Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Fórmula:C20H26N4O5SPureza:98%Forma y color:SolidPeso molecular:434.51Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Fórmula:C15H20BrIN4SPureza:98%Forma y color:SolidPeso molecular:495.22PF-03654746 Tosylate
CAS:<p>PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.</p>Fórmula:C25H32F2N2O4SPureza:98%Forma y color:SolidPeso molecular:494.6JNJ-39220675
CAS:<p>JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.</p>Fórmula:C21H24FN3O2Pureza:98.13% - 99.89%Forma y color:SolidPeso molecular:369.43JNJ-28610244
CAS:<p>JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.</p>Fórmula:C16H21N3OPureza:98%Forma y color:SolidPeso molecular:271.36Hetramine
CAS:<p>Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.</p>Fórmula:C15H20N4Pureza:98%Forma y color:SolidPeso molecular:256.35Fenethazine
CAS:<p>Fenethazine is an effective antihistamine used as an antiallergic drug.</p>Fórmula:C16H18N2SForma y color:SolidPeso molecular:270.39HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Fórmula:C21H21FN2O3Pureza:98%Forma y color:SolidPeso molecular:368.4Setastine
CAS:<p>Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.</p>Fórmula:C22H28ClNOForma y color:SolidPeso molecular:357.92BMH-7
CAS:<p>BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.</p>Fórmula:C20H21N5OPureza:99.71%Forma y color:SolidPeso molecular:347.41Tei 6472
CAS:<p>Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.</p>Fórmula:C32H39N3O5Pureza:98%Forma y color:SolidPeso molecular:545.67Nα-Methylhistamine dihydrochloride
CAS:<p>Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.</p>Fórmula:C6H13Cl2N3Pureza:98%Forma y color:SolidPeso molecular:198.094Embramine
CAS:<p>Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.</p>Fórmula:C18H22BrNOPureza:98%Forma y color:SolidPeso molecular:348.28PF 03654746 FA
<p>PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.</p>Fórmula:C19H26F2N2O3Pureza:99.44%Forma y color:SoildPeso molecular:368.42VUF 8430 dihydrobromide
CAS:<p>histamine H4 receptor full agonist</p>Fórmula:C4H12BrN5SPureza:98%Forma y color:SolidPeso molecular:242.14Bavisant dihydrochloride
CAS:<p>Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.</p>Fórmula:C19H29Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:402.36ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Fórmula:C11H17F3N6OPureza:97.45%Forma y color:SolidPeso molecular:306.29Setastine HCl
CAS:<p>Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.</p>Fórmula:C22H29Cl2NOForma y color:SolidPeso molecular:394.38A 987306
CAS:<p>A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.</p>Fórmula:C18H25N5OForma y color:SolidPeso molecular:327.42Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Fórmula:C22H24ClN3OPureza:99.35%Forma y color:White Crystal PowderPeso molecular:381.90Zaltidine
CAS:<p>Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.</p>Fórmula:C8H10N6SPureza:98%Forma y color:SolidPeso molecular:222.27JNJ-10191584
CAS:<p>JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation</p>Fórmula:C13H15ClN4OForma y color:SolidPeso molecular:278.74Alimemazine
CAS:<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Fórmula:C18H22N2SPureza:98%Forma y color:Crystals SolidPeso molecular:298.45Aminopotentidine
CAS:<p>H2 antagonist</p>Fórmula:C26H35N7O2Pureza:98%Forma y color:SolidPeso molecular:477.6Zolantidine dimaleate
CAS:<p>H2 receptor antagonist</p>Fórmula:C26H31N3O5SPureza:98%Forma y color:SolidPeso molecular:497.61BMY-25271
CAS:<p>BMY-25271 is an antagonist of histamine H2 receptor.</p>Fórmula:C12H19N5O2S2Pureza:98%Forma y color:SolidPeso molecular:329.44ABT-239
CAS:<p>ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.</p>Fórmula:C22H22N2OPureza:>99.99%Forma y color:SolidPeso molecular:330.42(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SForma y color:SolidPeso molecular:322.47A-304121
CAS:<p>A-304121 is a histamine H(3) receptor.</p>Fórmula:C20H29N3O3Forma y color:SolidPeso molecular:359.46OUP-186
