AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Fórmula:C58H73F6N11O14S2Forma y color:SolidPeso molecular:1326.39[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Fórmula:C82H120N20O25Forma y color:SolidPeso molecular:1785.95Small Cardioactive Peptide B (SCPB)
CAS:<p>SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).</p>Fórmula:C52H80N14O11S2Pureza:98%Forma y color:SolidPeso molecular:1141.41(-)-OPC-51803
CAS:<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Fórmula:C26H32ClN3O2Pureza:98.73% - 99.59%Forma y color:SoildPeso molecular:454LtIA-F
<p>LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.</p>Fórmula:C86H121N25O22S4Forma y color:SolidPeso molecular:1985.31Aceclidine (hydrochloride)
CAS:<p>agonist of muscarinic receptors</p>Fórmula:C9H16ClNO2Pureza:98%Forma y color:SolidPeso molecular:205.68R-(+)-Cotinine
CAS:<p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>Fórmula:C10H12N2OForma y color:SolidPeso molecular:176.22nAChR modulator-2
CAS:<p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Fórmula:C12H8ClN3O2Forma y color:SolidPeso molecular:261.66nAChR modulator-1
CAS:<p>nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Fórmula:C12H8ClN3O2Forma y color:SolidPeso molecular:261.66Octamylamine
CAS:<p>Octamylamine is a bioactive chemical.</p>Fórmula:C13H29NForma y color:SolidPeso molecular:199.3761sabcomeline
CAS:<p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>Fórmula:C10H15N3OForma y color:SolidPeso molecular:193.25Bencycloquidium Bromide
CAS:<p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>Fórmula:C21H32BrNO2Forma y color:SolidPeso molecular:410.39nAChR agonist 2
CAS:<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Fórmula:C11H16N2Forma y color:SolidPeso molecular:176.263NNC 11-1607
CAS:<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Fórmula:C30H32N6O2S2Forma y color:SolidPeso molecular:572.74(Rac)-5-Carboxy tolterodine
CAS:<p>(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C22H29NO3Forma y color:SolidPeso molecular:355.47Perindoprilat
CAS:<p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>Fórmula:C17H28N2O5Pureza:99.48%Forma y color:SolidPeso molecular:340.41Methylatropine (nitrate)
CAS:<p>Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>Fórmula:C18H26N2O6Forma y color:SolidPeso molecular:366.414Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Forma y color:SolidPeso molecular:926.09M4 mAChR agonist-1
CAS:<p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).</p>Fórmula:C14H18N4OSPureza:99.14%Forma y color:SolidPeso molecular:290.38Epiboxidine
CAS:<p>Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.</p>Fórmula:C10H14N2OForma y color:SolidPeso molecular:178.23
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