AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Orphenadrine Citrate
CAS:<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Fórmula:C18H23NO·C6H8O7Pureza:98% - 99.58%Forma y color:White SolidPeso molecular:461.5Ipratropium bromide monohydrate
CAS:<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Fórmula:C20H32BrNO4Pureza:97.85%Forma y color:SolidPeso molecular:430.38Gallamine triethiodide
CAS:<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Fórmula:C30H60I3N3O3Pureza:98.90%Forma y color:White Amorphous Powder SolidPeso molecular:891.53Nicardipine hydrochloride
CAS:<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Fórmula:C26H30ClN3O6Pureza:99.58% - 99.89%Forma y color:Yellow SolidPeso molecular:515.99Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Fórmula:C18H30ClN3O5Pureza:99.53% - 99.61%Forma y color:White SolidPeso molecular:403.91Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Fórmula:C22H22FN3O2Pureza:97.16% - 98%Forma y color:SolidPeso molecular:379.43DL-trihexyphenidyl hydrochloride
CAS:<p>DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.</p>Fórmula:C20H32ClNOPureza:99.63% - 99.71%Forma y color:SolidPeso molecular:337.93Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Fórmula:C19H36ClNO2Pureza:99.81%Forma y color:SolidPeso molecular:345.95Nebracetam hydrochloride
CAS:<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Fórmula:C12H17ClN2OPureza:99.23%Forma y color:SolidPeso molecular:240.729MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.48Homatropine Methylbromide
CAS:<p>Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with antimuscarinic properties.</p>Fórmula:C17H24BrNO3Pureza:98.97%Forma y color:SolidPeso molecular:370.29Acetamiprid
CAS:<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Fórmula:C10H11ClN4Pureza:99.66%Forma y color:White PowderPeso molecular:222.67Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Fórmula:C16H20O6P2S3Pureza:≥95%Forma y color:White Crystalline Solid Or LiquidPeso molecular:466.47Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Forma y color:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Methscopolamine
CAS:<p>Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.</p>Fórmula:C18H24BrNO4Pureza:99.12% - ≥98%Forma y color:SolidPeso molecular:398.29Valethamate bromide
CAS:<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Fórmula:C19H32BrNO2Pureza:>99.99%Forma y color:SolidPeso molecular:386.37Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59Diphenmanil methylsulfate
CAS:<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Fórmula:C20H24N·CH3O4SPureza:98% - 99.27%Forma y color:SolidPeso molecular:389.51Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Fórmula:C14H18N2O2Pureza:97.37%Forma y color:White To Off-White Crystalline PowderPeso molecular:246.3Procainamide hydrochloride
CAS:<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Fórmula:C13H21N3O·HClPureza:99.83% - 99.97%Forma y color:White To Slightly Yellow PowderPeso molecular:271.79Trospium chloride
CAS:<p>Trospium chloride treats urinary incontinence without causing liver damage.</p>Fórmula:C25H30ClNO3Pureza:99.84% - >99.99%Forma y color:White To Off-White PowderPeso molecular:427.964Neostigmine methyl sulfate
CAS:<p>Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.</p>Fórmula:C13H22N2O6SPureza:99.34% - 99.53%Forma y color:Crystalline SolidPeso molecular:334.39Dipivefrin hydrochloride
CAS:<p>Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.</p>Fórmula:C19H27NO5·HClPureza:99.22% - 99.92%Forma y color:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorPeso molecular:387.9Methacholine Chloride
CAS:<p>Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of acetylcholine.</p>Fórmula:C8H18ClNO2Pureza:99.37% - 99.74%Forma y color:White Hygroscopic Crystals With Slight Odor Of Dead FishPeso molecular:195.69PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Fórmula:C36H51Cl3N4O7SPureza:99.85%Forma y color:SolidPeso molecular:790.24Adiphenine hydrochloride
