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AChR

AChR

Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.

Se han encontrado 575 productos de "AChR"

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  • Benzetimide hydrochloride

    CAS:
    <p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>
    Fórmula:C23H27ClN2O2
    Pureza:99.32%
    Forma y color:Off-White Powder
    Peso molecular:398.93
  • mAChR-IN-1 hydrochloride

    CAS:
    <p>mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.</p>
    Fórmula:C23H26ClIN2O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:524.82
  • Pirmenol

    CAS:
    <p>Pirmenol is a new antiarrhythmic drug</p>
    Fórmula:C22H30N2O
    Pureza:97.24%
    Forma y color:Solid
    Peso molecular:338.49
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Fórmula:C22H21O2P
    Pureza:97.985%
    Forma y color:White Or Slight Yellow Powder
    Peso molecular:348.37
  • LY2119620

    CAS:
    <p>LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.</p>
    Fórmula:C19H24ClN5O3S
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:437.94
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Fórmula:C19H23Cl2N3
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:364.31
  • KH7

    CAS:
    <p>KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.</p>
    Fórmula:C17H15BrN4O2S
    Pureza:98.43%
    Forma y color:Solid
    Peso molecular:419.3
  • Ilmetropium iodide

    CAS:
    <p>Ilmetropium iodide is a bronchodilator.</p>
    Fórmula:C20H30INO3
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:459.36
  • Brompheniramine

    CAS:
    <p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>
    Fórmula:C16H19BrN2
    Forma y color:Solid
    Peso molecular:319.24
  • Darifenacin

    CAS:
    <p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>
    Fórmula:C28H30N2O2
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:426.55
  • Nor-benzetimide

    CAS:
    <p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>
    Fórmula:C16H20N2O2
    Pureza:98.63%
    Forma y color:Solid
    Peso molecular:272.34
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Fórmula:C32H44Br2N4O4
    Pureza:95.56%
    Forma y color:Solid
    Peso molecular:708.52
  • Ursulcholic acid

    CAS:
    <p>Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.</p>
    Fórmula:C24H40O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:552.7
  • Mivacurium dichloride

    CAS:
    <p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>
    Fórmula:C58H80Cl2N2O14
    Pureza:99.2% - 99.48%
    Forma y color:Off-White Solid
    Peso molecular:1100.17
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Fórmula:C19H15Cl2N3O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:388.25
  • Glycopyrrolate

    CAS:
    <p>Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.</p>
    Fórmula:C19H28BrNO3
    Pureza:99.41% - 99.64%
    Forma y color:Solid
    Peso molecular:398.33
  • Nitrocaramiphen hydrochloride

    CAS:
    <p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>
    Fórmula:C18H27ClN2O4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:370.87
  • Fesoterodine

    CAS:
    <p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>
    Fórmula:C26H37NO3
    Pureza:97.1%
    Forma y color:Solid
    Peso molecular:411.58
  • Batefenterol

    CAS:
    <p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>
    Fórmula:C40H42ClN5O7
    Pureza:97.94% - 98.4%
    Forma y color:Solid
    Peso molecular:740.24
  • 9-Ethyladenine

    CAS:
    <p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>
    Fórmula:C7H9N5
    Pureza:99.35% - 99.41%
    Forma y color:Solid
    Peso molecular:163.18