AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Milameline
CAS:<p>Milameline is a muscarinic receptor agonist that improves cognition.</p>Fórmula:C8H14N2OForma y color:SolidPeso molecular:154.21Biricodar dicitrate
CAS:<p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>Fórmula:C46H57N3O21Pureza:97.78% - 99.78%Forma y color:SolidPeso molecular:987.95Sofiniclin
CAS:<p>Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).</p>Fórmula:C10H11Cl2N3Pureza:98%Forma y color:SolidPeso molecular:244.12Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Fórmula:C31H42ClN5O3Forma y color:SolidPeso molecular:568.15VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Fórmula:C24H17ClF2N2O2Pureza:98%Forma y color:SolidPeso molecular:438.85Rivanicline
CAS:<p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.</p>Fórmula:C10H14N2Pureza:98%Forma y color:SolidPeso molecular:162.23Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Fórmula:C37H61BrN2O4Pureza:98%Forma y color:SolidPeso molecular:677.8ML375
CAS:<p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>Fórmula:C23H15ClF2N2O2Forma y color:SolidPeso molecular:424.83CP-601927
CAS:<p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>Fórmula:C12H12F3NForma y color:SolidPeso molecular:227.23Arecaidine propargyl ester tosylate
CAS:<p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>Fórmula:C17H21NO5SPureza:98%Forma y color:SolidPeso molecular:351.42VMY-2-95
CAS:<p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>Fórmula:C17H16N2OForma y color:SolidPeso molecular:264.32RJR 2429 dihydrochloride
CAS:<p>nAChR agonist that displays selectivity for α4β2</p>Fórmula:C12H18Cl2N2Pureza:98%Forma y color:SolidPeso molecular:261.19J 104129 fumarate
CAS:<p>M3 muscarinic receptor antagonist</p>Fórmula:C24H36N2O2Pureza:98%Forma y color:SolidPeso molecular:384.55Alvameline maleate
CAS:<p>Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.</p>Fórmula:C13H19N5O4Forma y color:SolidPeso molecular:309.32Vinconate
CAS:<p>Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.</p>Fórmula:C18H20N2O2Pureza:98%Forma y color:SolidPeso molecular:296.36AT-1001
CAS:<p>AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.</p>Fórmula:C15H21BrN2Forma y color:SolidPeso molecular:309.24Rivanicline oxalate
CAS:<p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:252.27Bradanicline HCl
CAS:<p>Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.</p>Fórmula:C22H24ClN3O2Forma y color:SolidPeso molecular:397.9DREADD agonist 21 dihydrochloride
CAS:<p>DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].</p>Fórmula:C17H20Cl2N4Pureza:98%Forma y color:SolidPeso molecular:351.27BPIPP
CAS:<p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>Fórmula:C22H16BrN3O3Pureza:98%Forma y color:SolidPeso molecular:450.28Procyclidine
CAS:<p>Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.</p>Fórmula:C19H29NOForma y color:SolidPeso molecular:287.44Oxybutynin R-isomer HCl
CAS:<p>Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.</p>Fórmula:C22H32ClNO3Forma y color:SolidPeso molecular:393.95VU0455691
CAS:<p>VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.</p>Fórmula:C24H25N5O3SPureza:98%Forma y color:SolidPeso molecular:463.55Ambutonium bromide
CAS:<p>Ambutonium bromide is an antagonist of acetylcholine.</p>Fórmula:C20H27BrN2OPureza:98%Forma y color:SolidPeso molecular:391.35(±)-Muscarine chloride
CAS:<p>(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].</p>Fórmula:C9H20ClNO2Forma y color:SolidPeso molecular:209.71Methapyrilene
