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AChR

AChR

Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.

Se han encontrado 575 productos de "AChR"

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  • Xanomeline oxalate

    CAS:
    <p>Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.</p>
    Fórmula:C16H25N3O5S
    Pureza:99.1%
    Forma y color:Solid
    Peso molecular:371.45
  • NKY80

    CAS:
    <p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>
    Fórmula:C12H11N3O2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:229.23
  • Oxotremorine M iodide

    CAS:
    <p>Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.</p>
    Fórmula:C11H19IN2O
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:322.19
  • Iperoxo

    CAS:
    <p>Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.</p>
    Fórmula:C10H17IN2O2
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:324.16
  • Aceclidine

    CAS:
    <p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>
    Fórmula:C9H15NO2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:169.22
  • Posatirelin

    CAS:
    <p>Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.</p>
    Fórmula:C17H28N4O4
    Pureza:98.08% - 98.87%
    Forma y color:Solid
    Peso molecular:352.43
  • GSK233705

    CAS:
    <p>GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.</p>
    Fórmula:C24H29BrN2
    Pureza:99.87% - 99.98%
    Forma y color:Solid
    Peso molecular:425.4
  • Temiverine hydrochloride

    CAS:
    <p>Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.</p>
    Fórmula:C24H36ClNO3
    Pureza:99.26% - 99.43%
    Forma y color:Solid
    Peso molecular:422
  • Zamifenacin fumarate

    CAS:
    <p>Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.</p>
    Fórmula:C31H33NO7
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:531.6
  • LG 50643

    CAS:
    <p>LG 50643 is a muscarinic antagonist.</p>
    Fórmula:C24H34INO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:495.44
  • LY2033298

    CAS:
    <p>LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.</p>
    Fórmula:C13H14ClN3O2S
    Pureza:99.06%
    Forma y color:Solid
    Peso molecular:311.79
  • ICL-CCIC-0019

    CAS:
    <p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>
    Fórmula:C26H44Br2N4
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:572.46
  • PTAC oxalate

    CAS:
    <p>muscarinic receptor ligand</p>
    Fórmula:C14H21N3O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:359.46
  • N-Demethyl MK-6884

    CAS:
    <p>N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.</p>
    Fórmula:C24H23N5O
    Forma y color:Solid
    Peso molecular:397.47
  • Adenylyl cyclase-IN-1

    CAS:
    <p>Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].</p>
    Fórmula:C9H8N2S3
    Forma y color:Solid
    Peso molecular:240.37
  • Tiotropium Bromide hydrate

    CAS:
    <p>Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.</p>
    Fórmula:C19H24BrNO5S2
    Pureza:98.44% - 99.41%
    Forma y color:Solid
    Peso molecular:490.43
  • Timepidium bromide

    CAS:
    <p>Timepidium bromide is an agent of anticholinergic.</p>
    Fórmula:C17H22BrNOS2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:400.4
  • APS3

    CAS:
    <p>APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].</p>
    Fórmula:C18H7Cl2F6N5O5S2
    Forma y color:Solid
    Peso molecular:622.31
  • VU0453595

    CAS:
    <p>VU0453595 is a M1 positive allosteric modulator (PAM).</p>
    Fórmula:C18H15FN4O
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:322.34
  • VU 0255035

    CAS:
    <p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>
    Fórmula:C18H20N6O3S2
    Pureza:98.09% - 98.1%
    Forma y color:Solid
    Peso molecular:432.52