AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Fórmula:C18H23F3N2O5Pureza:99.9%Forma y color:SolidPeso molecular:404.38Monepantel
CAS:<p>Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.</p>Fórmula:C20H13F6N3O2SPureza:99.83%Forma y color:White PowderPeso molecular:473.39AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Fórmula:C20H27N3OSPureza:98.62% - 99.89%Forma y color:SolidPeso molecular:357.51Pipecuronium bromide
CAS:<p>Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.</p>Fórmula:C35H62Br2N4O4Pureza:>99.99%Forma y color:PowderPeso molecular:762.7Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Fórmula:C20H31NO3Pureza:97.11%Forma y color:SolidPeso molecular:333.47Velufenacin
CAS:<p>Velufenacin is an antagonist of muscarinic receptor[1].</p>Fórmula:C19H20ClFN2O2Pureza:99.65%Forma y color:SolidPeso molecular:362.83Xanomeline tartrate
CAS:<p>Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。</p>Fórmula:C18H29N3O7SPureza:99.19%Forma y color:SolidPeso molecular:431.5Mepenzolate Bromide
CAS:<p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>Fórmula:C21H26BrNO3Pureza:95.73% - 99.21%Forma y color:SolidPeso molecular:420.34Varenicline
CAS:<p>Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.</p>Fórmula:C13H13N3Pureza:99.76%Forma y color:SolidPeso molecular:211.26Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46Anatabine dicitrate
Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.Fórmula:C22H28N2O14Pureza:98%Forma y color:SolidPeso molecular:544.46Pyrantel
CAS:<p>Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.</p>Fórmula:C11H14N2SPureza:98%Forma y color:Crystals From Methanol Yellowish Crystalline PowderPeso molecular:206.31Atropine hydrobromide
CAS:<p>Atropine hydrobromide is a biochemical.</p>Fórmula:C17H24BrNO3Forma y color:SolidPeso molecular:370.28(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Fórmula:C17H20D3NO3Peso molecular:292.39Azacyclonol hydrochloride
CAS:<p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>Fórmula:C18H22ClNOForma y color:Off White Crystalline PowderPeso molecular:303.83Oxantel
CAS:<p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Fórmula:C21H27NOForma y color:Needles From Petroleum Ether SolidPeso molecular:309.45Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Fórmula:C107H173N37O26SPureza:98%Forma y color:SolidPeso molecular:2425.84Dianicline dihydrochloride
CAS:<p>Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.</p>Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28VU0029767
CAS:<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Fórmula:C21H21N3O3Forma y color:SolidPeso molecular:363.41
