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Receptor de histamina

Receptor de histamina

Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.

Se han encontrado 388 productos para "Receptor de histamina".

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  • Methapyrilene hydrochloride

    CAS:
    Methapyrilene hydrochloride is a biochemical.
    Fórmula:C14H20ClN3S
    Forma y color:Solid
    Peso molecular:297.85

    Ref: TM-T33316

    100mg
    241,00€
    250mg
    572,00€
  • 3-hydroxy Desloratidine

    CAS:
    3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.
    Fórmula:C19H19ClN2O
    Forma y color:Solid
    Peso molecular:326.82

    Ref: TM-T36119

    500µg
    166,00€
  • Methimepip dihydrobromide

    CAS:
    Methimepip dihydrobromide is a selective H3R agonist.
    Fórmula:C10H19Br2N3
    Forma y color:Solid
    Peso molecular:341.091

    Ref: TM-T37727

    200mg
    1.304,00€
  • AM-0466

    CAS:
    AM-0466 has a wide range of applications in life science related research.
    Fórmula:C27H19F3N4O4S
    Forma y color:Solid
    Peso molecular:552.52

    Ref: TM-T71696

    5mg
    964,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Granuliberin R

    CAS:
    Granuliberin R, a dodecapeptide from Rana rugosa skin, induces histamine release by degranulating rat mast cells.
    Fórmula:C69H103N19O14
    Forma y color:Solid
    Peso molecular:1422.68

    Ref: TM-T76095

    5mg
    A consultar
    50mg
    A consultar
  • Samelisant

    CAS:
    Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.
    Fórmula:C21H31N3O3
    Pureza:99.59%
    Forma y color:Solid
    Peso molecular:373.49

    Ref: TM-T9770

    1mg
    105,00€
    2mg
    158,00€
    5mg
    260,00€
    1mL*10mM (DMSO)
    268,00€
    10mg
    416,00€
    25mg
    687,00€
    50mg
    964,00€
    100mg
    1.288,00€
    500mg
    2.602,00€
  • Conessine hydrobromide

    CAS:
    Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.
    Fórmula:C24H41BrN2
    Forma y color:Solid
    Peso molecular:437.51

    Ref: TM-T31006

    100mg
    A consultar
    500mg
    A consultar
  • Levocarnitine propionate hydrochloride

    CAS:
    Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.
    Fórmula:C10H20ClNO4
    Pureza:90% - 99.77%
    Forma y color:White Solid
    Peso molecular:253.72

    Ref: TM-T1182

    25mg
    34,00€
    1mL*10mM (DMSO)
    34,00€
    50mg
    48,00€
    100mg
    62,00€
    500mg
    144,00€
  • Neurotransmitter Receptor Compound Library


    A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;

    Forma y color:Odour Solid

    Ref: TM-L2610

    1mg
    A consultar
  • Nizatidine

    CAS:
    Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.
    Fórmula:C12H21N5O2S2
    Pureza:98.39% - 99.43%
    Forma y color:White Solid
    Peso molecular:331.46

    Ref: TM-T1575

    1g
    33,00€
    1mL*10mM (DMSO)
    33,00€
    5g
    46,00€
    10g
    69,00€
  • Donetidine

    CAS:
    Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
    Fórmula:C20H25N5O3S
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:415.51

    Ref: TM-T68056

    1mg
    57,00€
    5mg
    124,00€
    10mg
    182,00€
    25mg
    298,00€
    50mg
    434,00€
    100mg
    620,00€
    200mg
    837,00€
  • Vapitadine

    CAS:
    Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
    Fórmula:C17H20N4O
    Pureza:99.77% - 99.86%
    Forma y color:Solid
    Peso molecular:296.37

    Ref: TM-T29096L

    1mg
    175,00€
    5mg
    434,00€
    10mg
    622,00€
    25mg
    973,00€
    50mg
    1.865,00€
  • Histamine H4 receptor antagonist-1

    CAS:
    Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
    Fórmula:C30H38N8O2
    Forma y color:Solid
    Peso molecular:542.68

    Ref: TM-T38634

    100mg
    A consultar
    500mg
    A consultar
  • Cetirizine Impurity C dihydrochloride

    CAS:
    Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.
    Fórmula:C21H27Cl3N2O3
    Forma y color:Solid
    Peso molecular:461.81

    Ref: TM-T73962

    5mg
    A consultar
    50mg
    A consultar
  • (S)-Azelastine hydrochloride

    CAS:
    (S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Fórmula:C22H25Cl2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:418.36

    Ref: TM-T21109

    1mg
    364,00€
  • (+)-Dropropizine

    CAS:
    (+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.
    Fórmula:C13H20N2O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:236.31

    Ref: TM-T0217L

    1g
    47,00€
  • Cetirizine Impurity C

    CAS:
    Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.
    Fórmula:C21H25ClN2O3
    Forma y color:Solid
    Peso molecular:388.89

    Ref: TM-T36945

    5mg
    109,00€
  • Alcaftadine carboxylic acid

    CAS:
    Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.
    Fórmula:C19H21N3O2
    Forma y color:Solid
    Peso molecular:323.39

    Ref: TM-T25033

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Dexchlorpheniramine free base

    CAS:
    Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.
    Fórmula:C16H19ClN2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:274.79

    Ref: TM-T0785L

    25mg
    1.369,00€
  • Cetirizine-D8 dihydrochloride

    CAS:
    Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.
    Fórmula:C21H26Cl2N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:433.4

    Ref: TM-T19234

    500µg
    500,00€
    1mg
    945,00€