
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 729 productos de "Receptor adrenérgico"
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Methyldopate hydrochloride
CAS:Methyldopate HCl is an agent of antihypertensive.Fórmula:C12H18ClNO4Forma y color:SolidPeso molecular:275.73UK 1745
CAS:UK 1745 is a novel drug of cardiotonic.Fórmula:C16H23ClN2O2Forma y color:SolidPeso molecular:310.82Guanethidine
CAS:Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.Fórmula:C10H22N4Forma y color:SolidPeso molecular:198.31A 55453
CAS:A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.Fórmula:C25H32N6O3Forma y color:SolidPeso molecular:464.56RS 79948 hydrochloride
CAS:α2-adrenoreceptor antagonistFórmula:C19H29ClN2O3SPureza:98%Forma y color:SolidPeso molecular:400.96MK761
CAS:MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.Fórmula:C13H19N3O2Forma y color:SolidPeso molecular:249.31Napamezole
CAS:Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.Fórmula:C14H16N2Pureza:98%Forma y color:SolidPeso molecular:212.29Flestolol sulfate
CAS:Flestolol sulfate is an anti-adrenergic beta-receptor.Fórmula:C15H24FN3O8SForma y color:SolidPeso molecular:425.43BMS-466442
CAS:BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.Fórmula:C31H30N4O5Forma y color:SolidPeso molecular:538.59Mabuterol hydrochloride
CAS:Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.Fórmula:C13H19Cl2F3N2OForma y color:SolidPeso molecular:347.20Arbutamine hydrochloride
CAS:Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.Fórmula:C18H24ClNO4Forma y color:SolidPeso molecular:353.84Fenmetozole
CAS:Fenmetozole is an antagonist of the actions of ethanol.Fórmula:C10H10Cl2N2OForma y color:SolidPeso molecular:245.11CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Fórmula:C21H22N8O3Forma y color:SolidPeso molecular:434.45Clencyclohexerol
CAS:Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.Fórmula:C14H20Cl2N2O2Forma y color:SolidPeso molecular:319.23Dapiprazole
CAS:Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.Fórmula:C19H27N5Pureza:98%Forma y color:SolidPeso molecular:325.45BRL 37344 sodium
CAS:BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.Fórmula:C19H22ClNNaO4Pureza:98%Forma y color:SolidPeso molecular:386.83Pronethalol hydrochloride
CAS:β-adrenergic antagonistFórmula:C15H20ClNOPureza:98%Forma y color:SolidPeso molecular:265.78Naminterol
CAS:Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.Fórmula:C19H26N2O3Pureza:98%Forma y color:SolidPeso molecular:330.42Zenidolol
CAS:Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.Fórmula:C17H27NO2Forma y color:SolidPeso molecular:277.4ONO-2952
CAS:ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.Fórmula:C22H20ClFN2O2Pureza:98%Forma y color:SolidPeso molecular:398.86
