Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Fórmula:C8H10N6SPureza:98%Forma y color:SolidPeso molecular:222.27JNJ-10191584
CAS:<p>JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation</p>Fórmula:C13H15ClN4OForma y color:SolidPeso molecular:278.74Alimemazine
CAS:<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Fórmula:C18H22N2SPureza:98%Forma y color:Crystals SolidPeso molecular:298.45Aminopotentidine
CAS:<p>H2 antagonist</p>Fórmula:C26H35N7O2Pureza:98%Forma y color:SolidPeso molecular:477.6Zolantidine dimaleate
CAS:<p>H2 receptor antagonist</p>Fórmula:C26H31N3O5SPureza:98%Forma y color:SolidPeso molecular:497.61BMY-25271
CAS:<p>BMY-25271 is an antagonist of histamine H2 receptor.</p>Fórmula:C12H19N5O2S2Pureza:98%Forma y color:SolidPeso molecular:329.44ABT-239
CAS:<p>ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.</p>Fórmula:C22H22N2OPureza:>99.99%Forma y color:SolidPeso molecular:330.42(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SForma y color:SolidPeso molecular:322.47A-304121
CAS:<p>A-304121 is a histamine H(3) receptor.</p>Fórmula:C20H29N3O3Forma y color:SolidPeso molecular:359.46OUP-186
CAS:<p>OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.</p>Fórmula:C19H30ClN3SForma y color:SolidPeso molecular:367.98JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Forma y color:SolidPeso molecular:312.45Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Forma y color:SolidPeso molecular:264.36Wy 49051
CAS:<p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>Fórmula:C28H33N5O3Pureza:99.89%Forma y color:SolidPeso molecular:487.59ROS 234
CAS:<p>ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.</p>Fórmula:C13H15N5Forma y color:SolidPeso molecular:241.29PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Fórmula:C18H24F2N2OPureza:98.85% - 99.57%Forma y color:SolidPeso molecular:322.39AZD5213
CAS:<p>AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.</p>Fórmula:C19H25N3O2Forma y color:SolidPeso molecular:327.42Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Fórmula:C20H21NO5Forma y color:SolidPeso molecular:355.38Immepip
CAS:<p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>Fórmula:C9H15N3Forma y color:SolidPeso molecular:165.24Phenyltoloxamine
CAS:<p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>Fórmula:C17H21NOForma y color:SolidPeso molecular:255.35Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Fórmula:C24H27Cl2FN6OPureza:98%Forma y color:SolidPeso molecular:505.42
