Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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Benztropine mesylate
CAS:Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Forma y color:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Hydroxyzine Pamoate
CAS:Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.Fórmula:C44H43ClN2O8Pureza:99.49%Forma y color:SolidPeso molecular:763.27Pemirolast potassium
CAS:Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.Fórmula:C10H7KN6OPureza:98.91% - 99.63%Forma y color:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Fórmula:C19H29ClN2O4Pureza:99.49%Forma y color:SolidPeso molecular:384.9Cyproheptadine hydrochloride sesquihydrate
CAS:Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Fórmula:C21H24ClNOPureza:99.77% - >99.99%Forma y color:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Fórmula:C21H25ClN2O3Pureza:98% - 99.94%Forma y color:White PowderPeso molecular:388.89Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Fórmula:C13H16N4Pureza:98.34% - 99.73%Forma y color:SolidPeso molecular:228.29MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.Fórmula:C24H26F3N3O4Pureza:99.98%Forma y color:SolidPeso molecular:477.48Ketotifen fumarate
CAS:Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.Fórmula:C23H23NO5SPureza:99.25% - 99.73%Forma y color:SolidPeso molecular:425.50Mebhydrolin napadisylate
CAS:Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.96%Forma y color:White Or Almost White CrystallinePeso molecular:420.52Mizolastine
CAS:Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.Fórmula:C24H25FN6OPureza:98% - 99.75%Forma y color:SolidPeso molecular:432.49Terfenadine
CAS:Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Fórmula:C32H41NO2Pureza:98.76% - 99.75%Forma y color:SolidPeso molecular:471.67Doxepin hydrochloride
CAS:Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Fórmula:C19H22ClNOPureza:99.65% - 99.91%Forma y color:White To Off-White PowderPeso molecular:315.84Doxylamine succinate
CAS:Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.Fórmula:C21H28N2O5Pureza:99.61%Forma y color:5 1 (Ntp 1992)Peso molecular:388.46Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Fórmula:C19H21N3OPureza:99.44% - 99.84%Forma y color:SolidPeso molecular:307.39Cinnarizine
CAS:Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Fórmula:C26H28N2Pureza:99.94%Forma y color:SolidPeso molecular:368.51Carbinoxamine Maleate Salt
CAS:Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.Fórmula:C20H23ClN2O5Pureza:99.97%Forma y color:Off-White SolidPeso molecular:406.86Clemastine fumarate
CAS:Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.Fórmula:C25H30ClNO5Pureza:99.52% - >99.99%Forma y color:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderPeso molecular:459.97Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Forma y color:SolidPeso molecular:350.86Diphenylpyraline hydrochloride
CAS:Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.Fórmula:C19H23NO·HClPureza:98.72%Forma y color:SolidPeso molecular:317.85
