
AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Fórmula:C22H31ClN2OForma y color:SolidPeso molecular:374.95N6-Methyladenosine 5'-monophosphate disodium salt
CAS:<p>N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.</p>Fórmula:C11H14N5Na2O7PPureza:99.36% - 99.36%Forma y color:SolidPeso molecular:405.21DL-Cystine
CAS:<p>DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .</p>Fórmula:C6H12N2O4S2Forma y color:SolidPeso molecular:240.3Solifenacin D5 hydrochloride
CAS:<p>Solifenacin D5 HCl: deuterium-labeled M1, M2, M3 muscarinic receptor antagonist with pKi 7.6, 6.9, 8.0.</p>Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:403.96Tolterodine
CAS:<p>Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.</p>Fórmula:C22H31NOPureza:99.71%Forma y color:White Like Or Light Brown Crystalline PowderPeso molecular:325.49NKH477
CAS:<p>NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.</p>Fórmula:C27H44ClNO8Pureza:98% - 98%Forma y color:SolidPeso molecular:546.09NSC 23766
CAS:<p>NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.</p>Fórmula:C24H35N7Pureza:99.49%Forma y color:SolidPeso molecular:421.58Telenzepine dihydrochloride
CAS:<p>muscarinic M1 receptor antagonist</p>Fórmula:C19H23ClN4O2SPureza:98%Forma y color:SolidPeso molecular:406.93Fipexide hydrochloride
CAS:<p>Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.</p>Fórmula:C20H22Cl2N2O4Forma y color:SolidPeso molecular:425.31SSR180711 hydrochloride
CAS:<p>SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.</p>Fórmula:C14H18BrClN2O2Pureza:99.22%Forma y color:SolidPeso molecular:361.66Clorprenaline
CAS:<p>Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.</p>Fórmula:C11H16ClNOPureza:98.9%Forma y color:SolidPeso molecular:213.7Cevimeline hydrochloride
CAS:<p>Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.</p>Fórmula:C10H18ClOSForma y color:SolidPeso molecular:235.77Cevimeline
CAS:<p>Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.</p>Fórmula:C10H17NOSForma y color:Off-White SolidPeso molecular:199.31Nanofin
CAS:<p>Nanofin (Lupetidine) is a neuropathic blocker, with antihypertensive effect.</p>Fórmula:C7H15NPureza:97.38% - 99.818%Forma y color:Clear Colorless To Slightly Yellow LiquidPeso molecular:113.2Encenicline hydrochloride
CAS:<p>Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).</p>Fórmula:C16H17ClN2OS·HClPureza:98.34% - 99.85%Forma y color:SolidPeso molecular:357.3PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Forma y color:SolidPeso molecular:288.34Tacrine hydrochloride (hydrate)
CAS:<p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>Fórmula:C13H14N2·XHCl·XH2OPureza:99.01% - 99.89%Forma y color:SolidPeso molecular:234.72NS3861
CAS:<p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>Fórmula:C12H14BrNSPureza:99.853%Forma y color:SolidPeso molecular:284.22Thiacloprid
CAS:<p>Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.</p>Fórmula:C10H9ClN4SPureza:98.66% - 99.95%Forma y color:Yellowish Crystalline PowderPeso molecular:252.72Cyclopentolate Hydrochloride
CAS:<p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>Fórmula:C17H26ClNO3Pureza:99.91%Forma y color:SolidPeso molecular:327.85A-867744
CAS:<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Fórmula:C20H19ClN2O3SPureza:95.66%Forma y color:SolidPeso molecular:402.89PSEM 89S TFA
CAS:<p>PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.</p>Fórmula:C18H23F3N2O5Pureza:99.9%Forma y color:SolidPeso molecular:404.38Mivacurium dichloride
CAS:<p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Forma y color:Off-White SolidPeso molecular:1100.17Fesoterodine
CAS:<p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>Fórmula:C26H37NO3Pureza:97.1%Forma y color:SolidPeso molecular:411.58DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Fórmula:C19H23Cl2N3Pureza:99.91%Forma y color:SolidPeso molecular:364.31Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Fórmula:C22H21O2PPureza:97.985%Forma y color:White Or Slight Yellow PowderPeso molecular:348.37NS9283
CAS:<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Fórmula:C14H8N4OPureza:99.12%Forma y color:SolidPeso molecular:248.24mAChR-IN-1 hydrochloride
