Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 389 productos para "Receptor de histamina".
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Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Fórmula:C21H24ClNOPureza:99.77% - 99.99%Forma y color:White SolidPeso molecular:341.88Fexofenadine hydrochloride
CAS:Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, withFórmula:C32H40ClNO4Pureza:>99.99%Forma y color:White SolidPeso molecular:538.12Pemirolast potassium
CAS:Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Fórmula:C10H7KN6OPureza:98.91% - 99.63%Forma y color:SolidPeso molecular:266.31Levodropropizine
CAS:Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.Fórmula:C13H20N2O2Pureza:99.87% - 99.89%Forma y color:SolidPeso molecular:236.31Fenspiride hydrochloride
CAS:Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Forma y color:SolidPeso molecular:296.79Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Forma y color:SolidPeso molecular:461.81Chloropyramine hydrochloride
CAS:Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.Fórmula:C16H20ClN3·HClPureza:99.45% - 99.83%Forma y color:White SolidPeso molecular:326.26Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Fórmula:C21H28N2O5Pureza:99.61%Forma y color:White SolidPeso molecular:388.46Mepyramine maleate
CAS:Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.Fórmula:C21H27N3O5Pureza:99.51% - 99.92%Forma y color:SolidPeso molecular:401.47Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Fórmula:C19H19NSPureza:97.50%Forma y color:SolidPeso molecular:293.43Ref: TM-T12489
2mg33,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg62,00€25mg101,00€50mg149,00€100mg215,00€200mg320,00€Methapyrilene hydrochloride
CAS:Methapyrilene hydrochloride is a biochemical.Fórmula:C14H20ClN3SForma y color:SolidPeso molecular:297.85Betahistine mesylate
CAS:Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.Fórmula:C8H12N2·2(CH4O3S)Pureza:98% - 99.85%Forma y color:SolidPeso molecular:328.4Sufotidine
CAS:Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.Fórmula:C20H31N5O3SPureza:99.03% - 99.92%Forma y color:SolidPeso molecular:421.56Granuliberin R
CAS:Granuliberin R, a dodecapeptide from Rana rugosa skin, induces histamine release by degranulating rat mast cells.Fórmula:C69H103N19O14Forma y color:SolidPeso molecular:1422.68Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Fórmula:C21H31N3O3Pureza:99.59%Forma y color:SolidPeso molecular:373.49Ref: TM-T9770
1mg105,00€2mg158,00€5mg260,00€1mL*10mM (DMSO)268,00€10mg416,00€25mg687,00€50mg964,00€100mg1.288,00€500mg2.602,00€Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Fórmula:C10H20ClNO4Pureza:90% - 99.77%Forma y color:White SolidPeso molecular:253.72Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Forma y color:Odour SolidDonetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Fórmula:C20H25N5O3SPureza:99.32%Forma y color:SolidPeso molecular:415.51Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCSForma y color:Odour SolidRef: TM-L3300
1mgA consultar10μL*10mM (DMSO)A consultar20μL*10mM (DMSO)A consultar30μL*10mM (DMSO)A consultar50μL*10mM (DMSO)A consultar100μL*10mM (DMSO)A consultar250μL*10mM (DMSO)A consultarCetirizine-D8 dihydrochloride
CAS:Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Fórmula:C21H26Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:433.4Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFórmula:C26H27N3OPureza:98%Forma y color:SolidPeso molecular:397.51Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:99.77% - 99.86%Forma y color:SolidPeso molecular:296.37Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Fórmula:C19H28N4O4SPureza:98.48%Forma y color:SolidPeso molecular:408.52Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Fórmula:C24H41BrN2Forma y color:SolidPeso molecular:437.51Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Fórmula:C21H27Cl3N2O3Forma y color:SolidPeso molecular:461.814-Methylhistamine
CAS:4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFórmula:C6H11N3Pureza:98%Forma y color:SolidPeso molecular:125.17Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFórmula:C7H13N3O2Pureza:>99.99%Forma y color:Yellow OilPeso molecular:171.2AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Fórmula:C27H19F3N4O4SForma y color:SolidPeso molecular:552.52Dalcotidine
CAS:Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.Fórmula:C18H29N3O2Pureza:99.09%Forma y color:Yellow SolidPeso molecular:319.44Ref: TM-T31195
1mg63,00€5mg140,00€1mL*10mM (DMSO)140,00€10mg200,00€25mg324,00€50mg470,00€100mg662,00€200mg893,00€Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Fórmula:C21H25ClN2O3Forma y color:SolidPeso molecular:388.89Oxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.Fórmula:C20H23N5O5SPureza:97.34%Forma y color:SoildPeso molecular:445.49KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Fórmula:C26H28N4O3Pureza:97.51%Forma y color:SolidPeso molecular:444.53Dexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Fórmula:C16H19ClN2Pureza:98%Forma y color:SolidPeso molecular:274.79(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Fórmula:C22H25Cl2N3OPureza:98%Forma y color:SolidPeso molecular:418.36Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Fórmula:C10H19Br2N3Forma y color:SolidPeso molecular:341.0913-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Fórmula:C19H19ClN2OForma y color:SolidPeso molecular:326.82JNJ-10181457 (hydrochloride)
CAS:JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFórmula:C20H30Cl2N2OForma y color:SolidPeso molecular:385.37Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Fórmula:C30H28Cl2N2Forma y color:SolidPeso molecular:487.46Tecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Fórmula:C19H21FN4Pureza:99.70%Forma y color:SolidPeso molecular:324.4Ref: TM-T26253
1mg54,00€5mg118,00€1mL*10mM (DMSO)131,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mg1.161,00€Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Fórmula:C19H21N5O3SPureza:99.71%Forma y color:White SolidPeso molecular:399.47Ref: TM-T68122
1mg358,00€5mg848,00€10mg1.153,00€25mg1.693,00€50mg2.313,00€100mg3.115,00€500mg6.255,00€Histamine H4 receptor antagonist-1
CAS:Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Fórmula:C30H38N8O2Forma y color:SolidPeso molecular:542.68Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Fórmula:C19H21N3O2Forma y color:SolidPeso molecular:323.39Diphenhydramine hydrochloride
CAS:DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.Fórmula:C17H22ClNOPureza:99.84%Forma y color:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Peso molecular:291.82KSK67
CAS:KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with KiFórmula:C22H27N3O2Pureza:99.94%Forma y color:SolidPeso molecular:365.47(+)-Dropropizine
CAS:(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Fórmula:C13H20N2O2Pureza:>99.99%Forma y color:SolidPeso molecular:236.31H4R antagonist 3
CAS:H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study ofFórmula:C19H21ClN4SPureza:97.22%Forma y color:White SolidPeso molecular:372.92Nizatidine
CAS:Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Fórmula:C12H21N5O2S2Pureza:98.39% - 99.43%Forma y color:White SolidPeso molecular:331.46Diphenylpyraline
CAS:Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.Fórmula:C19H23NOForma y color:SolidPeso molecular:281.39Cetirizine-D4
CAS:Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Fórmula:C21H25ClN2O3Pureza:98%Forma y color:SolidPeso molecular:392.91Emedastine Difumarate
CAS:Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Fórmula:C25H34N4O9Forma y color:SolidPeso molecular:534.56
