AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Atropine methyl bromide
CAS:<p>Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a muscarinic receptor (mAChR) antagonist.</p>Fórmula:C18H26BrNO3Pureza:99.7%Forma y color:SolidPeso molecular:384.308Nicardipine hydrochloride
CAS:<p>Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.</p>Fórmula:C26H30ClN3O6Pureza:99.58% - 99.89%Forma y color:Yellow SolidPeso molecular:515.99Deschloroclozapine
CAS:<p>Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs agonist.</p>Fórmula:C18H20N4Pureza:99.61% - 99.98%Forma y color:SolidPeso molecular:292.38Temephos
CAS:<p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>Fórmula:C16H20O6P2S3Pureza:≥95%Forma y color:White Crystalline Solid Or LiquidPeso molecular:466.47Cotinine
CAS:<p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>Fórmula:C10H12N2OPureza:98% - 99.89%Forma y color:Viscous Oil SolidPeso molecular:176.22Bambuterol hydrochloride
CAS:<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Fórmula:C18H30ClN3O5Pureza:99.53% - 99.61%Forma y color:White SolidPeso molecular:403.91Lysipressin acetate(50-57-7(fb_acetate))
CAS:<p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.</p>Fórmula:C48H69N13O14S2Pureza:98.08%Forma y color:SolidPeso molecular:1116.28Dequalinium chloride
CAS:<p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>Fórmula:C30H40Cl2N4Pureza:99.79% - 99.9%Forma y color:SolidPeso molecular:527.59Ipratropium bromide monohydrate
CAS:<p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>Fórmula:C20H32BrNO4Pureza:97.85%Forma y color:SolidPeso molecular:430.38Gallamine triethiodide
CAS:<p>Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.</p>Fórmula:C30H60I3N3O3Pureza:98.90%Forma y color:White Amorphous Powder SolidPeso molecular:891.53Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Fórmula:C22H22FN3O2Pureza:97.16% - 98%Forma y color:SolidPeso molecular:379.43Tiotropium bromide
CAS:<p>Tiotropium bromide (BA679 BR) is a long-acting, 24 hour, anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disease (COPD).</p>Fórmula:C19H22BrNO4S2Pureza:96.82% - 99.97%Forma y color:White SolidPeso molecular:472.42Orphenadrine Citrate
CAS:<p>Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.</p>Fórmula:C18H23NO·C6H8O7Pureza:98% - 99.58%Forma y color:White SolidPeso molecular:461.5Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Forma y color:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Adiphenine hydrochloride
CAS:<p>Adiphenine hydrochloride (Patrovina), a nicotinic receptor inhibitor, can be used as an antispasmodic drug.</p>Fórmula:C20H25NO2·HClPureza:97.76% - 99.53%Forma y color:White Or Almost White PowderPeso molecular:347.88DL-trihexyphenidyl hydrochloride
CAS:<p>DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.</p>Fórmula:C20H32ClNOPureza:99.63% - 99.71%Forma y color:SolidPeso molecular:337.93Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Fórmula:C34H30N2O6SPureza:99.71%Peso molecular:594.69Rivastigmine tartrate
CAS:<p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>Fórmula:C14H22N2O2·C4H6O6Pureza:98% - 99.66%Forma y color:White To Off-White PowderPeso molecular:400.43(Rac)-Sabcomeline HCl
CAS:<p>Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.</p>Fórmula:C10H16ClN3OPureza:99.58%Forma y color:SoildPeso molecular:229.71Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Forma y color:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.889-Cyclopentyladenine
CAS:<p>9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signaling</p>Fórmula:C10H13N5Pureza:99.98%Forma y color:SolidPeso molecular:203.24Fesoterodine fumarate
CAS:<p>Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.</p>Fórmula:C26H37NO3·C4H4O4Pureza:99.16%Forma y color:White SolidPeso molecular:527.65Zelminemab
CAS:<p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>Pureza:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)Forma y color:LiquidPrimidone
CAS:<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Fórmula:C12H14N2O2Pureza:99.91%Forma y color:Crystals (Ntp 1992)Peso molecular:218.25MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.48Methscopolamine
