Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 325 productos de "Receptor de opioides"
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(Rac)-SNC80
CAS:(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.Fórmula:C28H39N3O2Forma y color:SolidPeso molecular:449.63Deltorphin
CAS:Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.Fórmula:C44H62N10O10S2Pureza:98.96%Forma y color:SolidPeso molecular:955.15Ac-RYYRWK-NH2
CAS:Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.Fórmula:C49H69N15O9Pureza:98%Forma y color:SolidPeso molecular:1012.17β-Endorphin (6-31), human
CAS:β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.Fórmula:C131H218N34O40Pureza:98%Forma y color:SolidPeso molecular:2909.38β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Fórmula:C141H221N33O42SPureza:96.52%Forma y color:SolidPeso molecular:3082.52Naldemedine
CAS:Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.Fórmula:C32H34N4O6Forma y color:SolidPeso molecular:570.64SNC 80
CAS:SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Fórmula:C28H39N3O2Pureza:99.65%Forma y color:SolidPeso molecular:449.63[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway ofFórmula:C31H43N5O9Pureza:98%Forma y color:SolidPeso molecular:629.65DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Fórmula:C30H39N5O7S2Pureza:98%Forma y color:SolidPeso molecular:645.79Acetalin-2
CAS:Acetalin-2, an opioid peptide with the sequence Ac-Arg-Phe-Met-Trp-Met-Arg-NH2, selectively binds to [3 H]DAMGO with a Ki value of 93.3 nM [1].Fórmula:C44H66N14O7S2Peso molecular:967.21[Arg14,Lys15]Nociceptin
CAS:Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.Fórmula:C82H137N31O22Pureza:98%Forma y color:SolidPeso molecular:1909.18difelikefalin acetate(1024828-77-0 Free base)
CAS:is a ketone and a building block.
Fórmula:C38H57N7O8Pureza:96.94%Forma y color:SolidPeso molecular:739.9UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Fórmula:C84H142N32O23Pureza:95.92%Forma y color:SolidPeso molecular:1968.23β-Endorphin, equine
CAS:Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.Fórmula:C154H248N42O44SPureza:98%Forma y color:SolidPeso molecular:3423.94CTOP acetate
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.Fórmula:C52H71N11O13S2Pureza:99.87%Forma y color:SoildPeso molecular:1122.32MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Fórmula:C27H29ClN4O2Pureza:98%Forma y color:SolidPeso molecular:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,
Pureza:99.89%Forma y color:Soildβ-Lipotropin (61-69)
CAS:β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Fórmula:C45H66N10O15SPeso molecular:1019.13Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Fórmula:C30H33ClN2O7SForma y color:SolidPeso molecular:601.11Axelopran sulfate
CAS:Axelopran sulfate is used in Oral Therapies for Opioid-induced Bowel Dysfunction in Patients with Chronic Noncancer Pain.Fórmula:C26H41N3O8SForma y color:SolidPeso molecular:555.68Acetalin-3
CAS:Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Fórmula:C42H61N11O8S2Peso molecular:912.13[Met5]-Enkephalin, amide
CAS:[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.Fórmula:C27H36N6O6SPureza:98%Forma y color:SolidPeso molecular:572.68PL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Fórmula:C31H38F3N5O7Peso molecular:649.66BPRMU191
CAS:BPRMU191 is a distinct mu-opioid receptor (MOR) modulator with an EC50 of 2.17 μM in FLIPR Ca2+ assays conducted on CHO-K1/MOR/Gα15 cells. Additionally, BPRMU191 interacts with MOR in the presence of naloxone.Fórmula:C17H14FNO3SForma y color:SolidPeso molecular:331.36DuP 747 HCl
CAS:DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.Fórmula:C24H29Cl3N2O2Pureza:99.85%Forma y color:SoildPeso molecular:483.86[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.Fórmula:C65H107N21O15Pureza:99.59%Forma y color:SoildPeso molecular:1422.7[D-Ala2]-Met-Enkephalinamide
