Serina proteasa
Los inhibidores de serina proteasa son compuestos que inhiben las serina proteasas, un grupo de enzimas caracterizadas por un residuo de serina en su sitio activo. Estas proteasas están involucradas en numerosos procesos fisiológicos, incluyendo la digestión, la respuesta inmunitaria, la coagulación sanguínea y la inflamación. Los inhibidores de serina proteasa son fundamentales para estudiar enfermedades en las que estas enzimas están desreguladas, como enfermedades cardiovasculares, cáncer y condiciones inflamatorias. En CymitQuimica, ofrecemos inhibidores de serina proteasa para apoyar su investigación en enzimología, mecanismos de enfermedades e intervenciones terapéuticas.
Se han encontrado 81 productos para "Serina proteasa".
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hCAXII-IN-10
hCAXII-IN-10 (Compound 18b) acts as a dual inhibitor of human carbonic anhydrase isoenzyme XII (hCAXII) and cathepsin B, with a Ki value of 2.2 nM. It inhibits the function of hCAXII in creating a pH microenvironment conducive to tumor growth, showing promise for use in cancer research.Forma y color:Odour SolidMeOSuc-AAPF-CMK
CAS:MeOSuc-AAPF-CMK (MeOSuc-Ala-Ala-Pro-Phe-CH2Cl) is a potent inhibitor of the enzyme proteinase K [1].Fórmula:C26H35ClN4O7Forma y color:SolidPeso molecular:551.03Tiprelestat
CAS:Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.Fórmula:C254H416N72O75S10Forma y color:SolidPeso molecular:5999.09Lonodelestat TFA
Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.Fórmula:C73H112F3N15O21Forma y color:SolidPeso molecular:1592.75Z-APF-CMK
CAS:Z-APF-CMK is a selective inhibitor of the calcium (Ca2+)-regulated nuclear scaffold protease (CRNSP), as reported in reference [1].Fórmula:C26H30ClN3O5Forma y color:SolidPeso molecular:499.99Activated Protein C (390-404), human
CAS:Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.Fórmula:C91H130N22O23Pureza:98%Forma y color:SolidPeso molecular:1900.14α-Methyl-DL-aspartic acid
CAS:α-Methyl-DL-aspartic acid specifically inhibits argininosuccinate synthase (ASS), the rate-limiting enzyme in 1-citrulline-to-1-arginine recycling.Fórmula:C5H9NO4Pureza:99.91%Forma y color:SolidPeso molecular:147.129Suc-AAP-Abu-pNA
CAS:Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Fórmula:C25H34N6O9Forma y color:SolidPeso molecular:562.57Urinary Trypsin Inhibitor Fragment
CAS:Urinary Trypsin Inhibitor Fragment, a proteolysis product, inhibits tumor invasion.Fórmula:C40H66N14O9SPeso molecular:919.11PKR-IN-C51
CAS:PKR-IN-C51 is ATP-competitive protein kinase R (PKR) inhibitor that inhibits intracellular PKR activation and autophosphorylation. Ser/Thr kinase.Fórmula:C23H21N5Pureza:98.94%Forma y color:Yellow SolidPeso molecular:367.45Ref: TM-T24647
2mg82,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg192,00€25mg356,00€50mg530,00€100mg755,00€PKSI-527
CAS:PKSI-527 is a selective plasma kallikrein inhibitor with anti-arthritis activity.Fórmula:C25H32ClN3O4Forma y color:SolidPeso molecular:473.99DMP 777
CAS:DMP 777 is an oral selective HNE inhibitor that covalently binds to the active-site serine as a slow tight-binding competitive inhibitor.Fórmula:C31H40N4O6Forma y color:SolidPeso molecular:564.67Anti-KLK5/Kallikrein 5 Antibody
Anti-KLK5/Kallikrein 5 Antibody serves as a functional therapeutic tool specifically designed to enable the precise detection and neutralization of the serine protease KLK5 which plays a pivotal role in the deregulation of epidermal desquamation and the induction of Th2-driven inflammation during strictly monitored laboratory observation periods and molecular investigations to evaluate the pharmacological efficacy of targeted protease inhibition in specialized preclinical research environments to facilitate the study of severe skin disorders.ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Fórmula:C22H19N3O2SPureza:99.12% - 99.87%Forma y color:SolidPeso molecular:389.47Ref: TM-T3423
1mg34,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg92,00€25mg178,00€50mg295,00€100mg474,00€500mg1.035,00€2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFórmula:C13H16O3Pureza:99.53% - 99.81%Forma y color:SolidPeso molecular:220.26Ref: TM-T8802
1mg82,00€1mL*10mM (DMSO)146,00€5mg168,00€10mg244,00€25mg404,00€50mg567,00€100mg767,00€500mg1.521,00€Alvelestat
CAS:Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.Fórmula:C25H22F3N5O4SPureza:98% - >99.99%Forma y color:White SolidPeso molecular:545.53Ref: TM-T3107
1mg34,00€2mg43,00€5mg56,00€1mL*10mM (DMSO)74,00€10mg84,00€25mg148,00€50mg219,00€100mg349,00€500mg830,00€2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS:2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.Fórmula:C14H7BrClNO2Pureza:97.36%Forma y color:SolidPeso molecular:336.57WNK-IN-11
CAS:WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)Fórmula:C21H21Cl2N5OSPureza:98.32%Forma y color:SolidPeso molecular:462.4Ref: TM-T5456
1mg87,00€5mg172,00€1mL*10mM (DMSO)188,00€10mg280,00€25mg474,00€50mg683,00€100mg964,00€500mg1.918,00€Benzamidine hydrochloride
CAS:Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.Fórmula:C7H9ClN2Pureza:99.32% - 99.64%Forma y color:SolidPeso molecular:156.613Camostat
CAS:Camostat (FOY 305) inhibits serine protease, treats cancer, viral infections, fibrosis, and blocks SARS-CoV, Coronavirus, and SARS-CoV-2 in studies.Fórmula:C20H22N4O5Forma y color:SolidPeso molecular:398.41
