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AChR

AChR

Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.

Se han encontrado 623 productos de "AChR"

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productos por página.
  • YM-58790 hydrochloride

    CAS:
    YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).
    Fórmula:C27H32ClN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:466.02

    Ref: TM-T13372

    5mg
    308,00€
    50mg
    1.586,00€
    100mg
    2.555,00€
  • Palmatine hydroxide

    CAS:
    Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.
    Fórmula:C21H23NO5
    Forma y color:Solid
    Peso molecular:369.41

    Ref: TM-T72508

    50mg
    35,00€
    100mg
    48,00€
  • β2AR/M-receptor agonist-2

    CAS:
    <p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>
    Fórmula:C36H49ClN4O7S
    Forma y color:Solid
    Peso molecular:717.31

    Ref: TM-T72226

    25mg
    4.845,00€
    50mg
    6.346,00€
    100mg
    8.540,00€
  • Dexetimide

    CAS:
    Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.
    Fórmula:C23H26N2O2
    Forma y color:Solid
    Peso molecular:362.46

    Ref: TM-T15104

    2mg
    44,00€
    5mg
    63,00€
    1mL*10mM (DMSO)
    87,00€
  • Varenicline Hydrochloride

    CAS:
    Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).
    Fórmula:C13H14ClN3
    Pureza:99.854%
    Forma y color:Solid
    Peso molecular:247.72

    Ref: TM-T23502

    1mg
    38,00€
    5mg
    80,00€
    10mg
    105,00€
    25mg
    192,00€
    50mg
    297,00€
    100mg
    441,00€
    200mg
    646,00€
    1mL*10mM (DMSO)
    88,00€
  • Glycerophosphoinositol choline

    CAS:
    Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.
    Fórmula:C14H32NO12P
    Forma y color:Solid
    Peso molecular:437.38

    Ref: TM-T31951

    5mg
    2.042,00€
    50mg
    A consultar
    100mg
    A consultar
  • Cevimeline hydrochloride

    CAS:
    Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.
    Fórmula:C10H18ClOS
    Forma y color:Solid
    Peso molecular:235.77

    Ref: TM-T20131

    2mg
    65,00€
  • (±)-Darifenacin

    CAS:
    (±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.
    Fórmula:C28H30N2O2
    Forma y color:Solid
    Peso molecular:426.55

    Ref: TM-T12680

    5mg
    54,00€
    10mg
    A consultar
    25mg
    A consultar
    1mL*10mM (DMSO)
    75,00€
  • VU0467485

    CAS:
    VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.
    Fórmula:C17H17FN4O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:360.41

    Ref: TM-T17245

    2mg
    86,00€
  • Clorprenaline

    CAS:
    Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.
    Fórmula:C11H16ClNO
    Pureza:98.9%
    Forma y color:Solid
    Peso molecular:213.7

    Ref: TM-T60261

    5mg
    52,00€
    10mg
    75,00€
    25mg
    130,00€
    50mg
    203,00€
    100mg
    302,00€
    200mg
    449,00€
  • SSR180711 hydrochloride

    CAS:
    SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.
    Fórmula:C14H18BrClN2O2
    Pureza:99.22%
    Forma y color:Solid
    Peso molecular:361.66

    Ref: TM-T28856

    1mg
    35,00€
    5mg
    73,00€
    10mg
    111,00€
    25mg
    178,00€
    50mg
    271,00€
    1mL*10mM (DMSO)
    81,00€
  • Pirmenol hydrochloride

    CAS:
    Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM
    Fórmula:C22H31ClN2O
    Forma y color:Solid
    Peso molecular:374.95

    Ref: TM-T61529

    2mg
    35,00€
    1mL*10mM (DMSO)
    65,00€
  • Tebanicline dihydrochloride

    CAS:
    Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.
    Fórmula:C9H13Cl3N2O
    Forma y color:Solid
    Peso molecular:271.57

    Ref: TM-T60474

    2mg
    54,00€
    1mL*10mM (DMSO)
    95,00€
  • Biperiden

    CAS:
    Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.
    Fórmula:C21H29NO
    Pureza:99.65%
    Forma y color:Crystals Solid
    Peso molecular:311.46