CAS:<p>Methapyrilene is a histamine H1 antagonist with sedative action.</p>Fórmula:C14H19N3SForma y color:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Peso molecular:261.39Milameline hydrochloride
CAS:<p>Milameline hydrochloride is a Muscarinic receptor agonist.</p>Fórmula:C8H15ClN2OPureza:98%Forma y color:SolidPeso molecular:190.67Cycrimine
CAS:<p>Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.</p>Fórmula:C19H29NOForma y color:SolidPeso molecular:287.44Parapenzolate bromide
CAS:<p>Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.</p>Fórmula:C21H26BrNO3Forma y color:SolidPeso molecular:420.347DPNB-ABT594
<p>DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.</p>Fórmula:C31H46ClN3O11Forma y color:SolidPeso molecular:672.16AFDX384
CAS:<p>AFDX384 is potent M2/M4 selective antagonist.</p>Fórmula:C28H42N6O5SForma y color:SolidPeso molecular:574.74(S)-VQW-765
<p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>Fórmula:C19H22N2OForma y color:SolidPeso molecular:294.39Mazaticol
CAS:<p>Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.</p>Fórmula:C21H27NO3S2Forma y color:SolidPeso molecular:405.57J-104129 fumarate
CAS:<p>J-104129 fumarate is a potent M3 muscarinic receptor antagonist.</p>Fórmula:C28H40N2O6Forma y color:SolidPeso molecular:500.63BMS-902483
CAS:<p>BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.</p>Fórmula:C18H20N4OPureza:98%Forma y color:SolidPeso molecular:308.38RLH 033
CAS:<p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>Fórmula:C25H31ClN2O4Pureza:98%Forma y color:SolidPeso molecular:458.98Talsaclidine
CAS:<p>Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.</p>Fórmula:C10H15NOPureza:98%Forma y color:SolidPeso molecular:165.23A-85380 HCl
CAS:<p>A-85380 is an agonist of nicotinic acetylcholine receptor.</p>Fórmula:C9H14Cl2N2OForma y color:SolidPeso molecular:237.13Phenglutarimid
CAS:<p>Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.</p>Fórmula:C17H24N2O2Pureza:98%Forma y color:SolidPeso molecular:288.38Pirenzepine
CAS:<p>Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.</p>Fórmula:C19H21N5O2Forma y color:SolidPeso molecular:351.4ENS-163 phosphate
CAS:<p>Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.</p>Fórmula:C11H19N2O5PSPureza:98%Forma y color:SolidPeso molecular:322.32TMPH hydrochloride
CAS:<p>neuronal nicotinic ACh receptors (nAChRs) antagonist</p>Fórmula:C16H32ClNO2Pureza:98%Forma y color:SolidPeso molecular:305.889-CP-Ade Mesylate
CAS:<p>9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.</p>Fórmula:C11H17N5O3SPureza:99.81%Forma y color:SolidPeso molecular:299.35Arecaidine but-2-ynyl ester tosylate
CAS:<p>mAChR M2 agonist</p>Fórmula:C18H23NO5SPureza:98%Forma y color:SolidPeso molecular:365.44GSK575594A
CAS:<p>GSK575594A is a selective agonist of GPR55.</p>Fórmula:C24H23F2N3O3SForma y color:SolidPeso molecular:471.52(R)-Oxybutynin
CAS:<p>(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.</p>Fórmula:C22H31NO3Forma y color:SolidPeso molecular:357.49AC-42
CAS:<p>AC-42 is an allosteric agonist of M1 muscarinic receptor.</p>Fórmula:C20H31NOForma y color:SolidPeso molecular:301.47α7 nAchR-JAK2-STAT3 agonist 1
CAS:<p>α7 nAchR-JAK2-STAT3 agonist 1 is a potent inhibitor of the α7 nAchR-JAK2-STAT3 pathway that acts on nitric oxide (NO) (IC50: 0.32 μM).</p>Fórmula:C25H30O6Forma y color:SolidPeso molecular:426.5Ethybenztropine
CAS:<p>Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.</p>Fórmula:C22H27NOPureza:98%Forma y color:SolidPeso molecular:321.46Anabasine hydrochloride
CAS:<p>neuronal nicotinic ACh receptor partial agonist</p>Fórmula:C10H15ClN2Pureza:98%Forma y color:White To Off-White SolidPeso molecular:198.693
