
Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Fórmula:C20H26N4O5SPureza:98%Forma y color:SolidPeso molecular:434.51Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Fórmula:C15H20BrIN4SPureza:98%Forma y color:SolidPeso molecular:495.22PF-03654746 Tosylate
CAS:<p>PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.</p>Fórmula:C25H32F2N2O4SPureza:98%Forma y color:SolidPeso molecular:494.6JNJ-39220675
CAS:<p>JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.</p>Fórmula:C21H24FN3O2Pureza:98.13% - 99.89%Forma y color:SolidPeso molecular:369.43JNJ-28610244
CAS:<p>JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.</p>Fórmula:C16H21N3OPureza:98%Forma y color:SolidPeso molecular:271.36Hetramine
CAS:<p>Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.</p>Fórmula:C15H20N4Pureza:98%Forma y color:SolidPeso molecular:256.35Fenethazine
CAS:<p>Fenethazine is an effective antihistamine used as an antiallergic drug.</p>Fórmula:C16H18N2SForma y color:SolidPeso molecular:270.39HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Forma y color:SolidPeso molecular:368.4Setastine
CAS:<p>Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.</p>Fórmula:C22H28ClNOForma y color:SolidPeso molecular:357.92BMH-7
CAS:<p>BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.</p>Fórmula:C20H21N5OPureza:99.71%Forma y color:SolidPeso molecular:347.41Tei 6472
CAS:<p>Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.</p>Fórmula:C32H39N3O5Pureza:98%Forma y color:SolidPeso molecular:545.67Nα-Methylhistamine dihydrochloride
CAS:<p>Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.</p>Fórmula:C6H13Cl2N3Pureza:98%Forma y color:SolidPeso molecular:198.094Embramine
CAS:<p>Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.</p>Fórmula:C18H22BrNOPureza:98%Forma y color:SolidPeso molecular:348.28PF 03654746 FA
<p>PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.</p>Fórmula:C19H26F2N2O3Pureza:99.44%Forma y color:SoildPeso molecular:368.42VUF 8430 dihydrobromide
CAS:<p>histamine H4 receptor full agonist</p>Fórmula:C4H12BrN5SPureza:98%Forma y color:SolidPeso molecular:242.14Bavisant dihydrochloride
CAS:<p>Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.</p>Fórmula:C19H29Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:402.36ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Fórmula:C11H17F3N6OPureza:97.45%Forma y color:SolidPeso molecular:306.29Setastine HCl
CAS:<p>Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.</p>Fórmula:C22H29Cl2NOForma y color:SolidPeso molecular:394.38A 987306
CAS:<p>A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.</p>Fórmula:C18H25N5OForma y color:SolidPeso molecular:327.42Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Fórmula:C22H24ClN3OPureza:99.35%Forma y color:White Crystal PowderPeso molecular:381.90