CAS:<p>Methscopolamine (Hyoscine methyl bromide) (Pamine), as a natural plant alkaloid, is a muscarinic acetylcholine receptor blocker.</p>Fórmula:C18H24BrNO4Pureza:99.12% - ≥98%Forma y color:SolidPeso molecular:398.29Ribavirin
CAS:<p>Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.</p>Fórmula:C8H12N4O5Pureza:99.09% - 99.83%Forma y color:Less Solid Colourless SolidPeso molecular:244.20(Rac)-ABT-202 dihydrochloride
CAS:<p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>Fórmula:C9H15Cl2N3Pureza:97.4%Forma y color:SolidPeso molecular:236.142Procainamide hydrochloride
CAS:<p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>Fórmula:C13H21N3O·HClPureza:99.83% - 99.97%Forma y color:White To Slightly Yellow PowderPeso molecular:271.79PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Fórmula:C36H51Cl3N4O7SPureza:99.85%Forma y color:SolidPeso molecular:790.24Acetamiprid
CAS:<p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>Fórmula:C10H11ClN4Pureza:99.66%Forma y color:White PowderPeso molecular:222.67Rocuronium bromide
CAS:<p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>Fórmula:C32H53BrN2O4Pureza:99.77% - >99.99%Forma y color:White Or Off-White PowderPeso molecular:609.68TAK-071
CAS:<p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>Fórmula:C24H24FN3O3Pureza:98.02%Forma y color:SolidPeso molecular:421.46Carbachol
CAS:<p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>Fórmula:C6H15ClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:182.65Benzethonium chloride
CAS:<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Fórmula:C27H42ClNO2Pureza:99.91%Forma y color:White To Off-White Solid Solid Particulate/PowderPeso molecular:448.09Pyrantel tartrate
CAS:<p>Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.</p>Fórmula:C15H20N2O6SPureza:99.96%Forma y color:White CrystalsPeso molecular:356.39Dicyclomine hydrochloride
CAS:<p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>Fórmula:C19H36ClNO2Pureza:99.81%Forma y color:SolidPeso molecular:345.95VU 0365114
CAS:<p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>Fórmula:C22H14F3NO3Pureza:99.86%Forma y color:SolidPeso molecular:397.35Bethanechol chloride
CAS:<p>Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.</p>Fórmula:C7H17N2O2·ClPureza:95% - 99.73%Forma y color:White CrystallinePeso molecular:196.68Benactyzine hydrochloride
CAS:<p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>Fórmula:C20H26ClNO3Pureza:99.03% - 99.94%Forma y color:SolidPeso molecular:363.88Solifenacin succinate
CAS:<p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>Fórmula:C23H26N2O2·C4H6O4Pureza:99.85% - 99.98%Forma y color:SolidPeso molecular:480.56Diphenmanil methylsulfate
CAS:<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Fórmula:C20H24N·CH3O4SPureza:98% - 99.27%Forma y color:SolidPeso molecular:389.51Pirenzepine dihydrochloride
CAS:<p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>Fórmula:C19H21N5O2·2HClPureza:99.48% - 99.62%Forma y color:White PowderPeso molecular:424.32Neostigmine methyl sulfate
CAS:<p>Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of myasthenia gravis.</p>Fórmula:C13H22N2O6SPureza:99.34% - 99.53%Forma y color:Crystalline SolidPeso molecular:334.39Pancuronium dibromide
CAS:<p>Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide blocks neuromuscular transmission.</p>Fórmula:C35H60Br2N2O4Pureza:99.86%Forma y color:solidPeso molecular:732.67Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Fórmula:C14H18N2O2Pureza:97.37%Forma y color:White To Off-White Crystalline PowderPeso molecular:246.3Nebracetam hydrochloride
CAS:<p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>Fórmula:C12H17ClN2OPureza:99.23%Forma y color:SolidPeso molecular:240.729Carbetapentane citrate
CAS:<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Fórmula:C20H31NO3·C6H8O7Pureza:99.46%Forma y color:White To Off-White SolidPeso molecular:525.59Valethamate bromide
CAS:<p>Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.</p>Fórmula:C19H32BrNO2Pureza:>99.99%Forma y color:SolidPeso molecular:386.372',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Fórmula:C10H13N5O2Pureza:99.55%Forma y color:White SolidPeso molecular:235.24
