
Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Fórmula:C21H25ClN2O3Forma y color:SolidPeso molecular:388.89Dalcotidine
CAS:<p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>Fórmula:C18H29N3O2Pureza:99.11%Forma y color:SolidPeso molecular:319.44Nα-Methylhistamine FA
<p>Nα-Methylhistamine FA is a histamine H3 receptor agonist</p>Fórmula:C7H13N3O2Pureza:>99.99%Forma y color:SolidPeso molecular:171.2Dexchlorpheniramine free base
CAS:<p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>Fórmula:C16H19ClN2Pureza:98%Forma y color:Oily Liquid SolidPeso molecular:274.79(S)-Azelastine hydrochloride
CAS:<p>(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Fórmula:C22H25Cl2N3OPureza:98%Forma y color:SolidPeso molecular:418.36Cetirizine Impurity C dihydrochloride
CAS:<p>Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.</p>Fórmula:C21H27Cl3N2O3Forma y color:SolidPeso molecular:461.81JNJ-10181457 (hydrochloride)
CAS:<p>JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations</p>Fórmula:C20H30Cl2N2OForma y color:SolidPeso molecular:385.37Alcaftadine carboxylic acid
CAS:<p>Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.</p>Fórmula:C19H21N3O2Forma y color:SolidPeso molecular:323.39Cetirizine Impurity D
CAS:<p>Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.</p>Fórmula:C30H28Cl2N2Forma y color:SolidPeso molecular:487.46Sigma-1 receptor antagonist 5
<p>Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors</p>Fórmula:C26H27N3OPureza:98%Forma y color:SolidPeso molecular:397.51Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Fórmula:C22H27ClN2O3Forma y color:SolidPeso molecular:402.91Conessine hydrobromide
CAS:<p>Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.</p>Fórmula:C24H41BrN2Forma y color:SolidPeso molecular:437.51(+)-Dropropizine
CAS:<p>(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.</p>Fórmula:C13H20N2O2Pureza:>99.99%Forma y color:White Or Off White Crystalline PowderPeso molecular:236.31Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Forma y color:Odour SolidKSK94 FA
<p>KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.</p>Fórmula:C26H28N4O3Pureza:97.51%Forma y color:SoildPeso molecular:444.53Alimemazine D6
CAS:<p>Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.</p>Fórmula:C18H22N2SPureza:98%Forma y color:SolidPeso molecular:304.48Antazoline phosphate
CAS:<p>Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.</p>Fórmula:C17H22N3O4PPureza:98%Forma y color:CoaPeso molecular:363.35Hydroxyzine D8
CAS:<p>Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.</p>Fórmula:C21H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:382.95Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Forma y color:SolidPeso molecular:396.94Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOForma y color:SolidPeso molecular:281.39

