Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Fórmula:C32H39NO4Pureza:98%Forma y color:SolidPeso molecular:507.69Cetirizine D4
CAS:<p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Forma y color:SolidPeso molecular:392.91Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Fórmula:C19H23NOForma y color:SolidPeso molecular:281.39WZ4141
CAS:<p>WZ4141 is an intermediate in compound synthesis.</p>Fórmula:C16H13N3O2Pureza:98%Forma y color:SolidPeso molecular:279.29Acrivastine D7
CAS:<p>Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.</p>Fórmula:C22H24N2O2Pureza:98%Forma y color:SolidPeso molecular:355.48Doxepin D3 Hydrochloride
CAS:<p>Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and</p>Fórmula:C19H22ClNOPureza:98%Forma y color:SolidPeso molecular:318.86Emedastine Difumarate
CAS:<p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>Fórmula:C25H34N4O9Forma y color:SolidPeso molecular:534.56Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98%Forma y color:SolidPeso molecular:396.94Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Fórmula:C8H12N2Pureza:99.87% - 99.87%Forma y color:Yellowish Liquid Liquid LiquidPeso molecular:136.19S 38093
CAS:<p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>Fórmula:C17H24N2O2Pureza:99.95%Forma y color:SolidPeso molecular:288.38GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Fórmula:C21H25N3O2Pureza:98.71% - 99.858%Forma y color:SolidPeso molecular:351.44Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Fórmula:C17H26N4OPureza:97.1% - 97.76%Forma y color:OilPeso molecular:302.41Fexofenadine hydrochloride
CAS:<p>Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,</p>Fórmula:C32H39NO4·HClPureza:99.39% - ≥95%Forma y color:SolidPeso molecular:538.13Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Fórmula:C28H33ClN2·2HClPureza:98.05%Forma y color:Off-White PowderPeso molecular:505.95Conessine
CAS:<p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>Fórmula:C24H40N2Pureza:99.65%Forma y color:SolidPeso molecular:356.59Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Fórmula:C16H19ClN2Forma y color:SolidPeso molecular:274.79Dioxopromethazine hydrochloride
CAS:<p>Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.</p>Fórmula:C17H20N2O2S·HClPureza:99.58%Forma y color:SolidPeso molecular:352.88Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Fórmula:C21H27ClN2O2Pureza:99.54% - ≥95%Forma y color:Oil SolidPeso molecular:374.9SCH-37370
CAS:<p>SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.</p>Fórmula:C21H21ClN2OPureza:99.07%Forma y color:SolidPeso molecular:352.86H4 Receptor antagonist 1
CAS:<p>H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.</p>Fórmula:C16H17ClN4OPureza:98.81%Forma y color:SolidPeso molecular:316.79Triprolidine
CAS:<p>Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.</p>Fórmula:C19H22N2Forma y color:SolidPeso molecular:278.39Fenspiride
CAS:<p>Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.</p>Fórmula:C15H20N2O2Forma y color:SolidPeso molecular:260.33Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Forma y color:SolidPeso molecular:241.33Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Fórmula:C28H37N3O3Pureza:99.86% - >99.99%Forma y color:SolidPeso molecular:463.61Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Fórmula:C19H21Cl2N3Pureza:>99.99%Forma y color:SolidPeso molecular:362.3Clobenpropit dihydrobromide
CAS:<p>Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)</p>Fórmula:C14H19Br2ClN4SPureza:99.86%Forma y color:SolidPeso molecular:470.7Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Forma y color:SolidPeso molecular:477.57Antazoline
CAS:<p>Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.</p>Fórmula:C17H19N3Pureza:≥95%Forma y color:White Crystalline Powder SolidPeso molecular:265.35Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Fórmula:C21H28N2O2Pureza:99.53%Forma y color:White Or Similar To White PowderPeso molecular:340.46Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Forma y color:SolidPeso molecular:356.442-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Fórmula:C7H12Cl2N2Pureza:99.42%Forma y color:SolidPeso molecular:195.09Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86Clobenpropit 2HBr
CAS:<p>Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.</p>Fórmula:C14H17ClN4SForma y color:SolidPeso molecular:308.83Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Fórmula:C11H6ClN3O6Pureza:99.13% - 99.81%Forma y color:SolidPeso molecular:311.63cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Fórmula:C16H14O2Pureza:98.15%Forma y color:SolidPeso molecular:238.2812Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Forma y color:SolidPeso molecular:233.18Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Fórmula:C15H19Cl2N3O3SPureza:98.48%Forma y color:SolidPeso molecular:392.3HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Fórmula:C27H33F3N4O9Pureza:99.51%Forma y color:SolidPeso molecular:614.57Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Fórmula:C19H23ClN2Forma y color:SolidPeso molecular:314.852Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Fórmula:C29H34O6Pureza:≥98%Forma y color:LiquidPeso molecular:478.58Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Fórmula:C17H20N2O2SPureza:98%Forma y color:SolidPeso molecular:316.42Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Fórmula:C14H20F6N4O7Pureza:98.18%Forma y color:SolidPeso molecular:470.32Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Fórmula:C28H33ClN2Forma y color:SolidPeso molecular:433.03Desloratadine
CAS:<p>Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.</p>Fórmula:C19H19ClN2Pureza:99.79% - >99.99%Forma y color:SolidPeso molecular:310.82Fexofenadine
CAS:<p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>Fórmula:C32H39NO4Pureza:99.35%Forma y color:White To Off-White SolidPeso molecular:501.66JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Fórmula:C20H34Cl2N2OPureza:99.51%Forma y color:SolidPeso molecular:389.4Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Fórmula:C21H25ClN2O3·C6H6O3SPureza:99.83% - 99.9%Forma y color:Brown Viscous LiquidPeso molecular:547.06Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Fórmula:C19H22ClN3OPureza:98%Forma y color:SolidPeso molecular:343.86VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Fórmula:C15H19N5Pureza:99.44% - 99.57%Forma y color:SolidPeso molecular:269.34
