Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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KSK67
CAS:KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with KiFórmula:C22H27N3O2Pureza:99.94%Forma y color:SoildPeso molecular:365.47Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Fórmula:C21H25ClN2O3Forma y color:SolidPeso molecular:388.89Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Fórmula:C21H27Cl3N2O3Forma y color:SolidPeso molecular:461.81Methapyrilene hydrochloride
CAS:Methapyrilene hydrochloride is a biochemical.Fórmula:C14H20ClN3SForma y color:Liquid Solution) 5 5 (Ntp 1992)Peso molecular:297.85Cetirizine methyl ester
CAS:Cetirizine methyl ester is a Cetirizine impurity, a long-acting, oral H1-antihistamine and hydroxyzine metabolite.Fórmula:C22H27ClN2O3Forma y color:SolidPeso molecular:402.91AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Fórmula:C27H19F3N4O4SForma y color:SolidPeso molecular:552.523-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Fórmula:C19H19ClN2OForma y color:SolidPeso molecular:326.82Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Fórmula:C10H19Br2N3Forma y color:SolidPeso molecular:341.091Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Fórmula:C20H25N5O3SPureza:99.32%Forma y color:SolidPeso molecular:415.51Bodilisant
CAS:Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Fórmula:C27H34BF2N3OForma y color:SolidPeso molecular:465.4Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Fórmula:C21H31N3O3Pureza:99.59%Forma y color:SolidPeso molecular:373.49Ref: TM-T9770
1mg105,00€2mg158,00€5mg260,00€10mg416,00€25mg687,00€50mg964,00€100mg1.288,00€500mg2.602,00€1mL*10mM (DMSO)268,00€Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Fórmula:C10H20ClNO4Pureza:90% - 99.77%Forma y color:SolidPeso molecular:253.72Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Forma y color:Odour Solid(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Fórmula:C22H25Cl2N3OPureza:98%Forma y color:SolidPeso molecular:418.36Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS
Forma y color:Odour SolidNizatidine
CAS:Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Fórmula:C12H21N5O2S2Pureza:99.43%Forma y color:White To Off-White Crystalline PowderPeso molecular:331.46Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:99.77% - 99.86%Forma y color:SoildPeso molecular:296.37Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Fórmula:C19H21N3O2Forma y color:SolidPeso molecular:323.39Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Fórmula:C19H28N4O4SPureza:98.48%Forma y color:SolidPeso molecular:408.52Tecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Fórmula:C19H21FN4Pureza:99.70%Forma y color:SolidPeso molecular:324.4Ref: TM-T26253
1mg54,00€5mg118,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mg1.161,00€1mL*10mM (DMSO)131,00€