CAS:<p>OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.</p>Fórmula:C19H30ClN3SForma y color:SolidPeso molecular:367.98JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Forma y color:SolidPeso molecular:312.45Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Fórmula:C18H20N2Pureza:99.85%Forma y color:SolidPeso molecular:264.36Wy 49051
CAS:<p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>Fórmula:C28H33N5O3Pureza:99.89%Forma y color:SolidPeso molecular:487.59ROS 234
CAS:<p>ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.</p>Fórmula:C13H15N5Forma y color:SolidPeso molecular:241.29PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Fórmula:C18H24F2N2OPureza:98.85% - 99.57%Forma y color:SolidPeso molecular:322.39AZD5213
CAS:<p>AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.</p>Fórmula:C19H25N3O2Forma y color:SolidPeso molecular:327.42Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Fórmula:C20H21NO5Forma y color:SolidPeso molecular:355.38Immepip
CAS:<p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>Fórmula:C9H15N3Forma y color:SolidPeso molecular:165.24Phenyltoloxamine
CAS:<p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>Fórmula:C17H21NOForma y color:SolidPeso molecular:255.35Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Fórmula:C24H27Cl2FN6OPureza:98%Forma y color:SolidPeso molecular:505.42GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Fórmula:C21H26ClN3O2Pureza:98%Forma y color:SolidPeso molecular:387.9GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Fórmula:C20H29F3N4OForma y color:SolidPeso molecular:398.47Sequifenadine
CAS:<p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>Fórmula:C22H27NOForma y color:SolidPeso molecular:321.46A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Fórmula:C17H21N5Forma y color:SolidPeso molecular:295.38Loratadine N-oxide
CAS:<p>Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.</p>Fórmula:C22H23ClN2O3Forma y color:SolidPeso molecular:398.88MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Fórmula:C23H24F3N3O2Pureza:99.90%Forma y color:SolidPeso molecular:431.45N-Acetylhistamine
CAS:<p>N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.</p>Fórmula:C7H11N3OPureza:99.51%Forma y color:SolidPeso molecular:153.18Izuforant
CAS:<p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>Fórmula:C12H12BrN7Forma y color:SolidPeso molecular:334.17A-943931
CAS:<p>A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.</p>Fórmula:C17H21N5Pureza:99.79%Forma y color:SolidPeso molecular:295.38Pitolisant oxalate
CAS:<p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C19H28ClNO5Pureza:98%Forma y color:SolidPeso molecular:385.88Pirolate
CAS:<p>Pirolate is a receptor of histamine H1.</p>Fórmula:C16H15N3O5Pureza:98%Forma y color:SolidPeso molecular:329.31Bepotastine tosylate
CAS:<p>Bepotastine tosylate: Oral 2nd-gen H1 antagonist, inhibits histamine effects on NGF; treats conjunctivitis, urticaria.</p>Fórmula:C28H33ClN2O6SForma y color:SolidPeso molecular:561.09VUF-10497
CAS:<p>VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).</p>Fórmula:C18H20ClN5SPureza:98%Forma y color:SolidPeso molecular:373.9A331440
CAS:<p>A331440 is an modulator of L-histidine and histamine H3 receptor.</p>Fórmula:C22H27N3OForma y color:SolidPeso molecular:349.47Phenindamine
CAS:<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Fórmula:C19H19NForma y color:SolidPeso molecular:261.36Acreozast
CAS:<p>Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.</p>Fórmula:C15H14ClN3O6Forma y color:SolidPeso molecular:367.74CP19
CAS:<p>CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].</p>Fórmula:C26H30N2O5Forma y color:SolidPeso molecular:450.53Phenindamine Tartrate
CAS:<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Fórmula:C23H25NO6Forma y color:SolidPeso molecular:411.454INCB38579
CAS:<p>INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.</p>Fórmula:C25H34N6OForma y color:SolidPeso molecular:434.58Thioperamide
