
Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 388 productos para "Receptor de histamina".
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Methapyrilene hydrochloride
CAS:Methapyrilene hydrochloride is a biochemical.Fórmula:C14H20ClN3SForma y color:SolidPeso molecular:297.853-hydroxy Desloratidine
CAS:3-hydroxy Desloratidine is a major metabolite of desloratadine , a tricyclic antagonist of the histamine H1 receptor.Fórmula:C19H19ClN2OForma y color:SolidPeso molecular:326.82Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Fórmula:C10H19Br2N3Forma y color:SolidPeso molecular:341.091AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Fórmula:C27H19F3N4O4SForma y color:SolidPeso molecular:552.52Granuliberin R
CAS:Granuliberin R, a dodecapeptide from Rana rugosa skin, induces histamine release by degranulating rat mast cells.Fórmula:C69H103N19O14Forma y color:SolidPeso molecular:1422.68Samelisant
CAS:Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Fórmula:C21H31N3O3Pureza:99.59%Forma y color:SolidPeso molecular:373.49Ref: TM-T9770
1mg105,00€2mg158,00€5mg260,00€1mL*10mM (DMSO)268,00€10mg416,00€25mg687,00€50mg964,00€100mg1.288,00€500mg2.602,00€Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Fórmula:C24H41BrN2Forma y color:SolidPeso molecular:437.51Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Fórmula:C10H20ClNO4Pureza:90% - 99.77%Forma y color:White SolidPeso molecular:253.72Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;
Forma y color:Odour SolidNizatidine
CAS:Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity.Fórmula:C12H21N5O2S2Pureza:98.39% - 99.43%Forma y color:White SolidPeso molecular:331.46Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Fórmula:C20H25N5O3SPureza:99.32%Forma y color:SolidPeso molecular:415.51Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Fórmula:C17H20N4OPureza:99.77% - 99.86%Forma y color:SolidPeso molecular:296.37Histamine H4 receptor antagonist-1
CAS:Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.Fórmula:C30H38N8O2Forma y color:SolidPeso molecular:542.68Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Fórmula:C21H27Cl3N2O3Forma y color:SolidPeso molecular:461.81(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Fórmula:C22H25Cl2N3OPureza:98%Forma y color:SolidPeso molecular:418.36(+)-Dropropizine
CAS:(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex.Fórmula:C13H20N2O2Pureza:>99.99%Forma y color:SolidPeso molecular:236.31Cetirizine Impurity C
CAS:Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Fórmula:C21H25ClN2O3Forma y color:SolidPeso molecular:388.89Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Fórmula:C19H21N3O2Forma y color:SolidPeso molecular:323.39Dexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Fórmula:C16H19ClN2Pureza:98%Forma y color:SolidPeso molecular:274.79Cetirizine-D8 dihydrochloride
CAS:Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Fórmula:C21H26Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:433.4
