Receptor adrenérgico
Los receptores adrenérgicos son GPCR que son activados por catecolaminas, como la adrenalina y la noradrenalina. Estos receptores se clasifican en subtipos alfa y beta, cada uno de los cuales juega un papel clave en la regulación de la frecuencia cardíaca, la presión arterial y la respuesta de lucha o huida. Los moduladores de los receptores adrenérgicos son esenciales en el tratamiento de enfermedades cardiovasculares, asma y trastornos de ansiedad. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores adrenérgicos de alta calidad para apoyar su investigación en endocrinología, farmacología cardiovascular y respuesta al estrés.
Subcategorías de "Receptor adrenérgico"
Se han encontrado 729 productos de "Receptor adrenérgico"
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Bufuralol (hydrochloride)
CAS:Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Fórmula:C16H24ClNO2Forma y color:SolidPeso molecular:297.82Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Fórmula:C11H13ClN4O2Pureza:99.91%Forma y color:SolidPeso molecular:268.7Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Fórmula:C20H33N3O4·HClForma y color:White Crystalline SolidPeso molecular:415.96Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Fórmula:C16H23NO2Pureza:98.26%Forma y color:SolidPeso molecular:261.36Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Fórmula:C30H30ClN5O4SForma y color:SolidPeso molecular:592.11N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Fórmula:C20H23Cl2NO5Forma y color:SolidPeso molecular:428.31Indacaterol xinafoate
CAS:Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Fórmula:C35H36N2O6Forma y color:SolidPeso molecular:580.67Indacaterol acetate
CAS:Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Fórmula:C26H32N2O5Forma y color:SolidPeso molecular:452.54Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Fórmula:C18H22ClNO4Pureza:99.82%Forma y color:SolidPeso molecular:351.83Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Fórmula:C16H21N3Pureza:98.12% - 99.03%Forma y color:SolidPeso molecular:255.36CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Fórmula:C23H25F3N4O5Pureza:99.40% - 99.58%Forma y color:SolidPeso molecular:494.46Ref: TM-T30846
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€0990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFórmula:C21H21N5Pureza:98.99%Forma y color:SolidPeso molecular:343.42Ref: TM-T13983
1mg202,00€5mg512,00€10mg740,00€25mg1.121,00€50mg1.539,00€100mg2.072,00€1mL*10mM (DMSO)535,00€α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Fórmula:C20H24ClN5OPureza:99.20% - 99.29%Forma y color:SolidPeso molecular:385.89Ref: TM-T10003
1mg198,00€5mg393,00€10mg542,00€25mg785,00€50mg1.074,00€100mg1.454,00€200mg1.967,00€1mL*10mM (DMSO)467,00€OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Fórmula:C26H35N3O2Pureza:99.79%Forma y color:SolidPeso molecular:421.58Ref: TM-T13804
1mg187,00€5mg455,00€10mg620,00€25mg940,00€50mg1.264,00€100mg1.663,00€200mg2.252,00€1mL*10mM (DMSO)567,00€(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Fórmula:C12H19NO3Pureza:99.73%Forma y color:SolidPeso molecular:225.28Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Fórmula:C23H30N6O4Pureza:98%Forma y color:SolidPeso molecular:454.52LK 11
CAS:LK-11, an alkaloid derivative, inhibits the passive uptake of norepinephrine (NA) by synaptic vesicles in the thalamus, similarly to cocaine.Fórmula:C15H26N2O3Forma y color:SolidPeso molecular:282.38(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Fórmula:C18H29NO2Forma y color:SolidPeso molecular:291.43Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Fórmula:C26H28N4O3Forma y color:SolidPeso molecular:444.53Nipradolol
CAS:Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.Fórmula:C15H22N2O6Forma y color:SolidPeso molecular:326.35
