
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 645 productos de "Receptor adrenérgico"
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Bevantolol hydrochloride
CAS:<p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>Fórmula:C20H28ClNO4Pureza:99.49%Forma y color:SolidPeso molecular:381.9ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Fórmula:C19H22N4O3Pureza:99.92%Forma y color:SolidPeso molecular:354.4Dobutamine tartrate
CAS:<p>Dobutamine tartrate is a cardiotonic.</p>Fórmula:C22H29NO9Forma y color:SolidPeso molecular:451.472Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Fórmula:C12H17NO9Pureza:97.32% - 99.97%Forma y color:SolidPeso molecular:319.27LUN42518 HCl 47142-51-8(free base)
<p>LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.</p>Fórmula:C17H20ClN3OPureza:99.96%Forma y color:SolidPeso molecular:317.81Paroxetine
CAS:<p>Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.</p>Fórmula:C19H20FNO3Pureza:98.89% - 99.45%Forma y color:White To Off-White PowderPeso molecular:329.37Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Fórmula:C20H29N5O3Pureza:99.85% - >99.99%Forma y color:SolidPeso molecular:387.48Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Forma y color:SolidPeso molecular:433.57Rauwolscine hydrochloride
CAS:<p>Rauwolscine HCl, a natural α2-adrenergic antagonist (Ki: 12 nM) & weak 5-HT1A agonist, also blocks 5-HT2B (Ki: 14.3 nM), affects mood/behavior.</p>Fórmula:C21H27ClN2O3Pureza:99.86% - 99.95%Forma y color:White SolidPeso molecular:390.9Piperoxan hydrochloride
CAS:<p>Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.</p>Fórmula:C14H20ClNO2Pureza:99.61%Forma y color:SolidPeso molecular:269.77Harmane
CAS:<p>Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.</p>Fórmula:C12H10N2Pureza:97.89% - >99.99%Forma y color:Off-White SolidPeso molecular:182.22Procaterol hydrochloride hydrate
CAS:<p>Short-acting β2-adrenergic receptor agonist used to treat asthma.</p>Fórmula:C32H48Cl2N4O7Pureza:99.71% - 99.97%Forma y color:SolidPeso molecular:671.65Phentolamine
CAS:<p>Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist</p>Fórmula:C17H19N3OPureza:99.86% - 99.94%Forma y color:Crystals SolidPeso molecular:281.35Levobetaxolol hydrochloride
CAS:<p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>Fórmula:C18H29NO3·HClPureza:98.80% - 99.69%Forma y color:SolidPeso molecular:343.89Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Forma y color:SolidPeso molecular:477.57Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Fórmula:C21H32O2Pureza:99.59% - 99.92%Forma y color:SolidPeso molecular:316.48Olodaterol hydrochloride
CAS:<p>Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect by binding and activating β2-AR.</p>Fórmula:C21H27ClN2O5Pureza:99.11%Forma y color:SolidPeso molecular:422.9Terazosin
CAS:<p>Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.</p>Fórmula:C19H25N5O4Forma y color:SolidPeso molecular:387.43Droxidopa
CAS:<p>Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.</p>Fórmula:C9H11NO5Pureza:97.27% - 99.88%Forma y color:SolidPeso molecular:213.19Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Fórmula:C36H45NO7Pureza:98% - 98.24%Forma y color:White SolidPeso molecular:603.75Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Fórmula:C5H15ClNO4PPureza:99.481% - 99.85%Forma y color:SolidPeso molecular:219.6Higenamine hydrochloride
CAS:<p>Higenamine HCl is a β2 adrenoreceptor agonist active in fat and muscle tissue.</p>Fórmula:C16H18ClNO3Pureza:99.44% - 99.80%Forma y color:White PowderPeso molecular:307.772Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Forma y color:White SolidPeso molecular:506.47Amezinium methylsulfate
CAS:<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Fórmula:C12H15N3O5SPureza:99.64%Forma y color:SolidPeso molecular:313.33Nomifensine
CAS:<p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Talinolol
CAS:<p>(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.</p>Fórmula:C20H33N3O3Pureza:98.8%Forma y color:SolidPeso molecular:363.49Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Fórmula:C21H25NO4Pureza:99.42% - 99.56%Forma y color:SolidPeso molecular:355.43Vilanterol trifenatate
CAS:<p>Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)</p>Fórmula:C44H49Cl2NO7Pureza:99.51% - >99.99%Forma y color:SolidPeso molecular:774.77Salbutamol hemisulfate
CAS:<p>Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.</p>Fórmula:C13H21NO3H2O4SPureza:99.35%Forma y color:White Or Almost White Odourless PowderPeso molecular:576.70Fluparoxan HCl
CAS:<p>Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).</p>Fórmula:C10H11ClFNO2Forma y color:SolidPeso molecular:231.65Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Forma y color:White Or Almost White Crystalline PowderPeso molecular:236.74Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Fórmula:C10H13NO4H2OPureza:99.67%Forma y color:White SolidPeso molecular:238.24Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Fórmula:C19H23NO3·CH4O3SPureza:99.18% - 99.87%Forma y color:Tan Or Off-White Cyrstalline SolidPeso molecular:409.5Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Fórmula:C23H29NO5SPureza:98%Forma y color:SolidPeso molecular:431.55Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Fórmula:C14H22ClNO2Pureza:97.63%Forma y color:SolidPeso molecular:271.78Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Fórmula:C9H10Cl2N4Forma y color:SolidPeso molecular:245.11Tulobuterol hydrochloride
CAS:<p>Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.</p>Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Forma y color:Appearance White Crystalline PowderPeso molecular:264.19Reboxetine
CAS:<p>Reboxetine (Norebox) is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD.</p>Fórmula:C19H23NO3Pureza:98%Forma y color:SolidPeso molecular:313.39Piribedil hydrochloride
CAS:<p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>Fórmula:C16H19ClN4O2Forma y color:SolidPeso molecular:334.8Solabegron HCl
CAS:<p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>Fórmula:C23H24Cl2N2O3Forma y color:SolidPeso molecular:447.35Guanabenz Acetate
CAS:<p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>Fórmula:C8H8Cl2N4·C2H4O2Pureza:99% - 99.66%Forma y color:White Solid From Acetonitrile White SolidPeso molecular:291.13L755507
CAS:<p>L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).</p>Fórmula:C30H40N4O6SPureza:99% - 99.75%Forma y color:SolidPeso molecular:584.73Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Fórmula:C11H16N2O3Pureza:98%Forma y color:SolidPeso molecular:224.26Bunazosin
CAS:<p>Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].</p>Fórmula:C19H27N5O3Forma y color:SolidPeso molecular:373.45Parethoxycaine hydrochloride
CAS:<p>Parethoxycaine hydrochloride (2-(diethylamino)ethyl 4-ethoxybenzoate hydrochloride) is an anesthetic[1].</p>Fórmula:C15H24ClNO3Pureza:99.46%Forma y color:SolidPeso molecular:301.81Levalbuterol tartrate
CAS:<p>Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.</p>Fórmula:C17H27NO9Pureza:98.97% - 99.79%Forma y color:SolidPeso molecular:389.39Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Fórmula:C19H21N5O4Pureza:99.86%Forma y color:White To Tan Powder SolidPeso molecular:383.4LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Fórmula:C8H10Cl3NPureza:99.30% - 99.81%Forma y color:SolidPeso molecular:226.53Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Forma y color:SolidPeso molecular:240.69
