
AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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Xanomeline oxalate
CAS:<p>Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.</p>Fórmula:C16H25N3O5SPureza:99.1%Forma y color:SolidPeso molecular:371.45NKY80
CAS:<p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>Fórmula:C12H11N3O2Pureza:99.88%Forma y color:SolidPeso molecular:229.23Oxotremorine M iodide
CAS:<p>Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.</p>Fórmula:C11H19IN2OPureza:99.57%Forma y color:SolidPeso molecular:322.19Iperoxo
CAS:<p>Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.</p>Fórmula:C10H17IN2O2Pureza:99.81%Forma y color:SolidPeso molecular:324.16Aceclidine
CAS:<p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>Fórmula:C9H15NO2Pureza:>99.99%Forma y color:SolidPeso molecular:169.22Posatirelin
CAS:<p>Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.</p>Fórmula:C17H28N4O4Pureza:98.08% - 98.87%Forma y color:SolidPeso molecular:352.43GSK233705
CAS:<p>GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.</p>Fórmula:C24H29BrN2Pureza:99.87% - 99.98%Forma y color:SolidPeso molecular:425.4Temiverine hydrochloride
CAS:<p>Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.</p>Fórmula:C24H36ClNO3Pureza:99.26% - 99.43%Forma y color:SolidPeso molecular:422Zamifenacin fumarate
CAS:<p>Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.</p>Fórmula:C31H33NO7Pureza:99.88%Forma y color:SolidPeso molecular:531.6LG 50643
CAS:<p>LG 50643 is a muscarinic antagonist.</p>Fórmula:C24H34INO2Pureza:98%Forma y color:SolidPeso molecular:495.44LY2033298
CAS:<p>LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.</p>Fórmula:C13H14ClN3O2SPureza:99.06%Forma y color:SolidPeso molecular:311.79ICL-CCIC-0019
CAS:<p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>Fórmula:C26H44Br2N4Pureza:99.54%Forma y color:SolidPeso molecular:572.46PTAC oxalate
CAS:<p>muscarinic receptor ligand</p>Fórmula:C14H21N3O4S2Pureza:98%Forma y color:SolidPeso molecular:359.46N-Demethyl MK-6884
CAS:<p>N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.</p>Fórmula:C24H23N5OForma y color:SolidPeso molecular:397.47Adenylyl cyclase-IN-1
CAS:<p>Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].</p>Fórmula:C9H8N2S3Forma y color:SolidPeso molecular:240.37Tiotropium Bromide hydrate
CAS:<p>Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.</p>Fórmula:C19H24BrNO5S2Pureza:98.44% - 99.41%Forma y color:SolidPeso molecular:490.43Timepidium bromide
CAS:<p>Timepidium bromide is an agent of anticholinergic.</p>Fórmula:C17H22BrNOS2Pureza:98%Forma y color:SolidPeso molecular:400.4APS3
CAS:<p>APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].</p>Fórmula:C18H7Cl2F6N5O5S2Forma y color:SolidPeso molecular:622.31VU0453595
CAS:<p>VU0453595 is a M1 positive allosteric modulator (PAM).</p>Fórmula:C18H15FN4OPureza:99.91%Forma y color:SolidPeso molecular:322.34VU 0255035
CAS:<p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>Fórmula:C18H20N6O3S2Pureza:98.09% - 98.1%Forma y color:SolidPeso molecular:432.52