CAS:<p>histamine H3 and H4 antagonist/inverse agonist</p>Fórmula:C15H24N4SPureza:98%Forma y color:White SolidPeso molecular:292.44VUF 5681 dihydrobromide
CAS:<p>histamine H3 receptor silent antagonist</p>Fórmula:C11H21Br2N3Pureza:98%Forma y color:SolidPeso molecular:355.11Carbinoxamine
CAS:<p>Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.</p>Fórmula:C16H19ClN2OPureza:98%Forma y color:LiquidPeso molecular:290.79Nebidrazine
CAS:<p>Nebidrazine is an alpha-adrenoceptor agonist.</p>Fórmula:C9H8Cl2N6Forma y color:SolidPeso molecular:271.11Toreforant
CAS:<p>Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).</p>Fórmula:C23H32N6Pureza:98%Forma y color:SolidPeso molecular:392.54VUF 8430
CAS:<p>VUF 8430 is a selective agonist for the H4 receptor.</p>Fórmula:C4H11N5SPureza:98%Forma y color:SolidPeso molecular:161.23UK-9040
CAS:<p>UK-9040 inhibits gastric secretory.</p>Fórmula:C23H31NSPureza:98%Forma y color:SolidPeso molecular:353.56SUN 1334H
CAS:<p>SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).</p>Fórmula:C23H28Cl2F2N2O3Pureza:98%Forma y color:SolidPeso molecular:489.38Adriforant hydrochloride
CAS:<p>Adriforant hydrochloride is an antagonist of histamine H4 receptor.</p>Fórmula:C13H25Cl3N6Pureza:98%Forma y color:SolidPeso molecular:371.74Seliforant
CAS:<p>Seliforant is a histamine H4 receptor antagonist.</p>Fórmula:C12H21N5Pureza:98%Forma y color:SolidPeso molecular:235.33(R)-(-)-α-Methylhistamine dihydrobromide
CAS:<p>(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).</p>Fórmula:C6H13Br2N3Pureza:98%Forma y color:SolidPeso molecular:287Amthamine dihydrobromide
CAS:<p>H2 agonist</p>Fórmula:C6H13Br2N3SPureza:98%Forma y color:SolidPeso molecular:319.06Carcainium chloride
CAS:<p>Carcainium chloride (Carcainium (chloride)) is a derivative of Lidocaine and possesses an antitussive effect.</p>Fórmula:C18H22ClN3O2Pureza:99.89%Forma y color:SolidPeso molecular:347.84DA 4643
CAS:<p>DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.</p>Fórmula:C12H16Cl2N6SPureza:98%Forma y color:SolidPeso molecular:347.26Mequitamium iodide
CAS:<p>Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.</p>Fórmula:C21H25IN2SForma y color:SolidPeso molecular:464.41Impentamine dihydrobromide
CAS:<p>Impentamine dihydrobromide is a histamine H3 receptor antagonist.</p>Fórmula:C8H17Br2N3Pureza:98%Forma y color:SolidPeso molecular:315.05Chloracyzine
CAS:<p>Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.</p>Fórmula:C19H21ClN2OSForma y color:SolidPeso molecular:360.9AHR-13268D
CAS:<p>AHR-13268D is a new agent of antiallergic/antihistaminic.</p>Fórmula:C28H29F2NNaO4Pureza:98%Forma y color:SolidPeso molecular:504.53AHR-14310C
CAS:<p>AHR-14310C is a long-acting and nonsedating H1-antihistamine.</p>Fórmula:C24H28F2N2O3Pureza:98%Forma y color:SolidPeso molecular:430.49NNC-38-1049
CAS:<p>NNC-38-1049 is a novel selective antagonist of histamine H3.</p>Fórmula:C19H25ClN2O2Pureza:98%Forma y color:SolidPeso molecular:348.87Aplysamine-1
CAS:<p>Aplysamine-1 is an antagonist of histamine H3 receptor.</p>Fórmula:C15H24Br2N2OPureza:98%Forma y color:SolidPeso molecular:408.17Linadryl hydrochloride
CAS:<p>Linadryl hydrochloride may have antihistamine activity.</p>Fórmula:C19H24ClNO2Forma y color:SolidPeso molecular:333.85Ramixotidine
CAS:<p>Ramixotidine is a competitive antagonist of histamine H2-receptor.</p>Fórmula:C16H21N3O3SPureza:98%Forma y color:SolidPeso molecular:335.42JNJ 10191584 maleate
CAS:<p>JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).</p>Fórmula:C17H19ClN4O5Pureza:99.37%Forma y color:SolidPeso molecular:394.81Dacemazine hydrochloride
CAS:<p>Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.</p>Fórmula:C16H17ClN2OSPureza:98%Forma y color:SolidPeso molecular:320.84Carcinine
CAS:<p>Carcinine ditrifluoroacetate is a H3 receptor antagonist.</p>Fórmula:C8H14N4OPureza:98%Forma y color:SolidPeso molecular:182.22Azatadine