CAS:<p>Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.</p>Fórmula:C20H25NO2·HClPureza:97.76% - 99.53%Forma y color:White Or Almost White PowderPeso molecular:347.88Benzethonium chloride
CAS:<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Fórmula:C27H42ClNO2Pureza:99.91%Forma y color:White To Off-White Solid Solid Particulate/PowderPeso molecular:448.09VU 0365114
CAS:<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Fórmula:C22H14F3NO3Pureza:99.86%Forma y color:SolidPeso molecular:397.35Rivastigmine tartrate
CAS:<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Fórmula:C14H22N2O2·C4H6O6Pureza:98% - 99.66%Forma y color:White To Off-White PowderPeso molecular:400.43Zelminemab
CAS:<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Pureza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Forma y color:LiquidPyrantel tartrate
CAS:<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Fórmula:C15H20N2O6SPureza:99.96%Forma y color:White CrystalsPeso molecular:356.39Pirenzepine dihydrochloride
CAS:<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:White PowderPeso molecular:424.32Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Bethanechol chloride
CAS:<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Fórmula:C7H17N2O2·ClPureza:95% - 99.73%Forma y color:White CrystallinePeso molecular:196.68Deschloroclozapine
CAS:<p>Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.</p>Fórmula:C18H20N4Pureza:99.61% - 99.98%Forma y color:SolidPeso molecular:292.38Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Fórmula:C48H69N13O14S2Pureza:98.08%Forma y color:SolidPeso molecular:1116.28Fesoterodine fumarate
CAS:<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Fórmula:C26H37NO3·C4H4O4Pureza:99.16%Forma y color:White SolidPeso molecular:527.65Vecuronium bromide
CAS:<p>Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking agent, with muscle</p>Fórmula:C34H57BrN2O4Pureza:99.63% - 99.92%Forma y color:White PowderPeso molecular:637.73Pancuronium dibromide
CAS:<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Fórmula:C35H60Br2N2O4Pureza:99.86%Forma y color:solidPeso molecular:732.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Fórmula:C32H53BrN2O4Pureza:99.77% - >99.99%Forma y color:White Or Off-White PowderPeso molecular:609.68TAK-071
CAS:<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Fórmula:C24H24FN3O3Pureza:98.02%Forma y color:SolidPeso molecular:421.46nAChR agonist 1
CAS:<p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>Fórmula:C20H18ClNO3S2Pureza:97.59%Forma y color:SolidPeso molecular:419.94Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Fórmula:C34H30N2O6SPureza:99.71%Peso molecular:594.699-Cyclopentyladenine
CAS:<p>9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signaling</p>Fórmula:C10H13N5Pureza:99.98%Forma y color:SolidPeso molecular:203.24Clidinium bromide
CAS:<p>Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.</p>Fórmula:C22H26BrNO3Pureza:98.89% - 99.86%Forma y color:White Crystalline SolidPeso molecular:432.35Hexamethonium Bromide
CAS:<p>Hexamethonium Bromide blocks neural nicotinic AChR, poorly absorbed in the gut, doesn't pass the blood-brain barrier.</p>Fórmula:C12H30Br2N2Pureza:99.76%Forma y color:White Crystalline Powder And AgglomeratesPeso molecular:362.19Oxybutynin
CAS:<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Fórmula:C22H31NO3Pureza:97.81% - 99.57%Forma y color:White To Off-White Crystalline PowderPeso molecular:357.49Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Fórmula:C20H26ClNO3Pureza:99.03% - 99.94%Forma y color:SolidPeso molecular:363.88Flavoxate hydrochloride
CAS:<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Fórmula:C24H26ClNO4Pureza:99.78%Forma y color:White SolidPeso molecular:427.922',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Fórmula:C10H13N5O2Pureza:99.55%Forma y color:White SolidPeso molecular:235.24Fipexide
CAS:<p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>Fórmula:C20H21ClN2O4Pureza:97.6% - 99.95%Forma y color:SolidPeso molecular:388.84(Rac)-ABT-202 dihydrochloride
