidine

    CAS:
    <p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>
    Fórmula:C11H12Cl2N2O
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:259.13
  • Dobutamine

    CAS:
    <p>Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.</p>
    Fórmula:C18H23NO3
    Forma y color:Solid
    Peso molecular:301.38
  • Naftopidil hydrochloride

    CAS:
    <p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>
    Fórmula:C24H29ClN2O3
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:428.95
  • Rilmenidine hemifumarate

    CAS:
    <p>Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.</p>
    Fórmula:C10H16N2OC4H4O4
    Pureza:98.14%
    Forma y color:Solid
    Peso molecular:238.28
  • Norepinephrine

    CAS:
    <p>Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.</p>
    Fórmula:C8H11NO3
    Pureza:99.43% - 99.84%
    Forma y color:Colorless Microcrystals Solid
    Peso molecular:169.18
  • Fipamezole HCl

    CAS:
    <p>Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.</p>
    Fórmula:C14H16ClFN2
    Forma y color:Solid
    Peso molecular:266.74
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:477.57
  • Piribedil hydrochloride

    CAS:
    <p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>
    Fórmula:C16H19ClN4O2
    Forma y color:Solid
    Peso molecular:334.8
  • ACTH 1-14 acetate(25696-21-3 free base)


    <p>ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.</p>
    Fórmula:C79H113N21O22S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1740.96
  • Zotepine

    CAS:
    <p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>
    Fórmula:C18H18ClNOS
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:331.86
  • Dobutamine tartrate

    CAS:
    <p>Dobutamine tartrate is a cardiotonic.</p>
    Fórmula:C22H29NO9
    Forma y color:Solid
    Peso molecular:451.472
  • Norepinephrine bitartrate salt

    CAS:
    <p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>
    Fórmula:C12H17NO9
    Pureza:97.32% - 99.97%
    Forma y color:Solid
    Peso molecular:319.27
  • Rilmenidine Phosphate

    CAS:
    <p>Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.</p>
    Fórmula:C10H19N2O5P
    Pureza:99.87% - ≥95%
    Forma y color:Solid
    Peso molecular:278.24