Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Linadryl hydrochloride
CAS:<p>Linadryl hydrochloride may have antihistamine activity.</p>Fórmula:C19H24ClNO2Forma y color:SolidPeso molecular:333.85Ramixotidine
CAS:<p>Ramixotidine is a competitive antagonist of histamine H2-receptor.</p>Fórmula:C16H21N3O3SPureza:98%Forma y color:SolidPeso molecular:335.42JNJ 10191584 maleate
CAS:<p>JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).</p>Fórmula:C17H19ClN4O5Pureza:99.37%Forma y color:SolidPeso molecular:394.81Dacemazine hydrochloride
CAS:<p>Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.</p>Fórmula:C16H17ClN2OSPureza:98%Forma y color:SolidPeso molecular:320.84Carcinine
CAS:<p>Carcinine ditrifluoroacetate is a H3 receptor antagonist.</p>Fórmula:C8H14N4OPureza:98%Forma y color:SolidPeso molecular:182.22Azatadine
CAS:<p>Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).</p>Fórmula:C20H22N2Pureza:98%Forma y color:SolidPeso molecular:290.4H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Forma y color:SolidPeso molecular:377.86Impromidine
CAS:<p>Impromidine is a highly potent and specific agonist of the histamine H2 receptor.</p>Fórmula:C14H23N7SPureza:98%Forma y color:SolidPeso molecular:321.44Rocastine
CAS:<p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>Fórmula:C13H19N3OSPureza:98.26%Forma y color:SolidPeso molecular:265.37H3 receptor-MO-1
CAS:<p>H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.</p>Fórmula:C20H27N3O2Pureza:99.11%Forma y color:SolidPeso molecular:341.45Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Forma y color:SolidPeso molecular:369.29Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Forma y color:SolidPeso molecular:527.66CP-66948
CAS:<p>CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.</p>Fórmula:C13H20N6SPureza:99.14%Forma y color:SolidPeso molecular:292.4PF-03654764
CAS:<p>PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.</p>Fórmula:C20H28F2N2OPureza:>99.99%Forma y color:SolidPeso molecular:350.45Lavoltidine
CAS:<p>Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.</p>Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Forma y color:SolidPeso molecular:359.47UR-PI376
CAS:<p>UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.</p>Fórmula:C17H22N6SForma y color:SolidPeso molecular:342.46GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Forma y color:SolidPeso molecular:377.48S-1-Propenyl-L-cysteine
CAS:<p>S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive</p>Fórmula:C6H11NO2SPureza:98%Forma y color:SolidPeso molecular:161.22ROS 234 dioxalate
CAS:<p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>Fórmula:C17H19N5O8Pureza:98%Forma y color:SolidPeso molecular:421.37Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Forma y color:SolidPeso molecular:371.34