CAS:<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Fórmula:C9H15Cl2N3Pureza:97.4%Forma y color:SolidPeso molecular:236.142Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Fórmula:C6H15ClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:182.65Tolterodine tartrate
CAS:<p>Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.</p>Fórmula:C22H31NO·C4H6O6Pureza:99.95%Forma y color:White-To-Off-White Crystalline PowderPeso molecular:475.58Propantheline bromide
CAS:<p>Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on smooth muscle</p>Fórmula:C23H30BrNO3Pureza:98% - ≥98%Peso molecular:448.4Primidone
CAS:<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Fórmula:C12H14N2O2Pureza:99.91%Forma y color:Crystals (Ntp 1992)Peso molecular:218.25Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Fórmula:C30H40Cl2N4Pureza:99.79% - 99.9%Forma y color:SolidPeso molecular:527.59Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56Darifenacin hydrobromide
CAS:<p>Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.</p>Fórmula:C28H31BrN2O2Pureza:99.75% - >99.99%Forma y color:SolidPeso molecular:505.45SSR 180
CAS:<p>SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of Alzheimer;s disease and schizophrenia.</p>Fórmula:C14H17BrN2O2Pureza:98.82%Forma y color:SoildPeso molecular:325.20Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Fórmula:C18H26BrNO3Pureza:99.7%Forma y color:SolidPeso molecular:384.308Tazomeline
CAS:<p>Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.</p>Fórmula:C14H23N3S2Pureza:99.63%Forma y color:SolidPeso molecular:297.48V-11-0711 HCl
<p>V-11-0711 HCl is a selective and highly effective choline kinase α (ChoKα) inhibitor that inhibits the catalytic activity of Chk.</p>Fórmula:C27H36ClNO3Pureza:99.87%Forma y color:SolidPeso molecular:458.03(Rac)-Sabcomeline HCl
CAS:<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Fórmula:C10H16ClN3OPureza:99.58%Forma y color:SoildPeso molecular:229.71Cotinine
CAS:<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Fórmula:C10H12N2OPureza:98% - 99.89%Forma y color:Viscous Oil SolidPeso molecular:176.22Ribavirin
CAS:<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Fórmula:C8H12N4O5Pureza:99.09% - 99.83%Forma y color:Less Solid Colourless SolidPeso molecular:244.20Tiotropium bromide
CAS:<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Fórmula:C19H22BrNO4S2Pureza:96.82% - 99.97%Forma y color:White SolidPeso molecular:472.42DSPE-PEG1000-RVG29
<p>DSPE-PEG1000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 can specifically bind to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and cross the BBB.</p>Forma y color:Odour SolidMK-0969
CAS:<p>MK-0969 (J-104135) is a possible M3 antagonist for the treatment of chronic obstructive pulmonary disease.</p>Fórmula:C24H30F2N4O2Forma y color:SolidPeso molecular:444.52nAChR modulator-2
CAS:<p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Fórmula:C12H8ClN3O2Forma y color:SolidPeso molecular:261.66α-Muricholic acid
CAS:<p>α-Muricholic acid is the most abundant primary bile acid in rodents.</p>Fórmula:C24H40O5Pureza:98%Forma y color:SolidPeso molecular:408.57α-Conotoxin EI
CAS:<p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>Fórmula:C83H125N27O27S5Pureza:98%Forma y color:SolidPeso molecular:2093.37Octamylamine
CAS:<p>Octamylamine is a bioactive chemical.</p>Fórmula:C13H29NForma y color:SolidPeso molecular:199.3761Bencycloquidium Bromide
CAS:<p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>Fórmula:C21H32BrNO2Forma y color:SolidPeso molecular:410.39nAChR agonist CMPI hydrochloride
CAS:<p>CMPI hydrochloride: Potent α4:α4 nAChR PAM; EC50 0.26 μM for (α4)3(β2)2 response to ACh; may aid nicotine dependence, neuropsychiatric research.</p>Fórmula:C18H20Cl2N4OForma y color:SolidPeso molecular:379.29(S)-Dinotefuran
CAS:<p>(S)-Dinotefuran, a neonicotinoid, more toxic to bees than its R-isomer, targets α8 nAChR.</p>Fórmula:C7H14N4O3Forma y color:SolidPeso molecular:202.21Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Fórmula:C58H73F6N11O14S2Forma y color:SolidPeso molecular:1326.39[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Fórmula:C82H120N20O25Forma y color:SolidPeso molecular:1785.95LtIA-F
