AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 623 productos de "AChR"
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Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Fórmula:C10H22ClNForma y color:SolidPeso molecular:191.74EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Fórmula:C30H36Br2N4O2Pureza:99.48%Forma y color:SolidPeso molecular:644.4Ref: TM-T7955
1mg92,00€2mg120,00€5mg187,00€10mg274,00€25mg472,00€50mg655,00€100mg924,00€200mg1.225,00€1mL*10mM (DMSO)278,00€Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Fórmula:C31H44N2O5SPureza:98.85% - 99.99%Forma y color:SolidPeso molecular:556.76Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Fórmula:C10H21NPureza:98.18% - 99.28%Forma y color:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Fórmula:C7H14N4O3Pureza:99.89%Forma y color:White Crystalline PowderPeso molecular:202.21Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Fórmula:C22H32BrNO5Pureza:98.85%Forma y color:SolidPeso molecular:470.4Ref: TM-T28827
1mg74,00€5mg160,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€1mL*10mM (DMSO)165,00€Simufilam dihydrochloride
CAS:Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Fórmula:C15H23Cl2N3OPureza:98.83%Forma y color:SolidPeso molecular:332.3Ref: TM-T9172
1mg52,00€5mg90,00€10mg143,00€25mg294,00€50mg380,00€100mg497,00€200mg655,00€1mL*10mM (DMSO)101,00€Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Fórmula:C13H13N3·C4H6O6Pureza:98.23% - 98.32%Forma y color:Tan SolidPeso molecular:361.35JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.72%Forma y color:SolidPeso molecular:358.84Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Fórmula:C6H8ClN5O2SPureza:99.71% - 99.87%Forma y color:Solid PowderPeso molecular:249.68Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Forma y color:SolidPeso molecular:495.58α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Forma y color:SolidPeso molecular:1770.99VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Forma y color:SolidPeso molecular:369.89Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Forma y color:SolidPeso molecular:359.89KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Fórmula:C17H15BrN4O2SPureza:98.43%Forma y color:SolidPeso molecular:419.3Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Fórmula:C40H42ClN5O7Pureza:97.94% - 98.4%Forma y color:SolidPeso molecular:740.24Anisotropine Methylbromide
CAS:Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.Fórmula:C17H32BrNO2Pureza:99.73%Forma y color:Crystals From Acetone SolidPeso molecular:362.35Cyclodrine hydrochloride
CAS:Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study ofFórmula:C19H30ClNO3Pureza:98.59%Forma y color:SolidPeso molecular:355.9Umeclidinium bromide
CAS:Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.Fórmula:C29H34BrNO2Pureza:98.4% - 99.89%Forma y color:SolidPeso molecular:508.49Ref: TM-T4997
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg212,00€50mg350,00€100mg525,00€1mL*10mM (DMSO)87,00€PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Fórmula:C18H23F3N2O5Pureza:99.9%Forma y color:SolidPeso molecular:404.38PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Forma y color:SolidPeso molecular:288.34Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Fórmula:C19H23NOPureza:99.87%Forma y color:SolidPeso molecular:281.39PNU-120596
CAS:<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Fórmula:C13H14ClN3O4Pureza:99.82%Forma y color:SolidPeso molecular:311.72VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Forma y color:SolidPeso molecular:351.28Ipratropium Bromide
CAS:Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Fórmula:C20H30BrNO3Pureza:99.92%Forma y color:SolidPeso molecular:412.37SQ22536
