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Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Se han encontrado 645 productos de "Receptor adrenérgico"

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  • Romifidine hydrochloride

    CAS:
    <p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>
    Fórmula:C9H10BrClFN3
    Forma y color:Solid
    Peso molecular:294.55
  • Norepinephrine bitartrate salt

    CAS:
    <p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>
    Fórmula:C12H17NO9
    Pureza:97.32% - 99.97%
    Forma y color:Solid
    Peso molecular:319.27
  • Norepinephrine

    CAS:
    <p>Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.</p>
    Fórmula:C8H11NO3
    Pureza:99.43% - 99.84%
    Forma y color:Colorless Microcrystals Solid
    Peso molecular:169.18
  • Bunazosin

    CAS:
    <p>Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].</p>
    Fórmula:C19H27N5O3
    Forma y color:Solid
    Peso molecular:373.45
  • Nifenalol

    CAS:
    <p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>
    Fórmula:C11H16N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:224.26
  • Reboxetine mesylate

    CAS:
    <p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>
    Fórmula:C19H23NO3·CH4O3S
    Pureza:99.18% - 99.87%
    Forma y color:Tan Or Off-White Cyrstalline Solid
    Peso molecular:409.5
  • Piribedil hydrochloride

    CAS:
    <p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>
    Fórmula:C16H19ClN4O2
    Forma y color:Solid
    Peso molecular:334.8
  • Apraclonidine

    CAS:
    <p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>
    Fórmula:C9H10Cl2N4
    Forma y color:Solid
    Peso molecular:245.11
  • Napitane Mesylate

    CAS:
    <p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>
    Fórmula:C23H29NO5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:431.55
  • Xamoterol

    CAS:
    <p>Xamoterol is a cardiac stimulant.</p>
    Fórmula:C16H25N3O5
    Forma y color:Solid
    Peso molecular:339.39
  • Methyldopa hydrate

    CAS:
    <p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>
    Fórmula:C10H13NO4H2O
    Pureza:99.67%
    Forma y color:White Solid
    Peso molecular:238.24
  • Pimozide

    CAS:
    <p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>
    Fórmula:C28H29F2N3O
    Pureza:99.63% - >99.99%
    Forma y color:Solid
    Peso molecular:461.55
  • Desipramine

    CAS:
    <p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>
    Fórmula:C18H22N2
    Forma y color:Solid
    Peso molecular:266.38
  • Medetomidine hydrochloride

    CAS:
    <p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>
    Fórmula:C13H16N2·HCl
    Pureza:99.96%
    Forma y color:White Or Off White Crystalline Powder
    Peso molecular:236.74
  • Scopine

    CAS:
    <p>Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.</p>
    Fórmula:C8H13NO2
    Pureza:99.79% - >99.99%
    Forma y color:Solid
    Peso molecular:155.19
  • Bevantolol

    CAS:
    <p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>
    Fórmula:C20H27NO4
    Forma y color:Solid
    Peso molecular:345.43
  • Eformoterol Hemifumarate

    CAS:
    <p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>
    Fórmula:C19H24N2O4C4H4O4
    Pureza:99.86% - >99.99%
    Forma y color:White Powder
    Peso molecular:402.4
  • Dexmedetomidine

    CAS:
    <p>Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.</p>
    Fórmula:C13H16N2
    Pureza:99% - >99.99%
    Forma y color:Solid
    Peso molecular:200.28
  • nifenalol.HCl

    CAS:
    <p>Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.</p>
    Fórmula:C11H17ClN2O3
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:260.72
  • Phenylephrine

    CAS:
    <p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>
    Fórmula:C9H13NO2
    Pureza:99.5% - 99.89%
    Forma y color:Solid
    Peso molecular:167.21
  • Talinolol

    CAS:
    <p>(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.</p>
    Fórmula:C20H33N3O3
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:363.49
  • Isoetharine mesylate salt

    CAS:
    <p>Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.</p>
    Fórmula:C14H25NO6S
    Pureza:99.35% - 99.75%
    Forma y color:Solid
    Peso molecular:335.42
  • Betaxolol

    CAS:
    <p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>
    Fórmula:C18H29NO3
    Pureza:99.01%
    Forma y color:White Crystalline Solid
    Peso molecular:307.43
  • Droxidopa

    CAS:
    <p>Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.</p>
    Fórmula:C9H11NO5
    Pureza:97.27% - 99.88%
    Forma y color:Solid
    Peso molecular:213.19
  • Higenamine hydrochloride

