
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 645 productos de "Receptor adrenérgico"
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Benoxathian hydrochloride
CAS:<p>Benoxathian hydrochloride is effective α 1 Adrenaline receptor antagonist. Benoxathian hydrochloride has value in the study of anorexia.</p>Fórmula:C19H24ClNO4SForma y color:SolidPeso molecular:397.91Zilpaterol-d7
CAS:<p>Zilpaterol-d7 (trans-(±)-Zilpaterol-d7) is a deuterium-labeled version of Zilpaterol, a β-adrenergic receptor agonist.</p>Fórmula:C14H12D7N3O2Forma y color:SolidPeso molecular:268.36Clencyclohexerol-d10
CAS:<p>Argipressin inhibits central corticotropin-releasing hormone. Argipressin acts as an inhibitory factor in the regulation of central CRH levels.</p>Fórmula:C14H20Cl2N2O2Forma y color:SolidPeso molecular:329.29Doxazosin D8
CAS:<p>Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.</p>Fórmula:C23H25N5O5Pureza:98%Forma y color:SolidPeso molecular:459.52Propranolol-d7 hydrochloride
CAS:<p>Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.</p>Fórmula:C16H22ClNO2Pureza:98%Forma y color:SolidPeso molecular:302.85Levosalbutamol Hydrochloride
CAS:<p>Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.</p>Fórmula:C13H22ClNO3Pureza:98%Forma y color:SolidPeso molecular:275.77Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Fórmula:C21H32O2Pureza:99.59% - 99.92%Forma y color:SolidPeso molecular:316.48Phentolamine
CAS:<p>Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist</p>Fórmula:C17H19N3OPureza:99.86% - 99.94%Forma y color:Crystals SolidPeso molecular:281.35Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Forma y color:Off-White To Pale Yellow SolidPeso molecular:440.94ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Fórmula:C19H22N4O3Pureza:99.92%Forma y color:SolidPeso molecular:354.4Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Fórmula:C21H27ClN2O5Pureza:99.11%Forma y color:SolidPeso molecular:422.9Indacaterol
CAS:<p>Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.</p>Fórmula:C24H28N2O3Pureza:99.96%Forma y color:SolidPeso molecular:392.49LUN42518 HCl 47142-51-8(free base)
<p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>Fórmula:C17H20ClN3OPureza:99.96%Forma y color:SolidPeso molecular:317.81Carbazochrome
CAS:<p>Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.</p>Fórmula:C10H12N4O3Pureza:98.36%Forma y color:Nacarat Crystalline PowderPeso molecular:236.23Detomidine hydrochloride
CAS:<p>Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.</p>Fórmula:C12H14N2·HClPureza:99.97%Forma y color:SolidPeso molecular:222.71Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Fórmula:C5H15ClNO4PPureza:99.481% - 99.85%Forma y color:SolidPeso molecular:219.6Nomifensine
CAS:<p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Eformoterol Hemifumarate
CAS:<p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>Fórmula:C19H24N2O4C4H4O4Pureza:99.86% - >99.99%Forma y color:White PowderPeso molecular:402.4Phentolamine hydrochloride
CAS:<p>Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].</p>Fórmula:C17H20ClN3OForma y color:SolidPeso molecular:317.82Bevantolol
CAS:<p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>Fórmula:C20H27NO4Forma y color:SolidPeso molecular:345.43Yohimbine hydrochloride
CAS:<p>Yohimbine hydrochloride (Antagonil) is a plant alkaloid with α-2-adrenergic blocking activity, used as a mydriatic and in the treatment of erectile dysfunction</p>Fórmula:C21H27ClN2O3Pureza:99.86% - >99.99%Forma y color:Very Slightly Yellow NeedlesPeso molecular:390.90Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Romifidine hydrochloride
CAS:<p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>Fórmula:C9H10BrClFN3Forma y color:SolidPeso molecular:294.55Landiolol hydrochloride
CAS:<p>Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.</p>Fórmula:C25H40ClN3O8Pureza:99.91%Forma y color:White Crystalline PowderPeso molecular:546.05Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Fórmula:C31H44N2O5SPureza:98.85% - 99.58%Forma y color:SolidPeso molecular:556.76Reboxetine
CAS:<p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>Fórmula:C19H23NO3Pureza:98%Forma y color:SolidPeso molecular:313.39Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Fórmula:C14H22ClNO2Pureza:97.63%Forma y color:SolidPeso molecular:271.78Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Forma y color:SolidPeso molecular:301.81Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Fórmula:C14H16N2·HClPureza:99.74%Forma y color:SolidPeso molecular:248.75Midaglizole
CAS:<p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>Fórmula:C16H17N3Forma y color:SolidPeso molecular:251.33Droxidopa hydrochloride
CAS:<p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>Fórmula:C9H12ClNO5Forma y color:SolidPeso molecular:249.65Synephrine hydrochloride
CAS:<p>Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).</p>Fórmula:C9H14ClNO2Pureza:98.16% - 99.73%Forma y color:White Fine PowderPeso molecular:203.666Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Fórmula:C23H30N2O10Pureza:99.98%Forma y color:SolidPeso molecular:494.49Brefonalol
CAS:<p>Brefonalol is a vasodilating beta-adrenergic receptor blocker.</p>Fórmula:C22H28N2O2Forma y color:SolidPeso molecular:352.47Solabegron HCl
CAS:<p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>Fórmula:C23H24Cl2N2O3Forma y color:SolidPeso molecular:447.35BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Fórmula:C22H33Cl2N3O3Pureza:97.32% - 99.08%Forma y color:SolidPeso molecular:458.42LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Forma y color:SolidPeso molecular:226.53Lofexidine
CAS:<p>Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.</p>Fórmula:C11H12Cl2N2OPureza:98.78%Forma y color:SolidPeso molecular:259.13Dobutamine
CAS:<p>Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.</p>Fórmula:C18H23NO3Forma y color:SolidPeso molecular:301.38Naftopidil hydrochloride
CAS:<p>Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.</p>Fórmula:C24H29ClN2O3Pureza:99.5%Forma y color:SolidPeso molecular:428.95Rilmenidine hemifumarate
CAS:<p>Rilmenidine hemifumarate (S-3341 hemifumarate) is an I1 imidazoline receptor and α2-adrenergic receptor agonist that induces autophagy.</p>Fórmula:C10H16N2OC4H4O4Pureza:98.14%Forma y color:SolidPeso molecular:238.28Norepinephrine
CAS:<p>Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.</p>Fórmula:C8H11NO3Pureza:99.43% - 99.84%Forma y color:Colorless Microcrystals SolidPeso molecular:169.18Fipamezole HCl
CAS:<p>Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.</p>Fórmula:C14H16ClFN2Forma y color:SolidPeso molecular:266.74Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Forma y color:SolidPeso molecular:477.57Piribedil hydrochloride
CAS:<p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>Fórmula:C16H19ClN4O2Forma y color:SolidPeso molecular:334.8ACTH 1-14 acetate(25696-21-3 free base)
<p>ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.</p>Fórmula:C79H113N21O22SPureza:>99.99%Forma y color:SolidPeso molecular:1740.96Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86Dobutamine tartrate
CAS:<p>Dobutamine tartrate is a cardiotonic.</p>Fórmula:C22H29NO9Forma y color:SolidPeso molecular:451.472Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Fórmula:C12H17NO9Pureza:97.32% - 99.97%Forma y color:SolidPeso molecular:319.27Rilmenidine Phosphate
CAS:<p>Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.</p>Fórmula:C10H19N2O5PPureza:99.87% - ≥95%Forma y color:SolidPeso molecular:278.24