<p>LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.</p>Fórmula:C86H121N25O22S4Forma y color:SolidPeso molecular:1985.31α-Conotoxin PIA TFA
<p>α-Conotoxin PIA TFA, targeting nicotinic acetylcholine receptor (nAChR) subtypes with α6 and α3 subunits, acts as an antagonist.</p>Fórmula:C81H126F3N27O27S4Pureza:98.81%Forma y color:SolidPeso molecular:2095.3Muscarinic toxin 3
CAS:<p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>Fórmula:C319H489N89O97S8Pureza:98%Forma y color:SolidPeso molecular:7379.35DSPE-PEG5000-RVG29
<p>DSPE-PEG5000-RVG29 is a PEG compound comprised of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and facilitates passage through the BBB.</p>Forma y color:Odour Solid(-)-Coclaurine hydrochloride
CAS:<p>(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.</p>Fórmula:C17H20ClNO3Pureza:99.07%Forma y color:SoildPeso molecular:321.8Perlapine
CAS:<p>Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM).</p>Fórmula:C19H21N3Forma y color:SolidPeso molecular:291.39Atracurium
CAS:<p>Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.</p>Fórmula:C53H72N2O122Forma y color:SolidPeso molecular:929.14Anagyrine hydrochloride
CAS:<p>Anagyrine hydrochloride, a quinolizidine from Lupinus albus, targets muscarinic/nicotinic receptors; IC50: 132/2096 µM. It desensitizes nAChR directly.</p>Fórmula:C15H21ClN2OForma y color:SolidPeso molecular:280.798-Aminoadenine
CAS:<p>8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.</p>Fórmula:C5H6N6Pureza:99.82%Forma y color:SolidPeso molecular:150.14rac-Desethyl Oxybutynin (hydrochloride)
CAS:<p>rac-Desethyl oxybutynin, active oxybutynin metabolite, binds to mAChRs; K_i values 3.12-16 nM; lowers rat micturition pressure.</p>Fórmula:C20H28ClNO3Forma y color:SolidPeso molecular:365.89TMPH
CAS:<p>TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.</p>Fórmula:C16H31NO2Pureza:99.78%Forma y color:SoildPeso molecular:269.42Guanylyl Imidodiphosphate (lithium salt)
CAS:<p>Guanylyl Imidodiphosphate (lithium salt) is a non-hydrolyzable GTP analog that increases adenylate cyclase activity.</p>Fórmula:C10H13Li4N6O13P3Forma y color:SolidPeso molecular:545.93Doxacurium Chloride
CAS:<p>Doxacurium Chloride is a muscarinic acetylcholine receptor M2 antagonist.</p>Fórmula:C56H78ClN2O16Pureza:98%Forma y color:SolidPeso molecular:1070.69Epiboxidine hydrochloride
CAS:<p>Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.</p>Fórmula:C10H15ClN2OForma y color:SolidPeso molecular:214.69VU6028418
CAS:<p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>Forma y color:SolidPF-4348235 HCl
<p>PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).</p>Fórmula:C36H50Cl2N4O7SPureza:98.81%Forma y color:SolidPeso molecular:753.78R-(+)-Cotinine
CAS:<p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>Fórmula:C10H12N2OForma y color:SolidPeso molecular:176.22Cisatracurium besylate
CAS:<p>Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.</p>Fórmula:C53H72N2O12·2C6H5O3SPureza:97.89% - 99.85%Forma y color:White Or White Powder CategoryPeso molecular:1243.48Cyclodrine
CAS:<p>Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.</p>Fórmula:C19H29NO3Pureza:97.62%Forma y color:SoildPeso molecular:319.44Angiopeptin
CAS:<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Fórmula:C54H71N11O10S2Forma y color:SolidPeso molecular:1098.34Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Fórmula:C20H18O6Forma y color:SolidPeso molecular:354.358α-Bungarotoxin
CAS:<p>Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs).</p>Fórmula:C338H529N97O105S11Pureza:98%Forma y color:SolidPeso molecular:7984.14Cevimeline hydrochloride hemihydrate
CAS:<p>Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug for xerostomia in Sjogren's syndrome.</p>Fórmula:C20H38Cl2N2O3S2Pureza:97.00%Forma y color:SolidPeso molecular:489.55AC1-IN-1
CAS:<p>AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).</p>Fórmula:C18H18FN5O2Pureza:99.89%Forma y color:SolidPeso molecular:355.37ANQ-9040