    Ref: TM-T0218

    1mg
    54,00€
    5mg
    A consultar
    10mg
    A consultar
    1mL*10mM (DMSO)
    190,00€
  • Ispronicline

    CAS:
    Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive
    Fórmula:C14H22N2O
    Pureza:97.70% - 99.16%
    Forma y color:Solid
    Peso molecular:234.34

    Ref: TM-T27636

    2mg
    46,00€
    5mg
    66,00€
    10mg
    87,00€
    25mg
    154,00€
    50mg
    210,00€
    100mg
    311,00€
    1mL*10mM (DMSO)
    73,00€
  • (S)-(+)-Dimethindene maleate

    CAS:
    (S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors
    Fórmula:C24H28N2O4
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:408.49

    Ref: TM-T23297

    1mg
    49,00€
  • Sabcomeline hydrochloride

    CAS:
    Sabcomeline is a selective M1 receptor partial agonist.
    Fórmula:C10H16ClN3O
    Forma y color:Solid
    Peso molecular:229.71

    Ref: TM-T28654

    2mg
    464,00€
  • NS3861 fumarate

    CAS:
    NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.
    Fórmula:C16H18BrNO4S
    Forma y color:Solid
    Peso molecular:400.29

    Ref: TM-T9450

    2mg
    54,00€
  • NKH477

    CAS:
    NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.
    Fórmula:C27H44ClNO8
    Pureza:98% - 98%
    Forma y color:Solid
    Peso molecular:546.09

    Ref: TM-T16332

    2mg
    146,00€
  • ABT-107

    CAS:
    ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.
    Fórmula:C19H20N4O
    Forma y color:Solid
    Peso molecular:320.396

    Ref: TM-T40951

    5mg
    358,00€
    1mL*10mM (DMSO)
    358,00€
  • NSC 23766

    CAS:
    NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.
    Fórmula:C24H35N7
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:421.58

    Ref: TM-T40848

    2mg
    54,00€
  • DL-Cystine

    CAS:
    DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .
    Fórmula:C6H12N2O4S2
    Forma y color:Solid
    Peso molecular:240.3

    Ref: TM-T66846

    200mg
    34,00€
  • NBTGR

    CAS:
    NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
    Fórmula:C17H18N6O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:434.43

    Ref: TM-T12191

    2mg
    86,00€
    5mg
    142,00€
    1mL*10mM (DMSO)
    172,00€
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:359.89

    Ref: TM-T7555

    10mg
    37,00€
    25mg
    52,00€
    50mg
    77,00€
    100mg
    103,00€
    200mg
    158,00€
    1mL*10mM (DMSO)
    116,00€
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Fórmula:C14H30N2O4·2Cl·2H2O
    Pureza:99.87%
    Forma y color:White Solid
    Peso molecular:397.34

    Ref: TM-T6684

    1g
    507,00€
    10mg
    39,00€
    25mg
    55,00€
    50mg
    71,00€
    100mg
    116,00€
    200mg
    202,00€
    500mg
    341,00€
  • Tebanicline hydrochloride

    CAS:
    Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.
    Fórmula:C9H12Cl2N2O
    Pureza:91.74% - 98.78%
    Forma y color:Solid
    Peso molecular:235.11

    Ref: TM-T3720

    1mg
    44,00€
    2mg
    56,00€
    5mg
    89,00€
    10mg
    138,00€
    25mg
    264,00€
    50mg
    474,00€
    100mg
    688,00€
    500mg
    1.444,00€
  • VU0357017 hydrochloride

    CAS:
    VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.
    Fórmula:C18H28ClN3O3
    Pureza:99% - 99.97%
    Forma y color:Solid
    Peso molecular:369.89

    Ref: TM-T3619

    5mg
    40,00€
    10mg
    58,00€
    25mg
    97,00€
    50mg
    156,00€
    100mg
    221,00€
    200mg
    329,00€
    1mL*10mM (DMSO)
    44,00€
  • α-Conotoxin MII acetate


    α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.
    Fórmula:C69H107N23O24S4
    Pureza:94.82% - 97.79%
    Forma y color:Solid
    Peso molecular:1770.99