CAS:<p>Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).</p>Fórmula:C20H22N2Pureza:98%Forma y color:SolidPeso molecular:290.4H3R-IN-1 Hydrochloride
CAS:<p>H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .</p>Fórmula:C19H24ClN3O3Pureza:98%Forma y color:SolidPeso molecular:377.86Impromidine
CAS:<p>Impromidine is a highly potent and specific agonist of the histamine H2 receptor.</p>Fórmula:C14H23N7SPureza:98%Forma y color:SolidPeso molecular:321.44Rocastine
CAS:<p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>Fórmula:C13H19N3OSPureza:98.26%Forma y color:SolidPeso molecular:265.37H3 receptor-MO-1
CAS:<p>H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.</p>Fórmula:C20H27N3O2Pureza:99.11%Forma y color:SolidPeso molecular:341.45Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Forma y color:SolidPeso molecular:369.29Bamirastine
CAS:<p>Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on</p>Fórmula:C31H37N5O3Pureza:96.68%Forma y color:SolidPeso molecular:527.66CP-66948
CAS:<p>CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.</p>Fórmula:C13H20N6SPureza:99.14%Forma y color:SolidPeso molecular:292.4PF-03654764
CAS:<p>PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.</p>Fórmula:C20H28F2N2OPureza:>99.99%Forma y color:SolidPeso molecular:350.45Lavoltidine
CAS:<p>Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.</p>Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Forma y color:SolidPeso molecular:359.47UR-PI376
CAS:<p>UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.</p>Fórmula:C17H22N6SForma y color:SolidPeso molecular:342.46GSK-239512
CAS:<p>GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.</p>Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Forma y color:SolidPeso molecular:377.48S-1-Propenyl-L-cysteine
CAS:<p>S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive</p>Fórmula:C6H11NO2SPureza:98%Forma y color:SolidPeso molecular:161.22ROS 234 dioxalate
CAS:<p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>Fórmula:C17H19N5O8Pureza:98%Forma y color:SolidPeso molecular:421.37Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Fórmula:C19H17NO7Pureza:95% - 97.34%Forma y color:SolidPeso molecular:371.34FR-A 19
CAS:<p>FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.</p>Fórmula:C25H34Cl3F2N5Forma y color:SolidPeso molecular:548.93VUF 8328
CAS:<p>VUF 8328 is an agonist of histamine H(3) receptor.</p>Fórmula:C7H12N4SPureza:98%Forma y color:SolidPeso molecular:184.26Adriforant
CAS:<p>Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.</p>Fórmula:C13H22N6Pureza:99.84%Forma y color:SolidPeso molecular:262.35FRG8701
CAS:<p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>Fórmula:C22H30N2O4SPureza:98%Forma y color:SolidPeso molecular:418.55ReN-1869 hydrochloride
CAS:<p>ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.</p>Fórmula:C24H28ClNO2Pureza:98%Forma y color:SolidPeso molecular:397.94H4R antagonist 1
CAS:<p>H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.</p>Fórmula:C11H11BrN8Forma y color:SolidPeso molecular:335.16(±)-Tazifylline
CAS:<p>(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.</p>Fórmula:C23H32N6O3SPureza:99.54%Forma y color:SolidPeso molecular:472.6Noberastine
CAS:<p>Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.</p>Fórmula:C17H21N5OPureza:99.72% - >99.99%Forma y color:SolidPeso molecular:311.38KSK68
CAS:<p>KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.</p>Fórmula:C23H28N2O2Pureza:99.11%Forma y color:SolidPeso molecular:364.48Immethridine dihydrobromide
CAS:<p>Immethridine dihydrobromide is a histamine H3 receptor agonist.</p>Fórmula:C9H11Br2N3Pureza:97.61% - 98.14%Forma y color:SolidPeso molecular:321.01D18024
CAS:<p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>Fórmula:C29H31ClFN3OPureza:99.86%Forma y color:SolidPeso molecular:492.03Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Fórmula:C14H26Cl3N7SPureza:99.82%Forma y color:SolidPeso molecular:430.83Enerisant hydrochloride
