AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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N-0861 racemate
CAS:<p>N-0861 racemate is the racemate of N-0861.</p>Fórmula:C13H17N5Pureza:98%Forma y color:SolidPeso molecular:243.31Bradanicline
CAS:<p>Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.</p>Fórmula:C22H23N3O2Forma y color:SolidPeso molecular:361.44Afacifenacin
CAS:<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Fórmula:C27H26F3N3O2Pureza:99.83%Forma y color:SolidPeso molecular:481.51mAChr-in-1
CAS:<p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>Fórmula:C23H25IN2O2Pureza:98%Forma y color:SolidPeso molecular:488.364-DAMP
CAS:<p>4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.</p>Fórmula:C21H26INO2Pureza:98%Forma y color:SolidPeso molecular:451.34Asoxime dichloride
CAS:<p>Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.</p>Fórmula:C14H16Cl2N4O3Pureza:99.86%Forma y color:SolidPeso molecular:359.21Tarafenacin D-tartrate
CAS:Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Fórmula:C25H26F4N2O8Pureza:99.86%Forma y color:SolidPeso molecular:558.48Camylofine
CAS:<p>Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.</p>Fórmula:C19H32N2O2·2HClPureza:98%Forma y color:SolidPeso molecular:393.4(Rac)-VU 6008667
CAS:<p>(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.</p>Fórmula:C24H17ClF2N2O2Pureza:99.82%Forma y color:SolidPeso molecular:438.85Pentolinium Tartrate
CAS:<p>Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.</p>Fórmula:C15H32N2·2C4H5O6Pureza:98%Forma y color:SolidPeso molecular:538.6AF-DX 384 free base
CAS:<p>AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.</p>Fórmula:C27H38N6O2Pureza:98%Forma y color:SolidPeso molecular:478.63Pozanicline
CAS:<p>Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.</p>Fórmula:C11H16N2OPureza:98%Forma y color:SolidPeso molecular:192.26CB-6673567
CAS:<p>CB-6673567 is a selective inhibitor of adenylyl cyclase.</p>Fórmula:C19H14N4O3Forma y color:SolidPeso molecular:346.34NGX-267
CAS:<p>NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.</p>Fórmula:C10H18N2OSForma y color:SolidPeso molecular:214.33Dac 5945
CAS:<p>DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.</p>Fórmula:C19H30ClN3OPureza:98%Forma y color:SolidPeso molecular:351.91Hexocyclium metilsulfate
CAS:<p>Hexocyclium metilsulfate has anti-gastric secretory effects in humans.</p>Fórmula:C21H36N2O5SPureza:98%Forma y color:SolidPeso molecular:428.59GS 283
CAS:<p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>Fórmula:C17H17NO3Forma y color:SolidPeso molecular:283.32(R)-VU 6008667
CAS:(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).Fórmula:C24H17ClF2N2O2Forma y color:SolidPeso molecular:438.85Anisodine hydrobromide
CAS:<p>Anisodine hydrobromide is an inhibitor of adenosine kinase.</p>Fórmula:C17H22BrNO5Forma y color:White Crystals Or Crystalline PowderPeso molecular:400.27Btm 1042
CAS:<p>Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.</p>Fórmula:C21H26ClN3OSForma y color:SolidPeso molecular:403.97