    Ref: TM-TP2063L

    1mg
    145,00€
    5mg
    319,00€
    10mg
    472,00€
    25mg
    753,00€
    50mg
    1.074,00€
    100mg
    1.444,00€
  • VU0119498

    CAS:
    VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.
    Fórmula:C15H10BrNO2
    Pureza:97.56%
    Forma y color:Solid
    Peso molecular:316.15

    Ref: TM-T8224

    25mg
    44,00€
    50mg
    62,00€
    100mg
    90,00€
    200mg
    123,00€
    1mL*10mM (DMSO)
    34,00€
  • Clothianidin

    CAS:
    Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.
    Fórmula:C6H8ClN5O2S
    Pureza:99.71% - 99.87%
    Forma y color:Solid Powder
    Peso molecular:249.68

    Ref: TM-T21153

    1g
    133,00€
    100mg
    47,00€
    200mg
    62,00€
    500mg
    90,00€
    1mL*10mM (DMSO)
    34,00€
  • VU0152100

    CAS:
    <p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>
    Fórmula:C18H19N3O2S
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:341.43

    Ref: TM-T17238

    1mg
    40,00€
    5mg
    88,00€
    10mg
    118,00€
    25mg
    254,00€
    50mg
    406,00€
    100mg
    612,00€
    200mg
    842,00€
  • Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Fórmula:C17H17N5O6S
    Pureza:99.69% - 99.74%
    Forma y color:Off-White Solid
    Peso molecular:419.41

    Ref: TM-T8551

    5mg
    48,00€
    10mg
    66,00€
    25mg
    125,00€
    50mg
    188,00€
    100mg
    283,00€
    200mg
    434,00€
  • KH7

    CAS:
    KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
    Fórmula:C17H15BrN4O2S
    Pureza:98.43%
    Forma y color:Solid
    Peso molecular:419.3

    Ref: TM-T15658

    1mg
    44,00€
    2mg
    55,00€
    5mg
    89,00€
    10mg
    130,00€
    25mg
    251,00€
    50mg
    A consultar
    1mL*10mM (DMSO)
    89,00€
  • VU0467154

    CAS:
    VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.
    Fórmula:C17H15F3N4O3S2
    Pureza:99.51% - 99.53%
    Forma y color:Solid
    Peso molecular:444.45

    Ref: TM-T17244

    1mg
    49,00€
    2mg
    66,00€
    5mg
    97,00€
    10mg
    133,00€
    25mg
    250,00€
    50mg
    423,00€
    100mg
    735,00€
    200mg
    998,00€
    1mL*10mM (DMSO)
    106,00€
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Fórmula:C14H8N4O
    Pureza:99.12%
    Forma y color:Solid
    Peso molecular:248.24

    Ref: TM-T28199

    1mg
    46,00€
    5mg
    96,00€
    10mg
    144,00€
    25mg
    298,00€
    50mg
    469,00€
    100mg
    687,00€
    500mg
    1.444,00€
  • ML380

    CAS:
    <p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>
    Fórmula:C23H25F3N4O3S
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:494.53

    Ref: TM-T28069

    2mg
    49,00€
    5mg
    74,00€
    10mg
    119,00€
    25mg
    188,00€
    50mg
    354,00€
    100mg
    528,00€
    500mg
    1.159,00€
  • Varenicline Tartrate

    CAS:
    <p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>
    Fórmula:C13H13N3·C4H6O6
    Pureza:98.23% - 98.32%
    Forma y color:Tan Solid
    Peso molecular:361.35

    Ref: TM-T1657

    5mg
    35,00€
    10mg
    48,00€
    25mg
    80,00€
    50mg
    120,00€
    100mg
    187,00€
  • Cyclodrine hydrochloride

    CAS:
    Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of
    Fórmula:C19H30ClNO3
    Pureza:98.59%
    Forma y color:Solid
    Peso molecular:355.9

    Ref: TM-T10914

    1mg
    665,00€
    5mg
    1.710,00€
  • Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Fórmula:C23H33IN2O
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:480.43

    Ref: TM-T5051

    10mg
    42,00€
    25mg
    62,00€
    50mg
    88,00€
    100mg
    117,00€
  • Mc-​Val-​Ala-​PAB