CAS:<p>ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.</p>Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92Biperiden Hydrochloride
CAS:<p>Biperiden HCl is an anti-Parkinson's drug, blocks M1 receptors, manages all Parkinson's types, and is FDA-approved. Non-toxic at 0.11 mg/kg to rats' cognition.</p>Fórmula:C21H30ClNOPureza:98%Forma y color:SolidPeso molecular:347.92nAChR agonist 2
CAS:<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Fórmula:C11H16N2Forma y color:SolidPeso molecular:176.263Emraclidine
CAS:<p>Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.</p>Fórmula:C20H21F3N4OPureza:99.96%Forma y color:SolidPeso molecular:390.4TIP 39, Tuberoinfundibular Neuropeptide
CAS:<p>TIP39 is a synthetic neuropeptide agonist for human and rat PTH2 receptors from the hypothalamus.</p>Fórmula:C202H325N61O54SPureza:98%Forma y color:SolidPeso molecular:4504.2Lupanine hydrochloride
CAS:<p>Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.</p>Fórmula:C15H25ClN2OForma y color:SolidPeso molecular:284.83Pozanicline hydrochloride
<p>Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding to α7 nAChR.</p>Fórmula:C11H17ClN2OPureza:97.13% - 99.81%Forma y color:SolidPeso molecular:228.72PDE4-IN-4
CAS:<p>PDE4-IN-4 is a compound acting as both a potent M3 antagonist (p IC 50 = 10.2) and a PDE4 inhibitor (p IC 50 = 8.8), designed for inhalation-based treatment of</p>Fórmula:C36H37Cl2N3O7SForma y color:SolidPeso molecular:726.67Methylatropine (nitrate)
CAS:<p>Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>Fórmula:C18H26N2O6Forma y color:SolidPeso molecular:366.414nAChR modulator-1
CAS:<p>nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Fórmula:C12H8ClN3O2Forma y color:SolidPeso molecular:261.66Heliosupine N-oxide
<p>Heliosupine N-oxide is a useful organic compound for research related to life sciences and the catalog number is T125058.</p>Fórmula:C20H31NO8Forma y color:SolidPeso molecular:413.467Small Cardioactive Peptide B (SCPB)
CAS:<p>SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).</p>Fórmula:C52H80N14O11S2Pureza:98%Forma y color:SolidPeso molecular:1141.41Epiboxidine
CAS:<p>Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.</p>Fórmula:C10H14N2OForma y color:SolidPeso molecular:178.23M 8218
CAS:<p>M 8218 is a bioactive chemical.</p>Fórmula:C20H29NO2Forma y color:SolidPeso molecular:315.45Desfesoterodine
CAS:<p>Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.</p>Fórmula:C22H31NO2Pureza:99.77%Forma y color:SolidPeso molecular:341.49α-Conotoxin AuIB
CAS:<p>Selective antagonist of α3β4 nicotinic acetylcholine receptors.</p>Fórmula:C65H89N17O21S4Pureza:98%Forma y color:SolidPeso molecular:1572.76Flupyradifurone
CAS:<p>Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.</p>Fórmula:C12H11ClF2N2O2Pureza:99.83%Forma y color:SolidPeso molecular:288.68α-Conotoxin imi
CAS:<p>alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.</p>Fórmula:C52H78N20O15S4Pureza:98%Forma y color:SolidPeso molecular:1351.56Tiquizium
CAS:<p>Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.</p>Fórmula:C19H24NS2Pureza:99.82%Forma y color:SolidPeso molecular:330.53CVN417
<p>CVN417 is an orally active antagonist of nAChR containing the α6 subunit, modulating phasic dopaminergic neurotransmission in an impulse-dependent fashion.</p>Forma y color:Odour SolidPerindoprilat
CAS:<p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>Fórmula:C17H28N2O5Pureza:99.48%Forma y color:SolidPeso molecular:340.41Dicloromezotiaz
CAS:<p>Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.</p>Fórmula:C19H12Cl3N3O2SForma y color:SolidPeso molecular:452.74[D-Trp7,9,10]-Substance P
CAS:<p>Substance P analog that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.</p>Fórmula:C79H105N21O13SPureza:98%Forma y color:SolidPeso molecular:1588.89SIB 1553A
CAS:<p>SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.</p>Fórmula:C13H19NOSPureza:99.79%Forma y color:SoildPeso molecular:237.36(+)-Coclaurine hydrochloride
