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Receptor adrenérgico

Receptor adrenérgico

Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.

Subcategorías de "Receptor adrenérgico"

Se han encontrado 729 productos de "Receptor adrenérgico"

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  • (RS)-ICI-118551 Hydrochloride

    CAS:
    ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3
    Fórmula:C17H27NO2·HCl
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:313.86

    Ref: TM-T6860

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.341,00€
    100mg
    1.773,00€
  • LY 344864

    CAS:
    LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.
    Fórmula:C21H22FN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:351.42

    Ref: TM-T2344

    2mg
    38,00€
    5mg
    57,00€
    10mg
    93,00€
    25mg
    158,00€
    50mg
    280,00€
    100mg
    500,00€
    1mL*10mM (DMSO)
    63,00€
  • Falintolol

    CAS:

    Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study glaucoma.

    Fórmula:C12H24N2O2
    Pureza:>99.99% - >99.99%
    Forma y color:Solid
    Peso molecular:228.33

    Ref: TM-T68402

    1mg
    279,00€
    5mg
    685,00€
    10mg
    938,00€
    25mg
    1.388,00€
    50mg
    1.872,00€
    100mg
    2.527,00€
  • Bambuterol

    CAS:
    long acting beta-adrenoceptor agonist
    Fórmula:C18H29N3O5
    Pureza:98%
    Forma y color:Off-White Powder
    Peso molecular:367.44

    Ref: TM-T22599

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Landiolol

    CAS:
    Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.
    Fórmula:C25H39N3O8
    Pureza:98%
    Forma y color:White Crystalline Powder
    Peso molecular:509.59

    Ref: TM-T5028L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • D2343

    CAS:
    D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
    Fórmula:C20H27NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:329.43

    Ref: TM-T15042

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Salmefamol

    CAS:
    Salmefamol is a beta-adrenergic agonist. It may also be used as a bronchodilator.
    Fórmula:C19H25NO4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:331.41

    Ref: TM-T21352

    1mg
    264,00€
    5mg
    650,00€
    10mg
    888,00€
    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Efaroxan hydrochloride

    CAS:
    Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.
    Fórmula:C13H17ClN2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:252.74

    Ref: TM-T22760

    2mg
    36,00€
  • Protokylol hydrochloride

    CAS:
    Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.
    Fórmula:C18H22ClNO5
    Forma y color:Solid
    Peso molecular:367.83

    Ref: TM-T70854

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Clonidine

    CAS:
    Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
    Fórmula:C9H9Cl2N3
    Pureza:99.42% - 99.44%
    Forma y color:Crystals Solid
    Peso molecular:230.09

    Ref: TM-T7045

    5mg
    35,00€
    10mg
    46,00€
    25mg
    64,00€
    50mg
    89,00€
    100mg
    130,00€
    500mg
    306,00€
  • BRL 44408 Maleate Salt

    CAS:
    BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.
    Fórmula:C17H21N3O4
    Pureza:98.71%
    Forma y color:Solid
    Peso molecular:331.37

    Ref: TM-T26904

    1mg
    71,00€
    5mg
    155,00€
    10mg
    268,00€
    25mg
    442,00€
    50mg
    645,00€
    100mg
    950,00€
  • Butaxamine

    CAS:
    Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.
    Fórmula:C15H25NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:267.36

    Ref: TM-T25186

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Lusaperidone

    CAS:
    Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.
    Fórmula:C22H21N3O2
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:359.42

    Ref: TM-T11894

    1mg
    96,00€
    5mg
    207,00€
    10mg
    334,00€
    25mg
    687,00€
    50mg
    1.161,00€
    100mg
    1.710,00€
    200mg
    2.305,00€
  • IMTPPE

    CAS:
    IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.
    Fórmula:C20H27N3O2S
    Forma y color:Solid
    Peso molecular:373.51

    Ref: TM-T27601

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Abanoquil

    CAS:
    Abanoquil is an antagonist of alpha-1 adrenoceptor.
    Fórmula:C22H25N3O4
    Forma y color:Solid
    Peso molecular:395.45

    Ref: TM-T26507

    25mg
    907,00€
    50mg
    1.179,00€
    100mg
    1.529,00€
  • Zinterol

    CAS:
    Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).
    Fórmula:C19H26N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:378.49

    Ref: TM-T13399

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Metoprolol fumarate

    CAS:
    Metoprolol fumarate (CGP 2175C): selective β1-blocker with anti-inflammatory, antitumor, anti-angiogenic effects.
    Fórmula:C34H54N2O10
    Forma y color:Solid
    Peso molecular:650.8

    Ref: TM-T71752

    25mg
    421,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Clenproperol

    CAS:
    Clenproperol is a β2-adrenergic agonist.
    Fórmula:C11H16Cl2N2O
    Forma y color:Solid
    Peso molecular:263.16

    Ref: TM-T40480

    25mg
    1.444,00€
  • Isoetharine

    CAS:
    Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.
    Fórmula:C13H21NO3
    Forma y color:Solid
    Peso molecular:239.31

    Ref: TM-T4983L

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Denopamine

    CAS:
    Denopamine is an agonist of 1-Adrenoceptor.
    Fórmula:C18H23NO4
    Forma y color:Solid
    Peso molecular:317.38

    Ref: TM-T19707

    25mg
    973,00€
    50mg
    1.269,00€
    100mg
    1.998,00€