CAS:SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.Fórmula:C9H11N5OPureza:99.18%Forma y color:Off-White SolidPeso molecular:205.22Ref: TM-T2172
2mg35,00€5mg51,00€10mg79,00€25mg160,00€50mg274,00€100mg411,00€200mg615,00€1mL*10mM (DMSO)57,00€Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Fórmula:C21H28BrNO3Pureza:99.29%Forma y color:SolidPeso molecular:422.36OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Fórmula:C18H22N2O2SPureza:99.58%Forma y color:SolidPeso molecular:330.44JHU37160
CAS:JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.87%Forma y color:SolidPeso molecular:358.84Varenicline dihydrochloride
CAS:Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.Fórmula:C13H15Cl2N3Pureza:99.88% - 99.97%Forma y color:SolidPeso molecular:284.18Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Fórmula:C20H21N3OPureza:99.17%Forma y color:SolidPeso molecular:319.4Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Fórmula:C65H82N2O18S2Pureza:98.94% - 99.71%Forma y color:SolidPeso molecular:1243.49Ref: TM-T6397
10mg35,00€25mg52,00€50mg66,00€100mg100,00€200mg155,00€500mg240,00€1mL*10mM (DMSO)55,00€Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Fórmula:C11H18Cl2N2OPureza:98%Forma y color:SolidPeso molecular:265.18(-)-(S)-B-973B
CAS:<p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>Fórmula:C24H26F2N6OPureza:99.52%Forma y color:SolidPeso molecular:452.5Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Fórmula:C19H20ClFN2O2Pureza:99.65%Forma y color:SolidPeso molecular:362.83Ref: TM-T9771
1mg49,00€5mg101,00€10mg164,00€25mg285,00€50mg391,00€100mg552,00€200mg725,00€1mL*10mM (DMSO)111,00€AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Fórmula:C20H27N3OSPureza:98.62% - 99.89%Forma y color:SolidPeso molecular:357.51Xanomeline tartrate
CAS:Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。Fórmula:C18H29N3O7SPureza:99.19% - 99.99%Forma y color:SolidPeso molecular:431.5Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Fórmula:C20H13F6N3O2SPureza:99.83%Forma y color:White PowderPeso molecular:473.39Ref: TM-T16126
1mg87,00€5mg250,00€10mg359,00€25mg707,00€50mg1.017,00€100mg1.454,00€1mL*10mM (DMSO)274,00€Mepenzolate Bromide
CAS:Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.Fórmula:C21H26BrNO3Pureza:95.73% - 99.21%Forma y color:SolidPeso molecular:420.34Pipecuronium bromide
CAS:Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.Fórmula:C35H62Br2N4O4Pureza:>99.99%Forma y color:PowderPeso molecular:762.7Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Fórmula:C20H31NO3Pureza:97.11%Forma y color:SolidPeso molecular:333.47Varenicline
CAS:Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.Fórmula:C13H13N3Pureza:99.76%Forma y color:SolidPeso molecular:211.26Ref: TM-T4246L
2mg35,00€5mg52,00€10mg80,00€25mg144,00€50mg210,00€100mg329,00€200mg490,00€1mL*10mM (DMSO)58,00€Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46Pyrantel
CAS:Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.Fórmula:C11H14N2SPureza:98%Forma y color:Crystals From Methanol Yellowish Crystalline PowderPeso molecular:206.31Atropine hydrobromide
CAS:Atropine hydrobromide is a biochemical.Fórmula:C17H24BrNO3Forma y color:SolidPeso molecular:370.28Anatabine dicitrate
Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.Fórmula:C22H28N2O14Pureza:98%Forma y color:SolidPeso molecular:544.46(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Fórmula:C17H20D3NO3Peso molecular:292.39N-Biotinyl p-aminophenyl arsenic acid
CAS:N-Biotinyl p-aminophenyl arsenic acid is a bifunctional reagent that binds to streptavidin and disulfide compounds. It diminishes the binding sites of rbungarotoxin on reduced nicotinic receptors with an IC50 ranging from 10-300 nM, thus shielding the receptors from irreversible alkylation by bromoacetylcholine.Fórmula:C16H22AsN3O4SForma y color:SolidPeso molecular:427.35Azacyclonol hydrochloride