CAS:<p>mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.</p>Fórmula:C23H26ClIN2O2Pureza:99.87%Forma y color:SolidPeso molecular:524.82Umeclidinium bromide
CAS:<p>Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.</p>Fórmula:C29H34BrNO2Pureza:98.4% - 99.89%Forma y color:SolidPeso molecular:508.49ST034307
CAS:<p>ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).</p>Fórmula:C10H4Cl4O2Pureza:99.28%Forma y color:SolidPeso molecular:297.95(-)-(S)-B-973B
CAS:<p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>Fórmula:C24H26F2N6OPureza:99.52%Forma y color:SolidPeso molecular:452.5Pozanicline dihydrochloride
CAS:<p>Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)</p>Fórmula:C11H18Cl2N2OPureza:98%Forma y color:SolidPeso molecular:265.18Cyclodrine hydrochloride
CAS:<p>Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of</p>Fórmula:C19H30ClNO3Pureza:98.59%Forma y color:SolidPeso molecular:355.9NS 1738
CAS:<p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>Fórmula:C14H9Cl2F3N2O2Pureza:99.11%Forma y color:SolidPeso molecular:365.13BNC210
CAS:<p>BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.</p>Fórmula:C17H23N3O3Pureza:97.05% - >99.99%Forma y color:SolidPeso molecular:317.38Harman hydrochloride
CAS:<p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>Fórmula:C12H11ClN2Pureza:99.35%Forma y color:SolidPeso molecular:218.68Nitenpyram
CAS:<p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>Fórmula:C11H15ClN4O2Pureza:99.03%Forma y color:Light-Yellow CrystalPeso molecular:270.72PHA 543613 hydrochloride
CAS:<p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>Fórmula:C15H18ClN3O2Forma y color:SolidPeso molecular:307.78VU0238441
CAS:<p>VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.</p>Fórmula:C16H9ClF3NO2Pureza:100%Forma y color:SolidPeso molecular:339.7Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Fórmula:C23H26N2O2Pureza:99.87%Forma y color:SolidPeso molecular:362.46Anisotropine Methylbromide
CAS:<p>Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm and for the suppression of gastric acid secretion.</p>Fórmula:C17H32BrNO2Pureza:99.73%Forma y color:Crystals From Acetone SolidPeso molecular:362.35Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Fórmula:C31H44N2O5SPureza:98.85% - 99.58%Forma y color:SolidPeso molecular:556.76Pempidine
CAS:<p>Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.</p>Fórmula:C10H21NPureza:98.18% - 99.28%Forma y color:Colorless - Light Yellow Clear LiquidPeso molecular:155.28Dinotefuran
CAS:<p>Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.</p>Fórmula:C7H14N4O3Pureza:99.89%Forma y color:White Crystalline PowderPeso molecular:202.21Sofpironium bromide
CAS:<p>Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.</p>Fórmula:C22H32BrNO5Pureza:98.85%Forma y color:SolidPeso molecular:470.4Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Fórmula:C13H13N3·C4H6O6Pureza:98.23% - 98.32%Forma y color:Tan SolidPeso molecular:361.35JHU37152
CAS:<p>JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.</p>Fórmula:C19H20ClFN4Pureza:99.72%Forma y color:SolidPeso molecular:358.84Clothianidin
CAS:<p>Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.</p>Fórmula:C6H8ClN5O2SPureza:99.71% - 99.87%Forma y color:Solid PowderPeso molecular:249.68Syn-Ake acetate
CAS:<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Forma y color:SolidPeso molecular:495.58α-Conotoxin MII acetate
<p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Forma y color:SolidPeso molecular:1770.99VU0357017 hydrochloride
CAS:<p>VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.</p>Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Forma y color:SolidPeso molecular:369.89Piperidolate hydrochloride
CAS:<p>Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.</p>Fórmula:C21H26ClNO2Pureza:99.5%Forma y color:SolidPeso molecular:359.89KH7
CAS:<p>KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.</p>Fórmula:C17H15BrN4O2SPureza:98.43%Forma y color:SolidPeso molecular:419.3Batefenterol
