AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Fórmula:C23H33IN2OPureza:99.67%Forma y color:SolidPeso molecular:480.43Mc-Val-Ala-PAB
CAS:<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Fórmula:C25H34N4O6Pureza:98.34% - 99.24%Forma y color:SolidPeso molecular:486.56Donepezil Hydrochloride
CAS:<p>Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).</p>Fórmula:C24H29NO3·HClPureza:99.55% - 99.8%Forma y color:White To Off-White Crystalline SolidPeso molecular:415.96Nitenpyram
CAS:<p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>Fórmula:C11H15ClN4O2Pureza:99.03%Forma y color:Light-Yellow CrystalPeso molecular:270.72Mecamylamine hydrochloride
CAS:<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Fórmula:C11H22ClNPureza:99.76% - >99.99%Forma y color:White SolidPeso molecular:203.75Solifenacin hydrochloride
CAS:<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:398.93Encenicline
CAS:<p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>Fórmula:C16H17ClN2OSPureza:99.20%Forma y color:SolidPeso molecular:320.84Harman hydrochloride
CAS:<p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>Fórmula:C12H11ClN2Pureza:99.35%Forma y color:SolidPeso molecular:218.68Oxyphencyclimine Hydrochloride
CAS:<p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>Fórmula:C20H29ClN2O3Pureza:99.55%Forma y color:SolidPeso molecular:380.91Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Fórmula:C11H21NForma y color:SolidPeso molecular:167.29Propiverine
CAS:<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.48NS 1738
CAS:<p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>Fórmula:C14H9Cl2F3N2O2Pureza:99.11%Forma y color:SolidPeso molecular:365.13Mivacurium dichloride
CAS:<p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Forma y color:Off-White SolidPeso molecular:1100.17Fesoterodine
CAS:<p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>Fórmula:C26H37NO3Pureza:97.1%Forma y color:SolidPeso molecular:411.58Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Fórmula:C21H34BrNO3Pureza:98.96%Forma y color:SolidPeso molecular:428.404Cyclopentolate Hydrochloride
CAS:<p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>Fórmula:C17H26ClNO3Pureza:99.91%Forma y color:SolidPeso molecular:327.85A-867744
CAS:<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Fórmula:C20H19ClN2O3SPureza:95.66%Forma y color:SolidPeso molecular:402.89DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Fórmula:C19H23Cl2N3Pureza:99.91%Forma y color:SolidPeso molecular:364.31Propantheline
CAS:<p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>Fórmula:C23H30NO3Forma y color:SolidPeso molecular:368.49MC-Val-Cit-PABC-PNP
CAS:<p>MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.</p>Fórmula:C35H43N7O11Pureza:97.2% - 98.055%Forma y color:SolidPeso molecular:737.76