    CAS:
    <p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>
    Fórmula:C25H34N4O6
    Pureza:98.34% - 99.24%
    Forma y color:Solid
    Peso molecular:486.56

    Ref: TM-T4289

    25mg
    34,00€
    50mg
    42,00€
  • Nitenpyram

    CAS:
    Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.
    Fórmula:C11H15ClN4O2
    Pureza:99.03%
    Forma y color:Light-Yellow Crystal
    Peso molecular:270.72

    Ref: TM-T6607

    1g
    104,00€
    200mg
    48,00€
    500mg
    80,00€
    1mL*10mM (DMSO)
    34,00€
  • Mecamylamine hydrochloride

    CAS:
    Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
    Fórmula:C11H22ClN
    Pureza:99.76% - >99.99%
    Forma y color:White Solid
    Peso molecular:203.75

    Ref: TM-T2141

    5mg
    35,00€
    10mg
    56,00€
    25mg
    119,00€
    50mg
    187,00€
    100mg
    283,00€
    200mg
    432,00€
    1mL*10mM (DMSO)
    40,00€
  • Solifenacin hydrochloride

    CAS:
    Solifenacin Hcl is a muscarinic receptor antagonist.
    Fórmula:C23H27ClN2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:398.93

    Ref: TM-T23379

    2mg
    50,00€
    5mg
    97,00€
    1mL*10mM (DMSO)
    96,00€
  • JHU37152

    CAS:
    JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.
    Fórmula:C19H20ClFN4
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:358.84

    Ref: TM-T9019

    10mg
    35,00€
    25mg
    63,00€
    50mg
    88,00€
    100mg
    143,00€
    200mg
    208,00€
    1mL*10mM (DMSO)
    34,00€
  • Encenicline

    CAS:
    Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.
    Fórmula:C16H17ClN2OS
    Pureza:99.20%
    Forma y color:Solid
    Peso molecular:320.84

    Ref: TM-T7193

    1mg
    73,00€
    5mg
    140,00€
    10mg
    220,00€
    25mg
    369,00€
    50mg
    523,00€
    100mg
    712,00€
    200mg
    938,00€
    1mL*10mM (DMSO)
    153,00€
  • Syn-Ake acetate

    CAS:
    Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.
    Fórmula:C19H29N5O3·2(C2H4O2)
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:495.58

    Ref: TM-T7895

    50mg
    37,00€
    100mg
    52,00€
  • Sofpironium bromide

    CAS:
    Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.
    Fórmula:C22H32BrNO5
    Pureza:98.85%
    Forma y color:Solid
    Peso molecular:470.4

    Ref: TM-T28827

    1mg
    74,00€
    5mg
    160,00€
    10mg
    250,00€
    25mg
    452,00€
    50mg
    680,00€
    100mg
    1.008,00€
    200mg
    1.349,00€
    1mL*10mM (DMSO)
    165,00€
  • Mecamylamine

    CAS:
    Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.
    Fórmula:C11H21N
    Forma y color:Solid
    Peso molecular:167.29

    Ref: TM-T69019

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Oxyphencyclimine Hydrochloride

    CAS:
    Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.
    Fórmula:C20H29ClN2O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:380.91

    Ref: TM-T2138

    2mg
    39,00€
    5mg
    56,00€
    10mg
    87,00€
    25mg
    A consultar
    50mg
    A consultar
  • Pempidine

    CAS:
    Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
    Fórmula:C10H21N
    Pureza:98.18% - 99.28%
    Forma y color:Colorless - Light Yellow Clear Liquid
    Peso molecular:155.28

    Ref: TM-T0296

    1g
    57,00€
    5g
    88,00€
    200mg
    37,00€
    500mg
    52,00€
    1mL*10mM (DMSO)
    34,00€
  • Propiverine

    CAS:
    Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.
    Fórmula:C23H29NO3
    Forma y color:Solid
    Peso molecular:367.48

    Ref: TM-T61438

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • NS 1738

    CAS:
    NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)
    Fórmula:C14H9Cl2F3N2O2
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:365.13

    Ref: TM-T7884

    5mg
    51,00€
    10mg
    92,00€
    25mg
    169,00€
    50mg
    279,00€
    100mg
    472,00€
    1mL*10mM (DMSO)
    57,00€
  • Dinotefuran

