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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Se han encontrado 255 productos de "GluR"

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  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Forma y color:Solid
    Peso molecular:360.29
  • YM90K

    CAS:
    <p>YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.</p>
    Fórmula:C11H8ClN5O4
    Pureza:98.23%
    Forma y color:Solid
    Peso molecular:309.66
  • HBT1

    CAS:
    <p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>
    Fórmula:C16H17F3N4O2S
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:386.39
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Forma y color:Solid
    Peso molecular:215.23
  • VU 0357121

    CAS:
    <p>VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.</p>
    Fórmula:C17H17F2NO2
    Pureza:99% - >99.99%
    Forma y color:Solid
    Peso molecular:305.32
  • MTEP hydrochloride

    CAS:
    <p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>
    Fórmula:C11H9ClN2S
    Pureza:99.58%
    Forma y color:Solid
    Peso molecular:236.72
  • FITM

    CAS:
    <p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>
    Fórmula:C18H18FN5OS
    Pureza:97.25%
    Forma y color:Solid
    Peso molecular:371.43
  • ML 254

    CAS:
    <p>是一种化学合成中的砌块</p>
    Fórmula:C18H15FN2O2
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:310.32
  • AMN082 free base

    CAS:
    <p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>
    Fórmula:C28H28N2
    Pureza:97.75% - 97.79%
    Forma y color:Solid
    Peso molecular:392.54
  • MPEP hydrochloride

    CAS:
    <p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>
    Fórmula:C14H12ClN
    Pureza:99.87% - >99.99%
    Forma y color:Solid
    Peso molecular:229.7
  • CX516

    CAS:
    <p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>
    Fórmula:C14H15N3O
    Pureza:99.04% - ≥95%
    Forma y color:Tan Solid
    Peso molecular:241.29
  • MTEP

    CAS:
    <p>MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.</p>
    Fórmula:C11H8N2S
    Forma y color:Solid
    Peso molecular:200.26
  • Ro 67-7476

    CAS:
    <p>Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.</p>
    Fórmula:C17H18FNO2S
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:319.39
  • CTEP

    CAS:
    <p>CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows &gt;1000-fold</p>
    Fórmula:C19H13ClF3N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:391.77
  • VU0155094

    CAS:
    <p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>
    Fórmula:C24H24N2O4S
    Pureza:97.21%
    Forma y color:Solid
    Peso molecular:436.52
  • Caroverine hydrochloride

    CAS:
    <p>Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.</p>
    Fórmula:C22H28ClN3O2
    Pureza:98.37% - 98.75%
    Forma y color:Solid
    Peso molecular:401.9
  • VU 0364439

    CAS:
    <p>VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).</p>
    Fórmula:C18H13Cl2N3O3S
    Pureza:97.9%
    Forma y color:Solid
    Peso molecular:422.29
  • JNJ-42153605

    CAS:
    <p>JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).</p>
    Fórmula:C22H23F3N4
    Pureza:97.25% - 98.57%
    Forma y color:Solid
    Peso molecular:400.44
  • VU0155041

    CAS:
    <p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>
    Fórmula:C14H15Cl2NO3
    Pureza:99.52% - 99.56%
    Forma y color:Solid
    Peso molecular:316.18
  • JNJ-40411813

    CAS:
    <p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:344.88