
Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 730 productos de "Receptor adrenérgico"
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Bedoradrine sulfate
CAS:Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Fórmula:C24H32N2O5H2O4SPureza:99.31%Forma y color:SolidPeso molecular:477.56GP2-114
CAS:GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.Fórmula:C19H24N2O4Pureza:99.32%Forma y color:SolidPeso molecular:344.4Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Fórmula:C19H21ClFN5O2Pureza:97.49% - >99.99%Forma y color:SolidPeso molecular:405.85Amosulalol
CAS:Amosulalol is a combined alpha and beta adrenoceptor antagonist.Fórmula:C18H24N2O5SPureza:99.5%Forma y color:SolidPeso molecular:380.46Ref: TM-T30027
1mg175,00€2mg264,00€5mg404,00€1mL*10mM (DMSO)430,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€CL 316243
CAS:CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Fórmula:C20H18ClNNa2O7Pureza:98.00% - 99.68%Forma y color:SolidPeso molecular:465.79Midaglizole hydrochloride
CAS:Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Fórmula:C16H19Cl2N3Pureza:99.39% - 99.82%Forma y color:SolidPeso molecular:324.25Ref: TM-T11015
1mg54,00€5mg119,00€1mL*10mM (DMSO)152,00€10mg188,00€25mg306,00€50mg416,00€100mg532,00€200mg705,00€Soquinolol
CAS:Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a longFórmula:C17H26N2O3Pureza:97.48% - 98.63%Forma y color:SolidPeso molecular:306.4Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Fórmula:C18H25N5O4Pureza:99.76% - 99.97%Forma y color:SolidPeso molecular:375.42Oxyfedrine L-form HCl
CAS:Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Fórmula:C19H24ClNO3Pureza:99.5% - 99.57%Forma y color:SolidPeso molecular:349.85Ref: TM-T24579
1mg92,00€5mg178,00€1mL*10mM (DMSO)203,00€10mg313,00€25mg485,00€50mg700,00€100mg893,00€200mg1.198,00€JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Fórmula:C24H24N4Pureza:99.96%Forma y color:SolidPeso molecular:368.47Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Fórmula:C26H33N3O6Pureza:99.89%Forma y color:SolidPeso molecular:483.56Ref: TM-T11148
1mg349,00€5mg697,00€1mL*10mM (DMSO)880,00€10mg888,00€25mg1.395,00€50mg1.783,00€100mg2.530,00€Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Fórmula:C10H11Cl2N3Pureza:98.06% - 98.83%Forma y color:SolidPeso molecular:244.12Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Fórmula:C17H26FNO3Pureza:98.96% - >99.99%Forma y color:SolidPeso molecular:311.392Rafabegron
CAS:Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Fórmula:C21H23ClN2O4Pureza:99.81%Forma y color:SolidPeso molecular:402.87Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Fórmula:C14H20N4OPureza:98.58% - 99.53%Forma y color:SolidPeso molecular:260.33Taprizosin
CAS:Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Fórmula:C25H26N6O4SPureza:98.10% - 99.11%Forma y color:SolidPeso molecular:506.58Milveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Fórmula:C25H30ClN3O4Pureza:99.9%Forma y color:SolidPeso molecular:471.98Dabelotine
CAS:Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.Fórmula:C15H22N2O2Pureza:97.96%Forma y color:SolidPeso molecular:262.35(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Fórmula:C36H40ClN3O6Pureza:98.27%Forma y color:SolidPeso molecular:646.17Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Fórmula:C16H17N3Pureza:97.15% - 98.85%Forma y color:SolidPeso molecular:251.33