    CAS:
    Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.
    Fórmula:C7H14N4O3
    Pureza:99.89%
    Forma y color:White Crystalline Powder
    Peso molecular:202.21

    Ref: TM-T7124

    1g
    144,00€
    100mg
    52,00€
    200mg
    72,00€
    500mg
    97,00€
    1mL*10mM (DMSO)
    34,00€
  • Procyclidine hydrochloride

    CAS:
    Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.
    Fórmula:C19H30ClNO
    Pureza:99.24% - 99.88%
    Forma y color:Crystals From Petroleum Ether White Powder
    Peso molecular:323.9

    Ref: TM-T4979

    25mg
    34,00€
    1mL*10mM (DMSO)
    58,00€
  • Dronedarone

    CAS:
    Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
    Fórmula:C31H44N2O5S
    Pureza:98.85% - 99.99%
    Forma y color:Solid
    Peso molecular:556.76

    Ref: TM-T7056

    10mg
    47,00€
    25mg
    87,00€
    50mg
    117,00€
    100mg
    170,00€
    1mL*10mM (DMSO)
    50,00€
  • EB-3D

    CAS:
    EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.
    Fórmula:C30H36Br2N4O2
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:644.4

    Ref: TM-T7955

    1mg
    92,00€
    2mg
    120,00€
    5mg
    187,00€
    10mg
    274,00€
    25mg
    472,00€
    50mg
    655,00€
    100mg
    924,00€
    200mg
    1.225,00€
    1mL*10mM (DMSO)
    278,00€
  • Oxyphenonium bromide

    CAS:
    <p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>
    Fórmula:C21H34BrNO3
    Pureza:98.96%
    Forma y color:Solid
    Peso molecular:428.404

    Ref: TM-T33846

    10mg
    47,00€
    25mg
    67,00€
    50mg
    89,00€
    100mg
    131,00€
  • MC-Val-Cit-PABC-PNP

    CAS:
    MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.
    Fórmula:C35H43N7O11
    Pureza:97.2% - 98.055%
    Forma y color:Solid
    Peso molecular:737.76

    Ref: TM-T3503

    50mg
    34,00€
  • Propantheline

    CAS:
    Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.
    Fórmula:C23H30NO3
    Forma y color:Solid
    Peso molecular:368.49

    Ref: TM-T61453

    25mg
    2.033,00€
    50mg
    2.645,00€
    100mg
    3.345,00€
  • Bestim

    CAS:
    Bestim is an immunomodulatory dipeptide that is synthetic.
    Fórmula:C16H19N3O5
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:333.34

    Ref: TM-T25146

    1mg
    88,00€
    5mg
    172,00€
    10mg
    259,00€
    25mg
    425,00€
    50mg
    598,00€
    100mg
    810,00€
    200mg
    1.074,00€
    1mL*10mM (DMSO)
    182,00€
  • VU0152099

    CAS:
    VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
    Fórmula:C18H17N3O3S
    Pureza:98.46%
    Forma y color:Solid
    Peso molecular:355.41

    Ref: TM-T29123

    10mg
    40,00€
    25mg
    74,00€
    50mg
    115,00€
    100mg
    178,00€
    200mg
    256,00€
    1mL*10mM (DMSO)
    37,00€
  • Adiphenine

    CAS:
    Adiphenine is an inhibitor of nicotinic receptors.
    Fórmula:C20H25NO2
    Forma y color:Solid
    Peso molecular:311.42

    Ref: TM-T68940

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Rivanicline hemioxalate


    Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.
    Fórmula:C12H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:207.23

    Ref: TM-T12738

    500mg
    1.685,00€
  • Simufilam dihydrochloride

    CAS:
    Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.
    Fórmula:C15H23Cl2N3O
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:332.3

    Ref: TM-T9172

    1mg
    52,00€
    5mg
    90,00€
    10mg
    143,00€
    25mg
    294,00€
    50mg
    380,00€
    100mg
    497,00€
    200mg
    655,00€
    1mL*10mM (DMSO)
    101,00€
  • Batefenterol

    CAS:
    Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).
    Fórmula:C40H42ClN5O7
    Pureza:97.94% - 98.4%
    Forma y color:Solid
    Peso molecular:740.24