CAS:<p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>Fórmula:C40H42ClN5O7Pureza:97.94% - 98.4%Forma y color:SolidPeso molecular:740.24Dicyclomine
CAS:<p>Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.</p>Fórmula:C19H35NO2Forma y color:SolidPeso molecular:309.49Tebanicline hydrochloride
CAS:<p>Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.</p>Fórmula:C9H12Cl2N2OPureza:91.74% - 98.71%Forma y color:SolidPeso molecular:235.11TBPB
CAS:<p>TBPB is an allosteric M1 mAChR agonist.</p>Fórmula:C25H32N4OPureza:97.87% - 99.9%Forma y color:SolidPeso molecular:404.559-Ethyladenine
CAS:<p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>Fórmula:C7H9N5Pureza:99.35% - 99.41%Forma y color:SolidPeso molecular:163.18suvn-911
CAS:<p>suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.</p>Fórmula:C11H14Cl2N2OPureza:98.88%Forma y color:SolidPeso molecular:261.15Atracurium besylate
CAS:<p>Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.</p>Fórmula:C65H82N2O18S2Pureza:98.94% - 99.71%Forma y color:SolidPeso molecular:1243.49A 582941 HCl (848591-90-2(free base))
<p>A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing properties</p>Fórmula:C17H21ClN4Pureza:99.83%Forma y color:SolidPeso molecular:316.834BP-TQS
CAS:<p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>Fórmula:C18H17BrN2O2SPureza:99.96%Forma y color:SolidPeso molecular:405.31Imidafenacin
CAS:<p>Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.</p>Fórmula:C20H21N3OPureza:99.17%Forma y color:SolidPeso molecular:319.4Brompheniramine
CAS:<p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>Fórmula:C16H19BrN2Forma y color:SolidPeso molecular:319.24Varenicline dihydrochloride
CAS:<p>Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.</p>Fórmula:C13H15Cl2N3Pureza:99.88% - 99.97%Forma y color:SolidPeso molecular:284.18SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Fórmula:C20H25N3O2Pureza:99.02%Forma y color:SolidPeso molecular:339.43Ilmetropium iodide
CAS:<p>Ilmetropium iodide is a bronchodilator.</p>Fórmula:C20H30INO3Pureza:98.45%Forma y color:SolidPeso molecular:459.36Ursulcholic acid
CAS:<p>Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.</p>Fórmula:C24H40O10S2Pureza:98%Forma y color:SolidPeso molecular:552.7Pirmenol
CAS:<p>Pirmenol is a new antiarrhythmic drug</p>Fórmula:C22H30N2OPureza:97.24%Forma y color:SolidPeso molecular:338.49Darifenacin
CAS:<p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>Fórmula:C28H30N2O2Pureza:99.78%Forma y color:SolidPeso molecular:426.55LY2119620
CAS:<p>LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.</p>Fórmula:C19H24ClN5O3SPureza:99.7%Forma y color:SolidPeso molecular:437.94Benzetimide hydrochloride
CAS:<p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>Fórmula:C23H27ClN2O2Pureza:99.32%Forma y color:Off-White PowderPeso molecular:398.93Oxyphencyclimine
CAS:<p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>Fórmula:C20H28N2O3Forma y color:SolidPeso molecular:344.45Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Fórmula:C26H30NO4S2·BrPureza:99.53% - 99.69%Forma y color:SolidPeso molecular:564.55Coluracetam
CAS:<p>Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.</p>Fórmula:C19H23N3O3Pureza:99.96%Forma y color:SolidPeso molecular:341.4Mecamylamine hydrochloride
CAS:<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Fórmula:C11H22ClNPureza:99.76% - >99.99%Forma y color:White SolidPeso molecular:203.75Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:207.23BQCA
CAS:<p>BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.</p>Fórmula:C18H15NO4Pureza:97.22%Forma y color:SolidPeso molecular:309.32Oxyphencyclimine Hydrochloride
CAS:<p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>Fórmula:C20H29ClN2O3Pureza:99.55%Forma y color:SolidPeso molecular:380.91Propantheline
CAS:<p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>Fórmula:C23H30NO3Forma y color:SolidPeso molecular:368.49Encenicline
CAS:<p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>Fórmula:C16H17ClN2OSPureza:99.20%Forma y color:SolidPeso molecular:320.84Propiverine
CAS:<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.48JHU37160