CAS:<p>(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.</p>Fórmula:C17H20ClNO3Pureza:98%Forma y color:SolidPeso molecular:321.8Destomycin A
CAS:<p>Destomycin A, an aminoglycoside antibiotic, exhibits activity against bacterial (Gram-positive and Gram-negative), antifungal, and anthelmintic agents. It inhibits peptide synthesis in Escherichia coli cells and stimulates adenylate cyclase in animal tissues.</p>Fórmula:C20H37N3O13Forma y color:SolidPeso molecular:527.52CDD0102 HCl
CAS:<p>CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.</p>Fórmula:C8H13ClN4OPureza:99.7%Forma y color:SoildPeso molecular:216.67Mant-GTPγS
CAS:<p>Mant-GTPγS, an effective GTP analog, displays strong competitive inhibition of adenylyl cyclase (AC). Additionally, it acts as a potent inhibitor of YdeH.</p>Fórmula:C18H23N6O14P3SForma y color:SolidPeso molecular:672.39Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Fórmula:C45H47N7O9S3Forma y color:SolidPeso molecular:926.09Thiothixene
CAS:<p>Thiothixene has a wide range of applications in life science related research.</p>Fórmula:C23H29N3O2S2Forma y color:SolidPeso molecular:443.62Fentonium bromide
CAS:<p>Fentonium bromide is a biochemical.</p>Fórmula:C31H34BrNO4Forma y color:SolidPeso molecular:564.51(S)-UFR2709 hydrochloride
CAS:<p>(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in rats, studies nicotine addiction.</p>Fórmula:C13H18ClNO2Pureza:98.94%Forma y color:SolidPeso molecular:255.74PF-06827443
<p>PF-06827443 is a orally bioavailable, CNS-penetrant M1-selective PAM with minimal agonist activity.</p>Fórmula:C24H24N2O4Forma y color:SolidPeso molecular:404.475-Hydroxymethyl tolterodine formate
CAS:<p>5-Hydroxymethyl tolterodine (formate) (PNU-200577 (formic)) is an active metabolite of the muscarinic acetylcholine receptor antagonists Tolterodine and Fesoterodine. It is synthesized by the cytochrome P450 (CYP) isoenzyme CYP2D6 and plasma esterases.</p>Fórmula:C23H33NO4Forma y color:SolidPeso molecular:387.51(Rac)-5-Carboxy tolterodine
CAS:<p>(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C22H29NO3Forma y color:SolidPeso molecular:355.47RuBi-Nicotine
CAS:<p>Nicotinic receptor agonist</p>Fórmula:C40H44Cl2N8RuPureza:98%Forma y color:SolidPeso molecular:808.81(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS:<p>(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.</p>Fórmula:C22H32ClNO2Forma y color:SolidPeso molecular:377.95NNC 11-1607
CAS:<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Fórmula:C30H32N6O2S2Forma y color:SolidPeso molecular:572.74N,N-Dicyclohexylcarbodiimide
CAS:<p>N,N-Dicyclohexylcarbodiimide (Dicyclohexylcarbodiimide) is a cross-linking agent used in the synthesis of active ester-containing reagents.</p>Fórmula:C13H22N2Pureza:98.28% - 99.73%Forma y color:SolidPeso molecular:206.33bPiDDB
CAS:<p>bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.</p>Fórmula:C24H38Br2N2Pureza:98.72%Forma y color:SolidPeso molecular:514.38TC-2216
CAS:<p>TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to treat anxiety and depression.</p>Fórmula:C12H17N3Pureza:99.33%Forma y color:SolidPeso molecular:203.28Irsogladine maleate
CAS:<p>Compound PDK0375, with CAS No. 84504-69-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0375 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C9H7Cl2N5Forma y color:SolidPeso molecular:256.09trans-Cevimeline hydrochloride
CAS:<p>AF 102A hydrochloride is a biochemical.</p>Fórmula:C10H18ClNOSForma y color:SolidPeso molecular:235.77Lobeline sulfate
CAS:<p>Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.</p>Fórmula:C22H29NO6SPureza:98%Forma y color:White PowderPeso molecular:435.54Hydroxybupropion
CAS:<p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>Fórmula:C13H18ClNO2Pureza:99.73%Forma y color:Off-White SolidPeso molecular:255.74Oxotremorine
CAS:<p>Oxotremorine acts as an agonist of mAChR, specifically activating the M1 and M3 acetylcholine receptors. In drug discrimination experiments with macaques, it exhibits effects similar to nicotine.</p>Fórmula:C12H18N2OForma y color:SolidPeso molecular:206.28Methyllycaconitine citrate