    Ref: TM-T7079

    1mg
    48,00€
    5mg
    95,00€
    10mg
    154,00€
    25mg
    274,00€
    50mg
    425,00€
    100mg
    615,00€
    1mL*10mM (DMSO)
    155,00€
  • suvn-911

    CAS:
    suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.
    Fórmula:C11H14Cl2N2O
    Pureza:98.88%
    Forma y color:Solid
    Peso molecular:261.15

    Ref: TM-T9787

    1mg
    71,00€
    5mg
    140,00€
    10mg
    215,00€
    25mg
    359,00€
    50mg
    510,00€
    100mg
    695,00€
    200mg
    937,00€
    1mL*10mM (DMSO)
    182,00€
  • Coluracetam

    CAS:
    Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.
    Fórmula:C19H23N3O3
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:341.4

    Ref: TM-T7591

    1g
    243,00€
    10mg
    37,00€
    25mg
    51,00€
    50mg
    67,00€
    100mg
    80,00€
    500mg
    170,00€
  • Aclidinium bromide

    CAS:
    <p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>
    Fórmula:C26H30NO4S2·Br
    Pureza:99.53% - 99.69%
    Forma y color:Solid
    Peso molecular:564.55

    Ref: TM-T2555

    2mg
    39,00€
    5mg
    57,00€
    10mg
    88,00€
    25mg
    145,00€
    50mg
    234,00€
    100mg
    350,00€
    500mg
    825,00€
  • Encenicline hydrochloride

    CAS:
    Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).
    Fórmula:C16H17ClN2OS·HCl
    Pureza:98.34% - 99.85%
    Forma y color:Solid
    Peso molecular:357.3

    Ref: TM-T2285

    1mg
    59,00€
    5mg
    125,00€
    10mg
    188,00€
    25mg
    393,00€
    50mg
    628,00€
    100mg
    998,00€
    1mL*10mM (DMSO)
    136,00€
  • Pempidine HCl

    CAS:
    Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.
    Fórmula:C10H22ClN
    Forma y color:Solid
    Peso molecular:191.74

    Ref: TM-T68992

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Umeclidinium bromide

    CAS:
    Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.
    Fórmula:C29H34BrNO2
    Pureza:98.4% - 99.89%
    Forma y color:Solid
    Peso molecular:508.49

    Ref: TM-T4997

    1mg
    40,00€
    2mg
    52,00€
    5mg
    85,00€
    10mg
    124,00€
    25mg
    212,00€
    50mg
    350,00€
    100mg
    525,00€
    1mL*10mM (DMSO)
    87,00€
  • PHA 568487 free base

    CAS:
    <p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>
    Fórmula:C16H20N2O3
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:288.34

    Ref: TM-T23146

    10mg
    44,00€
    25mg
    74,00€
    50mg
    130,00€
    100mg
    225,00€
    200mg
    314,00€
  • Batefenterol Succinate

    CAS:
    Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.
    Fórmula:C44H48ClN5O11
    Forma y color:Solid
    Peso molecular:858.34

    Ref: TM-T68272

    25mg
    2.015,00€
    50mg
    2.642,00€
    100mg
    3.515,00€
  • VU0238441

    CAS:
    VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
    Fórmula:C16H9ClF3NO2
    Pureza:100%
    Forma y color:Solid
    Peso molecular:339.7

    Ref: TM-T8219

    25mg
    42,00€
    50mg
    52,00€
    1mL*10mM (DMSO)
    A consultar
  • Benzetimide hydrochloride

    CAS:
    Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.
    Fórmula:C23H27ClN2O2
    Pureza:99.32%
    Forma y color:Off-White Powder
    Peso molecular:398.93

    Ref: TM-T7561

    25mg
    37,00€
    50mg
    48,00€
    100mg
    60,00€
    1mL*10mM (DMSO)
    34,00€
  • Oxyphencyclimine

    CAS:
    Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.
    Fórmula:C20H28N2O3
    Forma y color:Solid
    Peso molecular:344.45

    Ref: TM-T2138L

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • (S)-UFR2709

    CAS:
    (S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.
    Fórmula:C13H17NO2
    Forma y color:Solid
    Peso molecular:219.284

