Receptor de melatonina
Los receptores de ácido lisofosfatídico (LPA) son un grupo de GPCR que responden al LPA, un lípido bioactivo involucrado en la proliferación, migración y supervivencia celular. La señalización de LPA juega un papel crucial en varios procesos fisiológicos, incluyendo la cicatrización de heridas, el desarrollo vascular y la metástasis del cáncer. La modulación de la actividad de los receptores de LPA se está explorando para aplicaciones terapéuticas en el cáncer, la fibrosis y las enfermedades inflamatorias. En CymitQuimica, ofrecemos una gama de moduladores de receptores de LPA de alta calidad para apoyar su investigación en señalización celular, oncología y trastornos inflamatorios.
Se han encontrado 26 productos de "Receptor de melatonina"
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Agomelatine
CAS:Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Fórmula:C15H17NO2Pureza:99.92%Forma y color:White SolidPeso molecular:243.3Ramelteon
CAS:Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.Fórmula:C16H21NO2Pureza:97.21% - 99.92%Forma y color:Crystalline SolidPeso molecular:259.34Ref: TM-T1463
2mg44,00€5mg65,00€10mg88,00€25mg136,00€50mg202,00€100mg325,00€500mg512,00€1mL*10mM (DMSO)71,00€Luzindole
CAS:Luzindole (N-0774) is a selective melatonin receptor antagonist.Fórmula:C19H20N2OPureza:98.53%Forma y color:Off-White Amorphous SolidPeso molecular:292.37Ref: TM-T15795
1mg51,00€2mgA consultar5mg97,00€10mg145,00€25mg259,00€50mg369,00€100mg540,00€200mgA consultar1mL*10mM (DMSO)156,00€UCM 549
CAS:UCM 549 is a bioactive chemical.Fórmula:C19H21NO2Forma y color:SolidPeso molecular:295.38Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Forma y color:Odour Solid4-P-PDOT
CAS:4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.Fórmula:C19H21NOPureza:99.91%Forma y color:SolidPeso molecular:279.38Melatonin-Tamoxifen Conjugate
Melatonin-Tamoxifen Conjugate (compound 16c) is an anticancer drug conjugate made of Melatonin and Tamoxifen, serving as an effective antagonist of ERα (IC50 = 863 nM). In cells expressing the hMT1 receptor, it binds to MLT receptors (Ki = 3.1 nM) and exhibits the ability to promote β-arrestin activation (EC50 = 914 nM) and ERK activation (EC50 = 98 nM). The IC50 values for Melatonin-Tamoxifen Conjugate in MCF-7, MDA-MB-231, and HT-1080 cell lines are 6.8 μM, 6.4 μM, and 1.7 μM, respectively.Fórmula:C47H58N4O4Forma y color:SolidPeso molecular:742.99Ramelteon-d5
CAS:<p>Ramelteon-d5 is a deuterated compound of Ramelteon.</p>Fórmula:C16H16D5NO2Forma y color:SolidPeso molecular:264.37ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Fórmula:C13H16ClN3O3Pureza:98.15%Forma y color:SolidPeso molecular:297.74Ref: TM-T9193
1mg52,00€5mg116,00€10mg182,00€25mg320,00€50mg449,00€100mg615,00€200mg830,00€1mL*10mM (DMSO)128,00€Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Fórmula:C15H19NO2Pureza:98.93% - 99.93%Forma y color:SolidPeso molecular:245.32N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Fórmula:C12H14N2OPureza:98.79%Forma y color:PowderPeso molecular:202.25Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Forma y color:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Fórmula:C31H34N2O4Pureza:99.77%Forma y color:SolidPeso molecular:498.61UCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Fórmula:C19H20N2O2Pureza:98.88%Forma y color:SolidPeso molecular:308.37DH-97
CAS:DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Fórmula:C22H26N2OForma y color:SolidPeso molecular:334.45Cgp 52608
CAS:CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.Fórmula:C8H12N4OS2Forma y color:SolidPeso molecular:244.34GR 196429
CAS:GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.Fórmula:C14H18N2O2Pureza:98%Forma y color:SolidPeso molecular:246.3S-22153
CAS:S22153 is an antagonist of melatonin receptor.Fórmula:C14H17NOSForma y color:SolidPeso molecular:247.36Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Fórmula:C15H19N3O2Forma y color:SolidPeso molecular:273.33S20928
CAS:S20928 is an antagonist of melatonin receptor.Fórmula:C17H19NOForma y color:SolidPeso molecular:253.34