CAS:<p>Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.</p>Fórmula:C43H58N2O17Pureza:98.03% - 98.91%Forma y color:SolidPeso molecular:874.92G-Protein antagonist peptide
CAS:<p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>Fórmula:C57H64N12O9SPureza:98%Forma y color:SolidPeso molecular:1093.27M4 mAChR agonist-1
CAS:<p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).</p>Fórmula:C14H18N4OSPureza:99.14%Forma y color:SolidPeso molecular:290.38Muscarine
CAS:<p>Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Fórmula:C9H20NO2Pureza:98%Forma y color:SolidPeso molecular:174.26M3/PDE4 modulator-1
<p>M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.</p>Fórmula:C38H41Cl2N3O8SForma y color:SolidPeso molecular:770.725-AMAM-2-CP
CAS:<p>5-AMAM-2-CP, a significant metabolite of Acetamiprid, serves as a global insecticide within the neonicotinoid class and acts as an nAChR agonist [1] [2].</p>Fórmula:C9H11ClN2OForma y color:SolidPeso molecular:198.65(R)-Dinotefuran
CAS:<p>(R)-Dinotefuran, a neonicotinoid, is 1.7-2.4x more effective against pests like Aphis gossypii and safer for bees.</p>Fórmula:C7H14N4O3Forma y color:SolidPeso molecular:202.21Ebiratide TFA
<p>Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.</p>Fórmula:C48H73N11O10S·xC2HF3O2Forma y color:SolidPeso molecular:996.23 (free base)TDI-10229
CAS:<p>TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.</p>Fórmula:C16H16ClN5Pureza:99.85% - 99.89%Forma y color:SoildPeso molecular:313.78BTMPS
CAS:<p>BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.</p>Fórmula:C28H52N2O4Pureza:98.1%Forma y color:SolidPeso molecular:480.72Anabaseine
CAS:<p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>Fórmula:C10H12N2Forma y color:SolidPeso molecular:160.22N-Ethyl-N-(3-pyridylmethyl)amine
CAS:<p>N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.</p>Fórmula:C8H12N2Pureza:99.65%Forma y color:SolidPeso molecular:136.19Soclenicant
CAS:<p>Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availability</p>Fórmula:C24H26N4O3Pureza:99.57%Forma y color:SoildPeso molecular:418.49Rivanicline 2HCl
<p>Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.</p>Fórmula:C10H16Cl2N2Pureza:99.4%Forma y color:SoildPeso molecular:235.15Proadrenomedullin (1-20), human
CAS:<p>Endogenous peptide; agonist of MRGPRX2 (EC50=251 nM); noncompetitive inhibitor of nicotinic receptors; reduces catecholamine secretion; antihypertensive.</p>Fórmula:C112H178N36O27Pureza:98%Forma y color:SolidPeso molecular:2460.84TC-2559 difumarate
CAS:<p>TC-2559 difumarate: Oral α4β2 nAChR partial agonist, CNS-selective, EC50 0.18 μM, prefers α4β2 over α2β4/α4β4/α3β4, antinociceptive.</p>Fórmula:C20H26N2O9Forma y color:SolidPeso molecular:438.43Bensultap
CAS:<p>Bensultap is an agricultural chemical typically used as a pesticide.</p>Fórmula:C17H21NO4S4Pureza:98%Forma y color:SolidPeso molecular:431.61Ebiratide
CAS:<p>Ebiratide is an analog of ACTH 4-9.</p>Fórmula:C48H73N11O10SPureza:98%Forma y color:SolidPeso molecular:996.23GeX-2
CAS:<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Fórmula:C103H169N43O27Forma y color:SolidPeso molecular:2441.72Aceclidine (hydrochloride)
CAS:<p>agonist of muscarinic receptors</p>Fórmula:C9H16ClNO2Pureza:98%Forma y color:SolidPeso molecular:205.68Tropicamide
CAS:<p>Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for diagnostic use.</p>Fórmula:C17H20N2O2Pureza:99.78% - 99.94%Forma y color:White PowderPeso molecular:284.35Navafenterol
CAS:<p>AZD-8871, a potential COPD and asthma treatment, may work well with ICS.</p>Fórmula:C38H42N6O6S2Forma y color:SolidPeso molecular:742.91α-Conotoxin PIA
CAS:<p>Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM</p>Fórmula:C79H125N27O25S4Pureza:98%Forma y color:SolidPeso molecular:1981.3(-)-OPC-51803
CAS:<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Fórmula:C26H32ClN3O2Pureza:98.73% - 99.59%Forma y color:SoildPeso molecular:454(rel)-Asperparaline A
CAS:<p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>Fórmula:C20H29N3O3Forma y color:SolidPeso molecular:359.47sabcomeline