    Ref: TM-T38903

    5mg
    922,00€
  • mAChR-IN-1 hydrochloride

    CAS:
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
    Fórmula:C23H26ClIN2O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:524.82

    Ref: TM-T5655

    1mg
    40,00€
    5mg
    90,00€
    10mg
    133,00€
    25mg
    227,00€
    50mg
    314,00€
    100mg
    393,00€
    200mg
    520,00€
    1mL*10mM (DMSO)
    95,00€
  • Solifenacin

    CAS:
    Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,
    Fórmula:C23H26N2O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:362.46

    Ref: TM-T8147

    25mg
    47,00€
    50mg
    64,00€
    100mg
    92,00€
    500mg
    210,00€
    1mL*10mM (DMSO)
    34,00€
  • LY2119620

    CAS:
    LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.
    Fórmula:C19H24ClN5O3S
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:437.94

    Ref: TM-T6575

    1mg
    57,00€
    5mg
    123,00€
    10mg
    188,00€
    25mg
    328,00€
    50mg
    459,00€
    100mg
    645,00€
    1mL*10mM (DMSO)
    130,00€
  • Pirmenol

    CAS:
    Pirmenol is a new antiarrhythmic drug
    Fórmula:C22H30N2O
    Pureza:97.24%
    Forma y color:Solid
    Peso molecular:338.49

    Ref: TM-T7531

    5mg
    55,00€
    50mg
    105,00€
    100mg
    158,00€
    1mL*10mM (DMSO)
    58,00€
  • Anisotropine Methylbromide

    CAS:
    Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.
    Fórmula:C17H32BrNO2
    Pureza:99.73%
    Forma y color:Crystals From Acetone Solid
    Peso molecular:362.35

    Ref: TM-T4981

    5mg
    35,00€
    10mg
    48,00€
    25mg
    81,00€
    50mg
    120,00€
    100mg
    187,00€
  • Darifenacin

    CAS:
    Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.
    Fórmula:C28H30N2O2
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:426.55

    Ref: TM-T62320

    2mg
    42,00€
    5mg
    62,00€
    10mg
    87,00€
    25mg
    160,00€
    50mg
    250,00€
    100mg
    376,00€
    200mg
    550,00€
    1mL*10mM (DMSO)
    67,00€
  • Ilmetropium iodide

    CAS:
    Ilmetropium iodide is a bronchodilator.
    Fórmula:C20H30INO3
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:459.36

    Ref: TM-T27594

    5mg
    34,00€
    10mg
    49,00€
    25mg
    85,00€
    50mg
    113,00€
    100mg
    169,00€
    200mg
    246,00€
    1mL*10mM (DMSO)
    50,00€
  • BNC210

    CAS:
    BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.
    Fórmula:C17H23N3O3
    Pureza:97.05% - >99.99%
    Forma y color:Solid
    Peso molecular:317.38

    Ref: TM-T8318

    25mg
    48,00€
    50mg
    74,00€
    100mg
    97,00€
    1mL*10mM (DMSO)
    34,00€
  • Brompheniramine

    CAS:
    Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.
    Fórmula:C16H19BrN2
    Forma y color:Solid
    Peso molecular:319.24

    Ref: TM-T60843

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Harman hydrochloride

    CAS:
    Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.
    Fórmula:C12H11ClN2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:218.68

    Ref: TM-T3158L

    10mg
    43,00€
    25mg
    70,00€
    50mg
    97,00€
    100mg
    137,00€
    200mg
    208,00€
    1mL*10mM (DMSO)
    34,00€
  • Ursulcholic acid

    CAS:
    Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
    Fórmula:C24H40O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:552.7

    Ref: TM-T68019

    5mg
    46,00€
    10mg
    58,00€
    25mg
    92,00€
    50mg
    154,00€
    100mg
    227,00€
    500mg
    642,00€
  • Nor-benzetimide

    CAS:
    Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.
    Fórmula:C16H20N2O2
    Pureza:98.63%
    Forma y color:Solid
    Peso molecular:272.34