CAS:JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Fórmula:C19H20ClFN4Pureza:99.87%Forma y color:SolidPeso molecular:358.84OXOMEMAZINE
CAS:<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Fórmula:C18H22N2O2SPureza:99.58%Forma y color:SolidPeso molecular:330.44Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Fórmula:C11H21NForma y color:SolidPeso molecular:167.29Methylbenactyzium Bromide
CAS:<p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>Fórmula:C21H28BrNO3Pureza:99.29%Forma y color:SolidPeso molecular:422.36Solifenacin hydrochloride
CAS:<p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:398.93Donepezil Hydrochloride
CAS:<p>Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).</p>Fórmula:C24H29NO3·HClPureza:99.55% - 99.8%Forma y color:White To Off-White Crystalline SolidPeso molecular:415.96Isopropamide Iodide
CAS:<p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>Fórmula:C23H33IN2OPureza:99.67%Forma y color:SolidPeso molecular:480.43SQ22536
CAS:<p>SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.</p>Fórmula:C9H11N5OPureza:99.18%Forma y color:Off-White SolidPeso molecular:205.22ML380
CAS:<p>ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).</p>Fórmula:C23H25F3N4O3SPureza:99.69%Forma y color:SolidPeso molecular:494.53VU0467154
CAS:<p>VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.</p>Fórmula:C17H15F3N4O3S2Pureza:98.28% - 99.51%Forma y color:SolidPeso molecular:444.45VU0152100
CAS:<p>VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).</p>Fórmula:C18H19N3O2SPureza:99.56%Forma y color:SolidPeso molecular:341.43Ipratropium Bromide
CAS:<p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>Fórmula:C20H30BrNO3Pureza:99.92%Forma y color:SolidPeso molecular:412.37VU0119498
CAS:<p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>Fórmula:C15H10BrNO2Pureza:97.56%Forma y color:SolidPeso molecular:316.15Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Forma y color:White SolidPeso molecular:397.34VU10010
CAS:<p>VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.</p>Fórmula:C17H16ClN3OSPureza:99.36%Forma y color:SolidPeso molecular:345.85Procyclidine hydrochloride
CAS:<p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>Fórmula:C19H30ClNOPureza:99.24% - 99.88%Forma y color:Crystals From Petroleum Ether White PowderPeso molecular:323.9Oxotremorine sesquifumarate
CAS:<p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>Fórmula:C12H18N2OC4H4O4Pureza:97.94%Forma y color:SolidPeso molecular:380.39TQS
CAS:<p>TQS (4-Naphthalen-1-yl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide) is a positive allosteric modulator of α7 nACh receptors.</p>Fórmula:C22H20N2O2SPureza:98.56%Forma y color:SolidPeso molecular:376.47MC-Val-Cit-PAB
CAS:<p>MC-Val-Cit-PAB: cathepsin-cleavable ADC linker used in FDA-approved brentuximab vedotin.</p>Fórmula:C28H40N6O7Pureza:98.24%Forma y color:SolidPeso molecular:572.65Revefenacin
CAS:<p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>Fórmula:C35H43N5O4Pureza:98.12%Forma y color:SolidPeso molecular:597.75Nitrocaramiphen hydrochloride
CAS:<p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>Fórmula:C18H27ClN2O4Pureza:99.74%Forma y color:SolidPeso molecular:370.87Piperidolate
CAS:<p>Piperidolate inhibits intestinal cramp induced by acetylcholine</p>Fórmula:C21H25NO2Pureza:98.45%Forma y color:SolidPeso molecular:323.43PNU-282987 S enantiomer free base
CAS:<p>PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).</p>Fórmula:C14H17ClN2OPureza:99.74%Forma y color:SolidPeso molecular:264.75VU 0238429
CAS:<p>VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).</p>Fórmula:C17H12F3NO4Pureza:>99.99%Forma y color:SolidPeso molecular:351.28Glycopyrrolate
CAS:<p>Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.</p>Fórmula:C19H28BrNO3Pureza:99.41% - 99.64%Forma y color:SolidPeso molecular:398.33CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Fórmula:C19H15Cl2N3O2Pureza:>99.99%Forma y color:SolidPeso molecular:388.25W-84 dibromide
CAS:<p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>Fórmula:C32H44Br2N4O4Pureza:95.56%Forma y color:SolidPeso molecular:708.52Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Forma y color:SolidPeso molecular:386.37Nor-benzetimide