CAS:Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.Fórmula:C18H22ClNOForma y color:Off White Crystalline PowderPeso molecular:303.83VU0029767
CAS:<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Fórmula:C21H21N3O3Forma y color:SolidPeso molecular:363.41Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Fórmula:C107H173N37O26SPureza:98%Forma y color:SolidPeso molecular:2425.84Diphenidol
CAS:Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.Fórmula:C21H27NOForma y color:Needles From Petroleum Ether SolidPeso molecular:309.45Dianicline dihydrochloride
CAS:Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28Aprofene
CAS:Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.Fórmula:C21H27NO2Forma y color:SolidPeso molecular:325.44AN317
CAS:AN317 is a selective agonist for the nicotinic acetylcholine receptor (nAChR) containing α6β2, with dissociation constants (Ki) of 6.2 nM and 4.1 nM for the α6/α3β2β3 and α4β2 receptor subtypes, respectively. It induces dopamine release in rat striatal synaptosomes, enhances the activity of dopaminergic neurons in the substantia nigra, and exhibits protective effects against the dopaminergic neurotoxin MPP+ in rat neurons. AN317 also demonstrates favorable pharmacokinetic properties in rats and permeability across the blood-brain barrier (BB).Fórmula:C13H19N3Forma y color:SolidPeso molecular:217.31Biperiden lactate
CAS:<p>Biperiden lactate is a biochemical.</p>Fórmula:C24H35NO4Forma y color:SolidPeso molecular:401.54Phenglutarimide hydrochloride
CAS:Phenglutarimide hydrochloride is an anticholinergic. It is used as an antiparkinsonian agent.Fórmula:C17H25ClN2O2Forma y color:SolidPeso molecular:324.85Oxantel
CAS:Oxantel is a fumarate reductase inhibitor with anthelmintic activity.Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28Sulindac sulfide
CAS:Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.Fórmula:C20H17FO2SPureza:99.35%Forma y color:SolidPeso molecular:340.41Rispenzepine
CAS:Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.Fórmula:C19H20N4O2Pureza:98%Forma y color:SolidPeso molecular:336.39Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Fórmula:C19H32N2O2·2HClPureza:98%Forma y color:SolidPeso molecular:393.4Revatropate
CAS:Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.Fórmula:C19H27NO4SForma y color:SolidPeso molecular:365.49(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Fórmula:C24H17ClF2N2O2Pureza:99.82%Forma y color:SolidPeso molecular:438.85SR 16584
CAS:α3β4 nAChR antagonistFórmula:C17H22N2OPureza:99.84%Forma y color:SolidPeso molecular:270.37Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Fórmula:C15H32N2·2C4H5O6Pureza:98%Forma y color:SolidPeso molecular:538.6AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Fórmula:C27H38N6O2Pureza:98%Forma y color:SolidPeso molecular:478.63Pozanicline
CAS:<p>Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.</p>Fórmula:C11H16N2OPureza:98%Forma y color:SolidPeso molecular:192.26T761-0184
CAS:T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].Fórmula:C16H20FN3OForma y color:SolidPeso molecular:289.35CB-6673567
CAS:CB-6673567 is a selective inhibitor of adenylyl cyclase.Fórmula:C19H14N4O3Forma y color:SolidPeso molecular:346.34NGX-267
CAS:NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.Fórmula:C10H18N2OSForma y color:SolidPeso molecular:214.33Dac 5945
CAS:DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.Fórmula:C19H30ClN3OPureza:98%Forma y color:SolidPeso molecular:351.91Hexocyclium metilsulfate
CAS:Hexocyclium metilsulfate has anti-gastric secretory effects in humans.Fórmula:C21H36N2O5SPureza:98%Forma y color:SolidPeso molecular:428.59S-(+)-Mecamylamine hydrochloride
CAS:Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.Fórmula:C11H22ClNForma y color:SolidPeso molecular:203.75GS 283
