
Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Samelisant
CAS:<p>Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.</p>Fórmula:C21H31N3O3Pureza:99.59%Forma y color:SolidPeso molecular:373.49Roxatidine
CAS:<p>Roxatidine, a metabolite of Roxatidine acetate, is a H2-receptor antagonist that prevents ulcers and has anti-inflammatory properties.</p>Fórmula:C17H26N2O3Forma y color:SolidPeso molecular:306.4Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Fórmula:C21H25ClN2O3Forma y color:SolidPeso molecular:388.89Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Fórmula:C14H20ClN3SForma y color:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85Cetirizine methyl ester
CAS:<p>Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.</p>Fórmula:C22H27ClN2O3Forma y color:SolidPeso molecular:402.91Diphenhydramine hydrochloride
CAS:<p>DPH: antihistamine for cough, nausea, itching, allergy, Parkinson's, sleep aid, cold remedy.</p>Fórmula:C17H22ClNOPureza:99.84%Forma y color:Taste Ph (5% Aqueous Solution) 4-6 (Ntp 1992)Peso molecular:291.82Donetidine
CAS:<p>Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.</p>Fórmula:C20H25N5O3SPureza:99.32%Forma y color:SolidPeso molecular:415.51Cetirizine Impurity C dihydrochloride
CAS:<p>Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.</p>Fórmula:C21H27Cl3N2O3Forma y color:SolidPeso molecular:461.81Levocarnitine propionate hydrochloride
CAS:<p>Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.</p>Fórmula:C10H20ClNO4Pureza:90% - 99.77%Forma y color:SolidPeso molecular:253.72Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Forma y color:Odour SolidBodilisant
CAS:<p>Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.</p>Fórmula:C27H34BF2N3OForma y color:SolidPeso molecular:465.4Nizatidine
CAS:<p>Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.</p>Fórmula:C12H21N5O2S2Pureza:99.43%Forma y color:White To Off-White Crystalline PowderPeso molecular:331.46Vapitadine
CAS:<p>Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.</p>Fórmula:C17H20N4OPureza:99.77% - 99.86%Forma y color:SoildPeso molecular:296.37(S)-Azelastine hydrochloride
CAS:<p>(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Fórmula:C22H25Cl2N3OPureza:98%Forma y color:SolidPeso molecular:418.36Histamine H4 receptor antagonist-1
CAS:<p>Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.</p>Fórmula:C30H38N8O2Forma y color:SolidPeso molecular:542.68Tecastemizole
CAS:<p>Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.</p>Fórmula:C19H21FN4Pureza:99.70%Forma y color:SolidPeso molecular:324.4Dexchlorpheniramine free base
CAS:<p>Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.</p>Fórmula:C16H19ClN2Pureza:98%Forma y color:Oily Liquid SolidPeso molecular:274.79Sufotidine
CAS:<p>Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.</p>Fórmula:C20H31N5O3SPureza:99.03% - 99.92%Forma y color:SolidPeso molecular:421.56JNJ-10181457 (hydrochloride)
CAS:<p>JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrations</p>Fórmula:C20H30Cl2N2OForma y color:SolidPeso molecular:385.37Conessine hydrobromide
CAS:<p>Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.</p>Fórmula:C24H41BrN2Forma y color:SolidPeso molecular:437.51