CAS:<p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>Fórmula:C16H20N2O2Pureza:98.63%Forma y color:SolidPeso molecular:272.34PNU-120596
CAS:<p>PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.</p>Fórmula:C13H14ClN3O4Pureza:99.82%Forma y color:SolidPeso molecular:311.72MC-Val-Cit-PABC-PNP
CAS:<p>MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.</p>Fórmula:C35H43N7O11Pureza:97.2% - 98.055%Forma y color:SolidPeso molecular:737.76Blarcamesine
CAS:<p>Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.</p>Fórmula:C19H23NOPureza:99.87%Forma y color:SolidPeso molecular:281.39(S)-UFR2709
CAS:<p>(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.</p>Fórmula:C13H17NO2Forma y color:SolidPeso molecular:219.284Mc-Val-Ala-PAB
CAS:<p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>Fórmula:C25H34N4O6Pureza:98.34% - 99.24%Forma y color:SolidPeso molecular:486.56PHA 568487
CAS:<p>PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.</p>Fórmula:C20H24N2O7Forma y color:SolidPeso molecular:404.419VU0152099
CAS:<p>VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).</p>Fórmula:C18H17N3O3SPureza:98.46%Forma y color:SolidPeso molecular:355.41Bestim
CAS:<p>Bestim is an immunomodulatory dipeptide that is synthetic.</p>Fórmula:C16H19N3O5Pureza:99.76%Forma y color:SolidPeso molecular:333.34Oxyphenonium bromide
CAS:<p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>Fórmula:C21H34BrNO3Pureza:98.96%Forma y color:SolidPeso molecular:428.404Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Forma y color:Off-White SolidPeso molecular:419.41Monepantel
CAS:<p>Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.</p>Fórmula:C20H13F6N3O2SPureza:99.83%Forma y color:White PowderPeso molecular:473.39Velufenacin
CAS:<p>Velufenacin is an antagonist of muscarinic receptor[1].</p>Fórmula:C19H20ClFN2O2Pureza:99.65%Forma y color:SolidPeso molecular:362.83Pentoxyverine
CAS:<p>Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.</p>Fórmula:C20H31NO3Pureza:97.11%Forma y color:SolidPeso molecular:333.47Xanomeline tartrate
CAS:<p>Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂,具有抗精神病样活性,可改善认知,可用于研究精神分裂症和阿尔茨海默病。</p>Fórmula:C18H29N3O7SPureza:99.19%Forma y color:SolidPeso molecular:431.5AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Fórmula:C20H27N3OSPureza:98.62% - 99.89%Forma y color:SolidPeso molecular:357.51Mepenzolate Bromide
CAS:<p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>Fórmula:C21H26BrNO3Pureza:95.73% - 99.21%Forma y color:SolidPeso molecular:420.34Pipecuronium bromide
CAS:<p>Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.</p>Fórmula:C35H62Br2N4O4Pureza:>99.99%Forma y color:PowderPeso molecular:762.7Varenicline
CAS:<p>Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.</p>Fórmula:C13H13N3Pureza:99.76%Forma y color:SolidPeso molecular:211.26Atropine hydrobromide
CAS:<p>Atropine hydrobromide is a biochemical.</p>Fórmula:C17H24BrNO3Forma y color:SolidPeso molecular:370.28Anatabine dicitrate
<p>Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.</p>Fórmula:C22H28N2O14Pureza:98%Forma y color:SolidPeso molecular:544.46Pyrantel
CAS:<p>Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.</p>Fórmula:C11H14N2SPureza:98%Forma y color:Crystals From Methanol Yellowish Crystalline PowderPeso molecular:206.31Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Fórmula:C17H20D3NO3Peso molecular:292.39Oxantel
CAS:<p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28Aprofene
CAS:<p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>Fórmula:C21H27NO2Forma y color:SolidPeso molecular:325.44Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Fórmula:C107H173N37O26SPureza:98%Forma y color:SolidPeso molecular:2425.84Dianicline dihydrochloride
CAS:<p>Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.</p>Fórmula:C13H16N2OPureza:98%Forma y color:SolidPeso molecular:216.28Biperiden lactate
CAS:<p>Biperiden lactate is a biochemical.</p>Fórmula:C24H35NO4Forma y color:SolidPeso molecular:401.54VU0029767
