Serina proteasa

Gabexate mesylate is a serine proteinase inhibitor used therapeutically in the treatment of pancreatitis, disseminated …

Aprotinin a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases …

PF-3644022 is an effective, selective, and ATP-competitive MAPKAPK2 (MK2) inhibitor (IC50: 5.2 nM and a …

Diminazene is a trypanocidal agent.

Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) …

BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of …

Phenylmethanesulfonyl fluoride (PMSF) is an enzyme inhibitor that inactivates IRC-50 arvin, subtilisin, and the fatty …

AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).

4-Aminobenzamidine (p-Aminobenzamidine) dihydrochloride is a strong trypsin inhibitor and a relatively weak inhibitor of urokinase …

Sivelestat sodium tetrahydrate is a competitive inhibitor of human neutrophil elastase, with an IC50 of …

Alpha-Amyrin is an inhibitor of trypsin and chymotrypsin with antineoplastic effects. alpha-Amyrin can be used …

ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and …

MEGA-9 solubilizes membrane protein and can be used as a nonionic detergent.

UK-371804 is an effective and specific uPA inhibitor. It was selected as a candidate for …

Nafamostat mesylate, a synthetic serine protease inhibitor, has been used for the treatment of allergic …

Secologanoside shows anti-complementary, allelopathic, and anti-elastase activities.

ZK824190 is an orally available and selective inhibitor of urokinase plasminogen activator (uPA). The IC50 …

Zt-12-037-01 is a ATP competitive STK19 inhibitor(IC50 values of 23.96 nM and 27.94 nM for …

SC-514 is a selective, orally active, ATP-competitive IKK-2 inhibitor (IC50=11.2±4.7 μM), obstructs NF-κB-dependent gene expression.

2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.

AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.

Benzamidine HCl is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki …

AEBSF hydrochloride is an irreversible inhibitor of serine proteases, such as chymotrypsin, kallikrein, thrombin, plasmin, …

Demethylwedelolactone is a natural product isolated from Eclipta alba, has trypsin inhibitory effect an IC50 …

Chrysophanol 8-O-glucoside and chrysophanol have mild cytotoxicity and anti-diabetic properties and can play metabolic roles …

Alvelestat is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with …

GSK690693 is a pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 2 nM/13 nM/9 nM, also …

Trypsin inhibitor (human urine urinastatin protein moiety), as an urinary trypsin inhibitor (UTI), is a …

ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.

Sivelestat is a potent and selective inhibitor of neutrophil elastase with IC50 of 44 nM.

KKI-5 acetate is a serine protease inhibitor that inhibits kallikrein and plasmin. KKI 5 may …

2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).

Leupeptin hemisulfate is a reversible, competitive serine/cysteine protease inhibitor. It is an orally active, antioxidant …

3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitor

Ceritinib (LDK378) is a specific ALK inhibitor (IC50: 0.2 nM).

BCX 1470 methanesulfonate inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM …

BCX 1470 inhibits the esterolytic activity of factor D and C1s (IC50: 96 nM and …

UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency …

ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).

ZEN-3411 is an inhibitor of BET(IC50s of 0.05, 0.05 and 0.06 μM for BRD4(BD1), BRD4(BD2) …

FK706 is a slow-binding and competitive human neutrophil elastase inhibitor (IC50: 83 nM; Ki: 4.2 …

JCP174 is a depalmitoylase inhibitor that enhances Toxoplasma host-cell invasion by targeting TgPPT1.