CAS:GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.Fórmula:C17H17NO3Forma y color:SolidPeso molecular:283.32(R)-VU 6008667
CAS:(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).Fórmula:C24H17ClF2N2O2Forma y color:SolidPeso molecular:438.85Anisodine hydrobromide
CAS:Anisodine hydrobromide is an inhibitor of adenosine kinase.Fórmula:C17H22BrNO5Forma y color:White Crystals Or Crystalline PowderPeso molecular:400.27Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Fórmula:C21H26ClN3OSForma y color:SolidPeso molecular:403.97Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Fórmula:C17H24BrNO3Pureza:98%Forma y color:SolidPeso molecular:370.28Sazetidine A dihydrochloride
CAS:α4β2 nicotinic acetylcholine receptor ligandFórmula:C15H21ClN2O2Pureza:98%Forma y color:SolidPeso molecular:296.79FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Fórmula:C12H16FN3O3SForma y color:SolidPeso molecular:301.34Prifuroline
CAS:Prifuroline is an agent of antiarrhythmic.Fórmula:C14H16N2OPureza:98%Forma y color:SolidPeso molecular:228.29Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Fórmula:C11H15Cl3N2Pureza:98%Forma y color:SolidPeso molecular:281.61Flutropium Bromide
CAS:Flutropium Bromide is a competitive antagonist of acetylcholine. It is used to treat asthma and chronic obstructive pulmonary.Fórmula:C24H29BrFNO3Pureza:98%Forma y color:SolidPeso molecular:478.39Vesamicol
CAS:Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.Fórmula:C17H25NOPureza:98%Forma y color:SolidPeso molecular:259.39Siltenzepine
CAS:Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.Fórmula:C19H20ClN3O4Pureza:98%Forma y color:SolidPeso molecular:389.83Flupyrimin
CAS:Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].Fórmula:C13H9ClF3N3OForma y color:SolidPeso molecular:315.68VMY-2-95
CAS:VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.Fórmula:C17H16N2OForma y color:SolidPeso molecular:264.32Arecaidine propargyl ester tosylate
CAS:Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.Fórmula:C17H21NO5SPureza:98%Forma y color:SolidPeso molecular:351.42Adenylyl cyclase type 2 agonist-1
CAS:Potent AC2 agonist with an EC50 of 90 nM, potential for respiratory disease treatment.Fórmula:C27H17BrClNO5Forma y color:SolidPeso molecular:550.78CP-601927
CAS:CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.Fórmula:C12H12F3NForma y color:SolidPeso molecular:227.23RJR-2403 oxalate
CAS:RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.Fórmula:C14H18N2O4Pureza:98%Forma y color:SolidPeso molecular:278.308Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Fórmula:C32H44N4O3Pureza:98%Forma y color:SolidPeso molecular:532.72ML375
CAS:ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).Fórmula:C23H15ClF2N2O2Forma y color:SolidPeso molecular:424.83AZD 0328
CAS:AZD 0328 is a nicotinic receptor agonist for α7 neurons.Fórmula:C13H16N2OForma y color:SolidPeso molecular:216.28Nelonicline citrate
CAS:Nelonicline citrate (ABT-126) is a selective α7 nAChR agonist with a Ki of 12.3 nM, studied for schizophrenia and Alzheimer's.Fórmula:C23H27N3O8SForma y color:SolidPeso molecular:505.54Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Fórmula:C37H61BrN2O4Pureza:98%Forma y color:SolidPeso molecular:677.8Rivanicline
CAS:Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.Fórmula:C10H14N2Pureza:98%Forma y color:SolidPeso molecular:162.23VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Fórmula:C24H17ClF2N2O2Pureza:98%Forma y color:SolidPeso molecular:438.85N-0861 racemate
CAS:N-0861 racemate is the racemate of N-0861.Fórmula:C13H17N5Pureza:98%Forma y color:SolidPeso molecular:243.31Bradanicline
CAS:Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.Fórmula:C22H23N3O2Forma y color:SolidPeso molecular:361.44