CAS:<p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>Fórmula:C22H31ClN4O3Pureza:99.95%Forma y color:SolidPeso molecular:434.96Linetastine
CAS:<p>Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.</p>Fórmula:C35H40N2O6Pureza:99.76%Forma y color:SolidPeso molecular:584.7Pitolisant
CAS:<p>Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Fórmula:C17H26ClNOPureza:99.84%Forma y color:SolidPeso molecular:295.85KSK94
CAS:<p>KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.</p>Fórmula:C25H26N4OPureza:99.60%Forma y color:SolidPeso molecular:398.5Irdabisant
CAS:<p>Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.</p>Fórmula:C18H23N3O2Pureza:99.96%Forma y color:SolidPeso molecular:313.39Efletirizine
CAS:<p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>Fórmula:C21H24F2N2O3Pureza:99.39%Forma y color:SolidPeso molecular:390.42Antihistamine-1
CAS:<p>Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。</p>Fórmula:C23H24FN5Pureza:99.69%Forma y color:SolidPeso molecular:389.47NP10679
CAS:<p>NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.</p>Fórmula:C23H26F3N3O3Pureza:99.43%Forma y color:SolidPeso molecular:449.47Proxyfan
CAS:<p>Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.</p>Fórmula:C13H16N2OPureza:99.68%Forma y color:SolidPeso molecular:216.28ReN-1869
CAS:<p>ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases</p>Fórmula:C24H27NO2Pureza:99.83% - 99.98%Forma y color:SolidPeso molecular:361.48DF-1111301
CAS:<p>DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.</p>Fórmula:C15H25Cl2N3OPureza:99.17%Forma y color:SolidPeso molecular:334.29Eclazolast
CAS:<p>Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.</p>Fórmula:C12H12ClNO4Pureza:98.36% - 98.58%Forma y color:SolidPeso molecular:269.68KP136
CAS:<p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>Fórmula:C16H18N4O3Pureza:98.3% - 98.61%Forma y color:SolidPeso molecular:314.34Bavisant
CAS:<p>Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.</p>Fórmula:C19H27N3O2Pureza:99.21% - 99.65%Forma y color:SolidPeso molecular:329.44Abt-288
CAS:<p>ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.</p>Fórmula:C23H24N4OPureza:98.17% - 98.49%Forma y color:SolidPeso molecular:372.46Clemastine
CAS:<p>Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.</p>Fórmula:C21H26ClNOPureza:99.21%Forma y color:SolidPeso molecular:343.89JZP-361
CAS:<p>JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.</p>Fórmula:C22H20ClN5OPureza:99.82%Forma y color:SolidPeso molecular:405.88JNJ-28583867
CAS:<p>JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.</p>Fórmula:C24H32N2O2SForma y color:SolidPeso molecular:412.59Cipralisant maleate
CAS:<p>Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.</p>Fórmula:C18H24N2O4Forma y color:SolidPeso molecular:332.39CI-949
CAS:<p>CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).</p>Fórmula:C20H20N6O3Pureza:98%Forma y color:SolidPeso molecular:392.41Ebrotidine
CAS:<p>Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection.</p>Fórmula:C14H17BrN6O2S3Pureza:97.519%Forma y color:SolidPeso molecular:477.42GSK-1004723
CAS:<p>GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.</p>Fórmula:C39H49ClN4O2Forma y color:SolidPeso molecular:641.28Quinotolast sodium
CAS:<p>Quinotolast sodium inhibits histamine, LTC4 and PGD2 release in a concentration-dependent manner in the concentration range of 1-100 μg/mL.</p>Fórmula:C17H12N6NaO3Pureza:98%Forma y color:SolidPeso molecular:371.312UCB-35440
CAS:<p>UCB-35440, a 5-lipoxygenase inhibitor and a histamine H1 receptor antagonist, is used potentially for the treatment of dermatitis.</p>Fórmula:C31H34ClN5O4Forma y color:SolidPeso molecular:576.09Minocromil
CAS:<p>Minocromil is a new agent of Anti-asthmatic.</p>Fórmula:C18H16N2O6Pureza:98%Forma y color:SolidPeso molecular:356.33A-349821
CAS:<p>A-349821 is an H3 receptor agonist radioligand.</p>Fórmula:C28H35F3N2O5Forma y color:SolidPeso molecular:536.59GT-2331
