
GluR
Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.
Se han encontrado 255 productos de "GluR"
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CX717
CAS:<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Fórmula:C11H11N3O3Pureza:99.81%Forma y color:SoildPeso molecular:233.23(S)-4CPG
CAS:<p>(S)-4CPG ((S)-4-Carboxyphenylglycine) is a competitive mGlu1 receptor antagonist that attenuates nociceptive hypersensitivity and nociceptive abnormalities associated with sciatic nerve constriction injuries in rats, and may be used in the study of neurological disorders.</p>Fórmula:C9H9NO4Pureza:99.96%Forma y color:SolidPeso molecular:195.17VU0477886
CAS:<p>VU0477886: Potent mGlu4 PAM, effective in preclinical Parkinson's model HIC.</p>Fórmula:C20H13ClN4O3Pureza:98%Forma y color:SolidPeso molecular:392.80IEM 1754 2HBr
CAS:<p>IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.</p>Fórmula:C16H30N2·2HBrPureza:99.71% - 99.72%Forma y color:SolidPeso molecular:412.25LY456066
CAS:<p>LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.</p>Fórmula:C19H23N3OSPureza:98%Forma y color:SolidPeso molecular:341.47Methoxy-PEPy
CAS:<p>Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.</p>Fórmula:C13H10N2OPureza:99.22%Forma y color:SolidPeso molecular:210.23Z-Cyclopentyl-AP4
CAS:<p>Group III mGlu receptor agonist</p>Fórmula:C6H12NO5PPureza:98%Forma y color:SolidPeso molecular:209.14DFMTI
CAS:<p>DFMTI can completely block the rmGlu1 L757V glutamate response.</p>Fórmula:C20H18F2N4OForma y color:SolidPeso molecular:368.38LY392098
CAS:<p>LY392098 (AMPA receptor modulator-3) is an allosteric modulator of AMPA receptor with EC50 of 4.4 μM and can be used in studies about mammalian nervous system.</p>Fórmula:C18H22FNO2SPureza:99.86%Forma y color:SolidPeso molecular:335.44GRN-529
CAS:<p>GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.</p>Fórmula:C22H15F2N3O2Pureza:98%Forma y color:SolidPeso molecular:391.37NPEC-caged-LY379268
CAS:<p>NPEC-caged-LY379268 is a type II mGluR agonist [1].</p>Fórmula:C16H16N2O9Forma y color:SolidPeso molecular:380.31MAP4
CAS:<p>metabotropic glutamate receptor modulator</p>Fórmula:C5H12NO5PPureza:98%Forma y color:White SolidPeso molecular:197.13mGluR2 modulator 1
CAS:<p>Potent mGluR2 modulator 1 crosses blood-brain barrier, EC50: 0.03 μM, useful for psychiatric research.</p>Fórmula:C21H20F3N3O3Forma y color:SolidPeso molecular:419.4RO4988546
CAS:<p>RO4988546 is a potent negative allosteric modulator of mGlu₂/₃.</p>Fórmula:C21H10F6N4O3SPureza:98%Forma y color:SolidPeso molecular:512.38LSN2814617
CAS:<p>LSN2814617: oral, brain-penetrant mGlu5 PAM, EC50 = 52 nM (human), 42 nM (rat). Promotes wakefulness, useful in schizophrenia study.</p>Fórmula:C18H20FN5OPureza:98%Forma y color:SolidPeso molecular:341.38mGlu4 receptor agonist 1
CAS:<p>Compound 62, an mGlu4 agonist, has a 308 nM EC50 with anxiolytic and antipsychotic effects.</p>Fórmula:C21H15ClN4O2Forma y color:SolidPeso molecular:390.82A 841720
CAS:<p>Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.</p>Fórmula:C17H21N5OSForma y color:SolidPeso molecular:343.45RO5488608
CAS:<p>RO5488608 is a new type of high-efficiency mGlu2/3 NAM.</p>Fórmula:C23H17F3N2O4SForma y color:SolidPeso molecular:474.45ADX71743
CAS:<p>ADX71743 is a potent and selective negative allosteric modulator of metabotropic glutamate receptor 7.</p>Fórmula:C17H19NO2Forma y color:SolidPeso molecular:269.34VU0463841
CAS:<p>VU0463841 is a mGlu5 negative allosteric modulators.</p>Fórmula:C13H8ClFN4OForma y color:SolidPeso molecular:290.68