CAS:<p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>Fórmula:C21H21N3O3Forma y color:SolidPeso molecular:363.41Azacyclonol hydrochloride
CAS:<p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>Fórmula:C18H22ClNOForma y color:Off White Crystalline PowderPeso molecular:303.83Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Fórmula:C21H27NOForma y color:Needles From Petroleum Ether SolidPeso molecular:309.45Sulindac sulfide
CAS:<p>Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.</p>Fórmula:C20H17FO2SPureza:99.35%Forma y color:SolidPeso molecular:340.41N-0861 racemate
CAS:<p>N-0861 racemate is the racemate of N-0861.</p>Fórmula:C13H17N5Pureza:98%Forma y color:SolidPeso molecular:243.31Sulfoxaflor
CAS:<p>Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.</p>Fórmula:C10H10F3N3OSPureza:99.56%Forma y color:SolidPeso molecular:277.27Sch412348
CAS:<p>Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.</p>Fórmula:C22H21F2N9OPureza:98%Forma y color:SolidPeso molecular:465.46SR 16584
CAS:<p>α3β4 nAChR antagonist</p>Fórmula:C17H22N2OPureza:99.84%Forma y color:SolidPeso molecular:270.37Tarafenacin
CAS:<p>Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.</p>Fórmula:C21H20F4N2O2Pureza:98%Forma y color:SolidPeso molecular:408.39Meseclazone
CAS:<p>Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.</p>Fórmula:C11H10ClNO3Pureza:98%Forma y color:SolidPeso molecular:239.654-DAMP
CAS:<p>4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.</p>Fórmula:C21H26INO2Pureza:98%Forma y color:SolidPeso molecular:451.34mAChr-in-1
CAS:<p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>Fórmula:C23H25IN2O2Pureza:98%Forma y color:SolidPeso molecular:488.36Darenzepine
CAS:<p>Darenzepine is a muscarinic receptor inhibitor.</p>Fórmula:C21H21N3O2Pureza:99.87%Forma y color:SolidPeso molecular:347.41UB 165 fumarate
CAS:<p>UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.</p>Fórmula:C17H19ClN2O4Pureza:99.72%Forma y color:SolidPeso molecular:350.8CDD0102
CAS:<p>CDD0102 is a potent agonist of M1 Muscarinic receptor.</p>Fórmula:C8H12N4OPureza:98%Forma y color:SolidPeso molecular:180.215-Iodo-A-85380 dihydrochloride
CAS:<p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>Fórmula:C9H13Cl2IN2OPureza:98%Forma y color:SolidPeso molecular:363.02Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Fórmula:C34H48Br2N4O4Forma y color:SolidPeso molecular:736.59LY 2087101
CAS:<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Fórmula:C15H11FN2OS2Pureza:98%Forma y color:SolidPeso molecular:318.39AR-R 17779 hydrochloride
CAS:<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Fórmula:C9H15ClN2O2Forma y color:SolidPeso molecular:218.68Elucaine
CAS:<p>Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.</p>Fórmula:C19H23NO2Pureza:98%Forma y color:SolidPeso molecular:297.39(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Forma y color:SolidPeso molecular:398.34SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Fórmula:C16H18N2O4Pureza:98%Forma y color:SolidPeso molecular:302.33LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Fórmula:C12H13ClN4SPureza:>99.99%Forma y color:SolidPeso molecular:280.78Terodiline
CAS:<p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>Fórmula:C20H27NPureza:98.20% - 99.59%Forma y color:SolidPeso molecular:281.44Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Fórmula:C8H18BrNO2Forma y color:SolidPeso molecular:240.141Nuvenzepine
CAS:<p>Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.</p>Fórmula:C19H20N4O2Pureza:98%Forma y color:SolidPeso molecular:336.39DA 4626
CAS:<p>DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.</p>Fórmula:C14H18N4Pureza:98%Forma y color:SolidPeso molecular:242.32Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Fórmula:C19H22N4O2SPureza:98%Forma y color:SolidPeso molecular:370.47AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Fórmula:C20H29FN2O2Forma y color:SolidPeso molecular:348.45Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Fórmula:C12H27NO3SPureza:98%Forma y color:SolidPeso molecular:265.41Chlorisondamine diiodide
CAS:<p>long lasting nicotinic antagonist</p>Fórmula:C14H20Cl4I2N2Forma y color:SolidPeso molecular:611.94ML381