CAS:<p>GT-2331 is a histamine H3 receptor antagonist.</p>Fórmula:C14H20N2Forma y color:SolidPeso molecular:216.32Levocabastine
CAS:<p>Levocarbastine: 2nd-gen H1 antagonist, treats allergic conjunctivitis, selective NTS2 neurotensin inhibitor.</p>Fórmula:C26H29FN2O2Forma y color:SolidPeso molecular:420.52H3 receptor antagonist 1
CAS:<p>H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.</p>Fórmula:C20H28F2N2OPureza:98%Forma y color:SolidPeso molecular:350.45H4R antagonist 2
CAS:<p>H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid</p>Fórmula:C13H17N5OPureza:98%Forma y color:SolidPeso molecular:259.31Cipralisant
CAS:<p>Cipralisant: H3 receptor antagonist (in vivo), agonist (in vitro, pKi 9.9), Ki 0.47 nM in rats, may treat ADHD.</p>Fórmula:C14H20N2Pureza:98%Forma y color:SolidPeso molecular:216.32Levocabastine hydrochloride
CAS:<p>Levocabastine HCl is an agent with antihistaminic activity.</p>Fórmula:C26H30ClFN2O2Forma y color:SolidPeso molecular:456.98ST-1006
CAS:<p>ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.</p>Fórmula:C16H20Cl2N6Pureza:98.87% - 99.96%Forma y color:SolidPeso molecular:367.28Enerisant
CAS:<p>Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.</p>Fórmula:C22H30N4O3Pureza:99.7%Forma y color:SoildPeso molecular:398.50Tixanox sodium
CAS:<p>Tixanox sodium effectively blocks histamine release in the lungs triggered by anti-IgE. It has also been demonstrated that when administered orally, Tixanox sodium can successfully counteract exercise-induced asthma.</p>Fórmula:C15H9NaO5SForma y color:SolidPeso molecular:324.28CI-624
CAS:<p>CI-624 reduces the secretion and output of hydrogen ions, sodium ions, potassium ions, and pepsin. This compound may be utilized in research focusing on cancer and autoimmune diseases.</p>Fórmula:C8H8N2SForma y color:SolidPeso molecular:164.228H3R antagonist 5
CAS:<p>H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.</p>Fórmula:C23H32N2O4Forma y color:SolidPeso molecular:400.511Arpromidine
CAS:<p>Arpromidine (BU-E-50) acts as an agonist for the histamine H2 receptor and an antagonist for the histamine H1 receptor. It demonstrates positive inotropic effects with a lower risk of inducing arrhythmias. Arpromidine can be utilized in studies related to congestive heart failure.</p>Fórmula:C21H25FN6Forma y color:SolidPeso molecular:380.462H1R ligand-1
CAS:<p>H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R). It can serve as a scaffold for synthesizing a series of derivatives to investigate H1R binding kinetics.</p>Fórmula:C19H23NOForma y color:SolidPeso molecular:281.392Nedocromil sodium
CAS:<p>Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.</p>Fórmula:C19H17NNaO7Pureza:98%Forma y color:SolidPeso molecular:394.335UR-AK49
CAS:<p>UR-AK49 (compound 11) is an agonist for the human histamine H1 and H2 receptors. It exhibits an EC50 of 23 nM in the GTPase assay involving hH2R-Gsalpha fusion protein expressed in Sf9 insect cells. UR-AK49 is applicable in neurologically related research.</p>Fórmula:C16H27N5OForma y color:SolidPeso molecular:305.42FR-145715
CAS:<p>FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This compound is utilized in the study of gastric lesions.</p>Fórmula:C16H21N5O2SForma y color:SolidPeso molecular:347.44Histamine H3 antagonist-1
CAS:<p>Compound 10o, a histamine H3 antagonist-1, functions as both a histamine H3 antagonist and a serotonin reuptake inhibitor, making it useful for research in depression [1].</p>Fórmula:C24H28F3N3O2Forma y color:SolidPeso molecular:447.49H3R antagonist 1
CAS:<p>H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).</p>Fórmula:C19H23N3O3Forma y color:SolidPeso molecular:341.4(R)-(-)-α-Methylhistamine dihydrochloride
CAS:<p>R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.</p>Fórmula:C6H13Cl2N3Forma y color:SolidPeso molecular:198.09Imetit dihydrobromide
CAS:<p>Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).</p>Fórmula:C6H12Br2N4SPureza:98%Forma y color:SolidPeso molecular:332.06
