Serina proteasa
Los inhibidores de serina proteasa son compuestos que inhiben las serina proteasas, un grupo de enzimas caracterizadas por un residuo de serina en su sitio activo. Estas proteasas están involucradas en numerosos procesos fisiológicos, incluyendo la digestión, la respuesta inmunitaria, la coagulación sanguínea y la inflamación. Los inhibidores de serina proteasa son fundamentales para estudiar enfermedades en las que estas enzimas están desreguladas, como enfermedades cardiovasculares, cáncer y condiciones inflamatorias. En CymitQuimica, ofrecemos inhibidores de serina proteasa para apoyar su investigación en enzimología, mecanismos de enfermedades e intervenciones terapéuticas.
Se han encontrado 55 productos de "Serina proteasa"
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C1 Esterase Inhibitor (Human)
C1 Esterase Inhibitor (Human) is a glycoprotein derived from human plasma and acts as a serine protease inhibitor. It inactivates enzymes like C1r, C1s, and mannose-binding lectin-associated serine proteases (MASP) through covalent binding. This compound possesses anti-inflammatory properties and is utilized to prevent angioedema attacks associated with hereditary angioedema.Forma y color:Odour LiquidElastase (high purity)
Elastase (high purity) is a serine protease that hydrolyzes proteins and peptides.Forma y color:Odour SolidAE-3763
CAS:AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).Fórmula:C23H34F3N5O7Pureza:98%Forma y color:SolidPeso molecular:549.54Patamostat HCl
CAS:<p>Patamostat HCl is a highly potent and selective small molecule protease (protease) inhibitor that inhibits trypsin, fibrinolytic enzymes, and thrombin with IC50</p>Fórmula:C20H21ClN4O4SPureza:99.15% - 99.76%Forma y color:SoildPeso molecular:448.92Urokinase
CAS:<p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>Forma y color:SolidPKR-IN-C51
CAS:<p>PKR-IN-C51 is ATP-competitive protein kinase R (PKR) inhibitor that inhibits intracellular PKR activation and autophosphorylation. Ser/Thr kinase.</p>Fórmula:C23H21N5Pureza:98.94%Forma y color:SolidPeso molecular:367.45WNK463
CAS:WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).Fórmula:C21H24F3N7O2Pureza:>99.99% - ≥95%Forma y color:SolidPeso molecular:463.46WNK-IN-11
CAS:WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)Fórmula:C21H21Cl2N5OSPureza:98.32%Forma y color:SolidPeso molecular:462.42-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS:<p>2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.</p>Fórmula:C14H7BrClNO2Pureza:97.36%Forma y color:SolidPeso molecular:336.57Cetraxate hydrochloride
CAS:Cetraxate hydrochloride (DV10062) is an oral gastrointestinal medication. It has a cytoprotective effect.Fórmula:C17H24ClNO4Pureza:99.75%Forma y color:SolidPeso molecular:341.83Ceritinib
CAS:<p>Ceritinib (LDK378) is an ALK inhibitor with selective, ATP-competitive, and oral activity. Ceritinib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C28H36ClN5O3SPureza:98.52% - 99.77%Forma y color:SolidPeso molecular:558.14ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Fórmula:C22H19N3O2SPureza:99.12% - 99.87%Forma y color:SolidPeso molecular:389.47KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Fórmula:C37H59N11O11Pureza:99.44%Forma y color:SolidPeso molecular:833.95Alvelestat
CAS:<p>Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.</p>Fórmula:C25H22F3N5O4SPureza:98% - >99.99%Forma y color:SolidPeso molecular:545.532,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFórmula:C13H16O3Pureza:99.53% - 99.81%Forma y color:SolidPeso molecular:220.26Galegenimab
CAS:<p>Galegenimab (FHTR 2163; RG 6147; RO 7171009) is an HTRA1 antibody fragment for AMD research.</p>Pureza:95% - 95%Forma y color:LiquidLanadelumab
CAS:<p>Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.</p>Pureza:95% - 95%Forma y color:LiquidMEGA-9
CAS:<p>MEGA-9 (Nonanoyl-N-Methylglucamide) solubilizes membrane protein and can be used as a nonionic detergent.</p>Fórmula:C16H33NO6Pureza:99.9%Forma y color:SolidPeso molecular:335.44ZM223 hydrochloride (2031177-48-5 free base)
<p>ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.</p>Fórmula:C23H18ClF3N4O2S2Pureza:98%Forma y color:SolidPeso molecular:538.99AGLME
CAS:AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Fórmula:C11H21N3O4Forma y color:SolidPeso molecular:259.3
