
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 729 productos de "Receptor adrenérgico"
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Glaucine
CAS:Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.
Fórmula:C21H25NO4Pureza:99.42% - 99.56%Forma y color:SolidPeso molecular:355.43Salbutamol hemisulfate
CAS:Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.Fórmula:C13H21NO3H2O4SPureza:99.35%Forma y color:White Or Almost White Odourless PowderPeso molecular:576.70Desipramine
CAS:Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.Fórmula:C18H22N2Forma y color:SolidPeso molecular:266.38Vilanterol trifenatate
CAS:Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)Fórmula:C44H49Cl2NO7Pureza:99.51% - >99.99%Forma y color:SolidPeso molecular:774.77Scopine
CAS:Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.Fórmula:C8H13NO2Pureza:99.79% - >99.99%Forma y color:SolidPeso molecular:155.19Ref: TM-T6662
5mg47,00€10mg71,00€25mg108,00€50mg166,00€100mg280,00€200mg419,00€500mg672,00€1mL*10mM (DMSO)50,00€Fluparoxan HCl
CAS:Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).Fórmula:C10H11ClFNO2Forma y color:SolidPeso molecular:231.65Dexmedetomidine hydrochloride
CAS:Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Fórmula:C13H16N2·HClPureza:99.94% - 99.94%Forma y color:White Or Almost White Crystalline PowderPeso molecular:236.74Ref: TM-T6466
5mg42,00€10mg55,00€25mg88,00€50mg159,00€100mg226,00€200mg340,00€500mg563,00€1mL*10mM (DMSO)50,00€Phosphorylcholine chloride
CAS:Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integralFórmula:C5H15ClNO4PPureza:99.481% - 99.85%Forma y color:SolidPeso molecular:219.6Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Fórmula:C28H29F2N3OPureza:99.63% - >99.99%Forma y color:SolidPeso molecular:461.55Idazoxan hydrochloride
CAS:Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.Fórmula:C11H12N2O2·HClPureza:99.42% - 99.84%Forma y color:SolidPeso molecular:240.69Ref: TM-T0115
2mg35,00€5mg52,00€10mg78,00€25mg133,00€50mg187,00€100mg281,00€200mg416,00€1mL*10mM (DMSO)50,00€Xamoterol
CAS:Xamoterol is a cardiac stimulant.Fórmula:C16H25N3O5Forma y color:SolidPeso molecular:339.39Napitane Mesylate
CAS:Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Fórmula:C23H29NO5SPureza:98%Forma y color:SolidPeso molecular:431.55Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Apraclonidine
CAS:Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Fórmula:C9H10Cl2N4Forma y color:SolidPeso molecular:245.11Tulobuterol hydrochloride
CAS:Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.Fórmula:C12H19Cl2NOPureza:99.24% - >99.99%Forma y color:Appearance White Crystalline PowderPeso molecular:264.19Clebopride malate
CAS:Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Piribedil hydrochloride
CAS:Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.Fórmula:C16H19ClN4O2Forma y color:SolidPeso molecular:334.8Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Fórmula:C24H29ClN2O3Pureza:99.5%Forma y color:SolidPeso molecular:428.95Ref: TM-T9220
1mg42,00€5mg82,00€10mg111,00€25mg192,00€50mg289,00€100mg414,00€200mg580,00€1mL*10mM (DMSO)92,00€Guanabenz Acetate
CAS:Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.Fórmula:C8H8Cl2N4·C2H4O2Pureza:99% - 99.66%Forma y color:White Solid From Acetonitrile White SolidPeso molecular:291.13L755507
CAS:L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).Fórmula:C30H40N4O6SPureza:99% - 99.75%Forma y color:SolidPeso molecular:584.73