CAS:<p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>Fórmula:C10H15N3OForma y color:SolidPeso molecular:193.25DSPE-PEG2000-RVG29
<p>DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.</p>Forma y color:Odour SolidLu AE51090
CAS:<p>Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.</p>Fórmula:C24H29N3O3Pureza:99.57%Forma y color:SolidPeso molecular:407.515-AAM-2-CP
CAS:<p>5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.</p>Fórmula:C8H9ClN2OPureza:99.58%Forma y color:SolidPeso molecular:184.62(R)-(+)-Anatabine
CAS:<p>(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.</p>Fórmula:C10H12N2Pureza:98%Forma y color:SolidPeso molecular:160.22(Rac)-Sabcomeline
CAS:<p>(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.</p>Fórmula:C10H15N3OPureza:99.14%Forma y color:SolidPeso molecular:193.25LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Fórmula:C39H43ClN4O9S2Forma y color:SolidPeso molecular:811.36Br-PBTC
CAS:<p>Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.</p>Fórmula:C14H15BrN2OSForma y color:SolidPeso molecular:339.25β2AR/M-receptor agonist-1
CAS:<p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>Fórmula:C43H56BrN3O7Forma y color:SolidPeso molecular:806.82Dexetimide
CAS:<p>Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.</p>Fórmula:C23H26N2O2Forma y color:SolidPeso molecular:362.46Metixene hydrochloride hydrate
CAS:<p>Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.</p>Fórmula:C20H26ClNOSPureza:99.88%Forma y color:SolidPeso molecular:363.95Fipexide hydrochloride
CAS:<p>Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.</p>Fórmula:C20H22Cl2N2O4Forma y color:SolidPeso molecular:425.31NKH477
CAS:<p>NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.</p>Fórmula:C27H44ClNO8Pureza:98% - 98%Forma y color:SolidPeso molecular:546.09Tolterodine
CAS:<p>Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.</p>Fórmula:C22H31NOPureza:99.71%Forma y color:White Like Or Light Brown Crystalline PowderPeso molecular:325.49YM-58790 hydrochloride
CAS:<p>YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).</p>Fórmula:C27H32ClN3O2Pureza:98%Forma y color:SolidPeso molecular:466.02Palmatine hydroxide
CAS:<p>Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.</p>Fórmula:C21H23NO5Forma y color:SolidPeso molecular:369.41Cevimeline
CAS:<p>Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.</p>Fórmula:C10H17NOSForma y color:Off-White SolidPeso molecular:199.31Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Fórmula:C22H31ClN2OForma y color:SolidPeso molecular:374.95Varenicline Hydrochloride
CAS:<p>Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).</p>Fórmula:C13H14ClN3Pureza:99.854%Forma y color:SolidPeso molecular:247.72Cevimeline hydrochloride
CAS:<p>Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.</p>Fórmula:C10H18ClOSForma y color:SolidPeso molecular:235.77Glycerophosphoinositol choline
CAS:<p>Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.</p>Fórmula:C14H32NO12PForma y color:SolidPeso molecular:437.38Ispronicline
CAS:<p>Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitive</p>Fórmula:C14H22N2OPureza:97.70% - 99.16%Forma y color:SolidPeso molecular:234.34Sabcomeline hydrochloride
CAS:<p>Sabcomeline is a selective M1 receptor partial agonist.</p>Fórmula:C10H16ClN3OForma y color:SolidPeso molecular:229.71(±)-Darifenacin
CAS:<p>(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.</p>Fórmula:C28H30N2O2Forma y color:SolidPeso molecular:426.55VU0467485
CAS:<p>VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.</p>Fórmula:C17H17FN4O2SPureza:98%Forma y color:SolidPeso molecular:360.41Clorprenaline
CAS:<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Fórmula:C11H16ClNOPureza:98.9%Forma y color:SolidPeso molecular:213.7ABT-107
CAS:<p>ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.</p>Fórmula:C19H20N4OForma y color:SolidPeso molecular:320.396
![[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76363.webp&w=3840&q=75)
![[D-Trp7,9,10]-Substance P](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1932.webp&w=3840&q=75)
