
GluR
Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.
Se han encontrado 255 productos de "GluR"
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Ro0711401
CAS:<p>Ro0711401 is an agonist of mGlu1 receptor.</p>Fórmula:C18H11F3N2O3Pureza:97.57%Forma y color:SolidPeso molecular:360.29YM90K
CAS:<p>YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.</p>Fórmula:C11H8ClN5O4Pureza:98.23%Forma y color:SolidPeso molecular:309.66HBT1
CAS:<p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>Fórmula:C16H17F3N4O2SPureza:99.52%Forma y color:SolidPeso molecular:386.393-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Forma y color:SolidPeso molecular:215.23VU 0357121
CAS:<p>VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.</p>Fórmula:C17H17F2NO2Pureza:99% - >99.99%Forma y color:SolidPeso molecular:305.32MTEP hydrochloride
CAS:<p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>Fórmula:C11H9ClN2SPureza:99.58%Forma y color:SolidPeso molecular:236.72FITM
CAS:<p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>Fórmula:C18H18FN5OSPureza:97.25%Forma y color:SolidPeso molecular:371.43ML 254
CAS:<p>是一种化学合成中的砌块</p>Fórmula:C18H15FN2O2Pureza:98.09%Forma y color:SolidPeso molecular:310.32AMN082 free base
CAS:<p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>Fórmula:C28H28N2Pureza:97.75% - 97.79%Forma y color:SolidPeso molecular:392.54MPEP hydrochloride
CAS:<p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>Fórmula:C14H12ClNPureza:99.87% - >99.99%Forma y color:SolidPeso molecular:229.7CX516
CAS:<p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>Fórmula:C14H15N3OPureza:99.04% - ≥95%Forma y color:Tan SolidPeso molecular:241.29MTEP
CAS:<p>MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.</p>Fórmula:C11H8N2SForma y color:SolidPeso molecular:200.26Ro 67-7476
CAS:<p>Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.</p>Fórmula:C17H18FNO2SPureza:99.69%Forma y color:SolidPeso molecular:319.39CTEP
CAS:<p>CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold</p>Fórmula:C19H13ClF3N3OPureza:99.17%Forma y color:SolidPeso molecular:391.77VU0155094
CAS:<p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>Fórmula:C24H24N2O4SPureza:97.21%Forma y color:SolidPeso molecular:436.52Caroverine hydrochloride
CAS:<p>Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.</p>Fórmula:C22H28ClN3O2Pureza:98.37% - 98.75%Forma y color:SolidPeso molecular:401.9VU 0364439
CAS:<p>VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).</p>Fórmula:C18H13Cl2N3O3SPureza:97.9%Forma y color:SolidPeso molecular:422.29JNJ-42153605
CAS:<p>JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).</p>Fórmula:C22H23F3N4Pureza:97.25% - 98.57%Forma y color:SolidPeso molecular:400.44VU0155041
CAS:<p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>Fórmula:C14H15Cl2NO3Pureza:99.52% - 99.56%Forma y color:SolidPeso molecular:316.18JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Forma y color:SolidPeso molecular:344.88