    CAS:
    <p>Higenamine HCl is a β2 adrenoreceptor agonist active in fat and muscle tissue.</p>
    Fórmula:C16H18ClNO3
    Pureza:99.44% - 99.80%
    Forma y color:White Powder
    Peso molecular:307.772
  • Amezinium methylsulfate

    CAS:
    <p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>
    Fórmula:C12H15N3O5S
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:313.33
  • Levobetaxolol hydrochloride

    CAS:
    <p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>
    Fórmula:C18H29NO3·HCl
    Pureza:98.80% - 99.69%
    Forma y color:Solid
    Peso molecular:343.89
  • Meranzin

    CAS:
    <p>Meranzin, a bioactive from TCM CSS, targets alpha 2-adrenoceptor, affects AMPA-ERK1/2–BDNF pathway, and may prevent atherosclerosis and depression.</p>
    Fórmula:C15H16O4
    Pureza:95.08% - 99.3%
    Forma y color:Solid
    Peso molecular:260.29
  • (R)-Propranolol hydrochloride

    CAS:
    <p>(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.</p>
    Fórmula:C16H22ClNO2
    Pureza:98.63% - 99.01%
    Forma y color:Solid
    Peso molecular:295.8
  • Medetomidine

    CAS:
    <p>Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.</p>
    Fórmula:C13H16N2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:200.28
  • CGP 20712 A

    CAS:
    <p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>
    Fórmula:C24H29F3N4O8S
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:590.57
  • Tamsulosin

    CAS:
    <p>Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.</p>
    Fórmula:C20H28N2O5S
    Pureza:99.93%
    Forma y color:White Crystals
    Peso molecular:408.51
  • Atipamezole

    CAS:
    <p>Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.</p>
    Fórmula:C14H16N2
    Pureza:99.88%
    Forma y color:Off-White To Light Yellow Crystal Powder
    Peso molecular:212.29
  • Alfuzosin

    CAS:
    <p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>
    Fórmula:C19H27N5O4
    Pureza:99.64%
    Forma y color:White Crystaline Powder
    Peso molecular:389.45
  • Bucindolol

    CAS:
    <p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>
    Fórmula:C22H25N3O2
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:363.45
  • Latrepirdine dihydrochloride

    CAS:
    <p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>
    Fórmula:C21H25N3·2HCl
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:392.37
  • Fenoterol hydrobromide

    CAS:
    <p>Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.</p>
    Fórmula:C17H22BrNO4
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:384.27
  • SR59230A hydrochloride

    CAS:
    <p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>
    Fórmula:C21H28ClNO2
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:361.91
  • DL-Phenylephrine HCl

    CAS:
    <p>DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.</p>
    Fórmula:C9H14ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:203.67
  • Tulobuterol

    CAS:
    <p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>
    Fórmula:C12H18ClNO
    Forma y color:Crystalline Solid
    Peso molecular:227.73
  • PF-610355

    CAS:
    <p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>
    Fórmula:C34H39N3O6S
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:617.76
  • Buflomedil

    CAS:
    <p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>
    Fórmula:C17H25NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:307.38
  • Pardoprunox

    CAS:
    <p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>
    Fórmula:C12H15N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:233.27
  • Penbutolol sulfate

    CAS:
    <p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>
    Fórmula:C18H29NO2H2O4S
    Pureza:98.55%
    Forma y color:Solid
    Peso molecular:340.47
  • Esmolol hydrochloride

    CAS:
    <p>Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension.</p>
    Fórmula:C16H25NO4·HCl
    Pureza:98.72% - 99.48%
    Forma y color:White Solid
    Peso molecular:331.15
  • Norreticuline

    CAS:
    <p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>
    Fórmula:C18H21NO4
    Forma y color:Solid
    Peso molecular:315.36
  • Isoproterenol sulfate anhydrous

    CAS:
    <p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>
    Fórmula:C22H36N2O10S
    Pureza:98%
    Forma y color:Coa
    Peso molecular:520.59
  • Ridazolol HCl

    CAS:
    <p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>
    Fórmula:C15H19Cl3N4O3
    Pureza:99.48%
    Forma y color:Soild
    Peso molecular:409.7
  • (RS)-ICI-118551 Hydrochloride

    CAS:
    <p>ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3</p>
    Fórmula:C17H27NO2·HCl
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:313.86
  • Atenolol Hydrochloride

    CAS:
    <p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>
    Fórmula:C14H23ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.80