    Ref: TM-T22380

    1mg
    72,00€
    5mg
    136,00€
    10mg
    197,00€
    25mg
    324,00€
    50mg
    452,00€
    100mg
    607,00€
    200mg
    810,00€
    1mL*10mM (DMSO)
    135,00€
  • Nitrocaramiphen hydrochloride

    CAS:
    Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.
    Fórmula:C18H27ClN2O4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:370.87

    Ref: TM-T23071

    5mg
    35,00€
    10mg
    52,00€
    25mg
    95,00€
    50mg
    154,00€
    100mg
    219,00€
    200mg
    313,00€
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Fórmula:C32H44Br2N4O4
    Pureza:95.56%
    Forma y color:Solid
    Peso molecular:708.52

    Ref: TM-T23524

    2mg
    34,00€
    5mg
    50,00€
    10mg
    80,00€
    25mg
    156,00€
    50mg
    245,00€
    100mg
    364,00€
    200mg
    517,00€
  • PSEM 89S TFA

    CAS:
    <p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>
    Fórmula:C18H23F3N2O5
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:404.38

    Ref: TM-T8552

    5mg
    48,00€
    10mg
    72,00€
    25mg
    123,00€
    50mg
    185,00€
    100mg
    274,00€
    200mg
    386,00€
  • CCMI

    CAS:
    CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.
    Fórmula:C19H15Cl2N3O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:388.25

    Ref: TM-T7422

    2mg
    39,00€
    5mg
    52,00€
    10mg
    88,00€
    25mg
    135,00€
    50mg
    187,00€
    1mL*10mM (DMSO)
    59,00€
  • Glycopyrrolate

    CAS:
    Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.
    Fórmula:C19H28BrNO3
    Pureza:99.41% - 99.64%
    Forma y color:Solid
    Peso molecular:398.33

    Ref: TM-T2387

    10mg
    37,00€
    25mg
    58,00€
    50mg
    80,00€
    100mg
    97,00€
    500mg
    226,00€
    1mL*10mM (DMSO)
    34,00€
  • SEN12333

    CAS:
    SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist
    Fórmula:C20H25N3O2
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:339.43

    Ref: TM-T23348

    2mg
    39,00€
    5mg
    57,00€
    10mg
    95,00€
    25mg
    167,00€
    50mg
    269,00€
    100mg
    432,00€
    200mg
    622,00€
    1mL*10mM (DMSO)
    63,00€
  • 9-Ethyladenine

    CAS:
    9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
    Fórmula:C7H9N5
    Pureza:99.35% - 99.37%
    Forma y color:Solid
    Peso molecular:163.18

    Ref: TM-T14065

    100mg
    34,00€
    1mL*10mM (DMSO)
    34,00€
  • BQCA

    CAS:
    <p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>
    Fórmula:C18H15NO4
    Pureza:97.22%
    Forma y color:Solid
    Peso molecular:309.32

    Ref: TM-T3993

    10mg
    44,00€
    25mg
    88,00€
    50mg
    145,00€
    100mg
    255,00€
    200mg
    376,00€
  • PNU-282987 S enantiomer free base

    CAS:
    PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).
    Fórmula:C14H17ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:264.75

    Ref: TM-T7695

    1mg
    74,00€
    5mg
    170,00€
    10mg
    230,00€
    25mg
    356,00€
    50mg
    487,00€
    100mg
    658,00€
    200mg
    884,00€
    1mL*10mM (DMSO)
    190,00€
  • 4BP-TQS

    CAS:
    4BP-TQS is an allosteric agonist of α7 nAChRs.
    Fórmula:C18H17BrN2O2S
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:405.31

    Ref: TM-T8868

    10mg
    48,00€
    25mg
    88,00€
    50mg
    139,00€
    100mg
    215,00€
    200mg
    304,00€
    1mL*10mM (DMSO)
    35,00€
  • TBPB

    CAS:
    <p>TBPB is an allosteric M1 mAChR agonist.</p>
    Fórmula:C25H32N4O
    Pureza:97.87% - 99.9%
    Forma y color:Solid
    Peso molecular:404.55

    Ref: TM-T1760

    5mg
    47,00€
    10mg
    70,00€
    25mg
    116,00€
    50mg
    187,00€
    100mg
    350,00€
    200mg
    522,00€