CAS:<p>ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.</p>Fórmula:C21H21N3O4Forma y color:SolidPeso molecular:379.41ML169
CAS:<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Fórmula:C21H17BrFN3O4SPureza:98%Forma y color:SolidPeso molecular:506.34Zamifenacin
CAS:<p>Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.</p>Fórmula:C27H29NO3Pureza:98%Forma y color:SolidPeso molecular:415.52BNC375
CAS:<p>BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).</p>Fórmula:C19H23ClN2O3SPureza:98%Forma y color:SolidPeso molecular:394.92(R,R)-Reboxetine mesylate
CAS:<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Fórmula:C20H27NO6SForma y color:SolidPeso molecular:409.5M1 ligand 1
CAS:<p>Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.</p>Fórmula:C20H21NO2Forma y color:SolidPeso molecular:307.39Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Fórmula:C21H25NOPureza:98%Forma y color:SolidPeso molecular:307.43Muscarine iodide
CAS:<p>Muscarinic acetylcholine receptor agonist</p>Fórmula:C9H20INO2Pureza:98%Forma y color:SolidPeso molecular:301.17Tridihexethyl chloride
CAS:<p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>Fórmula:C21H36ClNOForma y color:SolidPeso molecular:353.97TC 2559 difumarate
CAS:<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Fórmula:C12H18N2OC4H404Pureza:98%Forma y color:SolidPeso molecular:380.39TC299423
CAS:<p>TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.</p>Fórmula:C11H15N3Forma y color:SolidPeso molecular:189.26SM-21 maleate
CAS:<p>Increases release of acetylcholine,σ2 antagonist</p>Fórmula:C22H28ClNO7Pureza:98%Forma y color:SolidPeso molecular:453.91TC 1698 dihydrochloride
CAS:<p>nicotinic α7 receptor agonist</p>Fórmula:C13H18N2Pureza:98%Forma y color:SolidPeso molecular:202.3Beperidium iodide
CAS:<p>Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).</p>Fórmula:C23H34IN3O3Forma y color:SolidPeso molecular:527.44WIN 62,577
CAS:<p>WIN 62,577 is a allosteric antagonist of mAChR.</p>Fórmula:C29H31N3OPureza:98%Forma y color:SolidPeso molecular:437.58Benzamide Derivative 1
CAS:<p>Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.</p>Fórmula:C22H34ClN3O3Pureza:>99.99%Forma y color:SolidPeso molecular:423.98Alvameline
CAS:<p>Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.</p>Fórmula:C9H15N5Pureza:98%Forma y color:SolidPeso molecular:193.25Muscarine chloride
CAS:<p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Fórmula:C9H20ClNO2Forma y color:SolidPeso molecular:209.71Quifenadine
CAS:<p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>Fórmula:C20H23NOPureza:98%Forma y color:SolidPeso molecular:293.4DAU 5884 hydrochloride
CAS:<p>muscarinic M3 receptor antagonist</p>Fórmula:C17H22ClN3O3Pureza:98%Forma y color:SolidPeso molecular:351.83Nelonicline
CAS:<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Fórmula:C17H19N3OSPureza:98%Forma y color:SolidPeso molecular:313.42BTM-1086
CAS:<p>BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.</p>Fórmula:C21H25N3OSPureza:98%Forma y color:SolidPeso molecular:367.51CP-601932
CAS:<p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>Fórmula:C12H12F3NForma y color:SolidPeso molecular:227.23Eucatropine
CAS:<p>Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.</p>Fórmula:C17H25NO3Forma y color:SolidPeso molecular:291.39Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Fórmula:C12H14N4OSPureza:98%Forma y color:SolidPeso molecular:262.33VU0090157
CAS:<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Fórmula:C19H21N3O7Pureza:98%Forma y color:SolidPeso molecular:403.39S-(+)-Mecamylamine hydrochloride
CAS:<p>Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.</p>Fórmula:C11H22ClNForma y color:SolidPeso molecular:203.75T761-0184
CAS:<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Fórmula:C16H20FN3OForma y color:SolidPeso molecular:289.35Revatropate
CAS:<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Fórmula:C19H27NO4SForma y color:SolidPeso molecular:365.49Rispenzepine
CAS:<p>Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.</p>Fórmula:C19H20N4O2Pureza:98%Forma y color:SolidPeso molecular:336.39