CAS:[D-Ala2]-Met-Enkephalinamide: potent opioid, reduces bile flow centrally, analgesic.Fórmula:C28H38N6O6SPeso molecular:586.7Bilaid C
CAS:Bilaid C: Tetrapeptide μ-opioid agonist from Penicillium (Ki=210 nM), inhibits cAMP (77% at 10 μM), induces Kir currents (EC50=4.2 μM).Fórmula:C28H38N4O6Peso molecular:526.62K-Opioid receptor agonist-1
CAS:K-Opioid receptor agonist-1 (Compound 5a) acts as an agonist for the κ-Opioid receptor, exhibiting a K_i of 0.25 nM and an EC_50 of 2 nM. This compound is capable of crossing the blood-brain barrier (BBB), evidenced by brain/plasma ratios ranging from 0.50 to 0.65. Additionally, K-Opioid receptor agonist-1 demonstrates anti-inflammatory effects in dermatitis models induced by either Arachidonic acid or oxazolidinone.Fórmula:C22H29Cl2N3O3Peso molecular:454.39Morphiceptin
CAS:Morphiceptin is a synthetic tetrapeptide with morphinelike activities, highly specific for morphine receptors, but not for enkephalin receptors.Fórmula:C28H35N5O5Peso molecular:521.61(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS:E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioidFórmula:C50H81N15O9Forma y color:SolidPeso molecular:1036.27[Nphe1]Nociceptin(1-13)NH2 TFA
[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.Fórmula:C63H101F3N22O17Forma y color:SolidPeso molecular:1495.61Loperamide phenyl
CAS:Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.Fórmula:C35H37ClN2O2Forma y color:SolidPeso molecular:553.14BAN ORL 24 dihydrochloride
CAS:BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.Fórmula:C27H37Cl2N3O2Pureza:95.03%Forma y color:SolidPeso molecular:506.51Porcine dynorphin A(1-13)
CAS:Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.Fórmula:C75H126N24O15Pureza:98%Forma y color:SolidPeso molecular:1603.95BMS-986121
CAS:BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.Fórmula:C15H9Cl2N3O2SPureza:99.67%Forma y color:SolidPeso molecular:366.22Alvimopan dihydrate (LY246736 dihydrate)
CAS:Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.Fórmula:C25H36N2O6Forma y color:SolidPeso molecular:460.56Endomorphin 2 TFA
CAS:Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.Fórmula:C34H38F3N5O7Forma y color:SolidPeso molecular:685.69Asimadoline
CAS:Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54[Leu5]-Enkephalin
CAS:[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nMFórmula:C28H37N5O7Pureza:99.87% - 99.88%Forma y color:SolidPeso molecular:555.62Deltorphin 2
CAS:Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.Fórmula:C38H54N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:782.88Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Fórmula:C21H26BrNO4Pureza:99.02%Forma y color:SolidPeso molecular:436.35Corydaline
CAS:Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.
Fórmula:C22H27NO4Pureza:98.97% - 99.86%Forma y color:SolidPeso molecular:369.45Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Fórmula:C79H129N27O22Pureza:99.35%Forma y color:SolidPeso molecular:1809.04N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Forma y color:Yellow Crystalline SolidPeso molecular:312.8Ref: TM-T5158
2mg34,00€5mg48,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€1mL*10mM (DMSO)58,00€Sec-O-Glucosylhamaudol
CAS:Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.Fórmula:C21H26O10Pureza:99.79%Forma y color:SolidPeso molecular:438.43Dermorphin TFA
CAS:Dermorphin TFA is a new class of opioids-like peptidesFórmula:C42H51F3N8O12Pureza:98% - >99.99%Forma y color:SolidPeso molecular:916.89Naloxegol (NKTR-118)
CAS:Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].Fórmula:C34H53NO11Forma y color:SolidPeso molecular:651.78DPDPE TFA (88373-73-3 free base)
CAS:DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.Fórmula:C32H40F3N5O9S2Pureza:99.39%Forma y color:SolidPeso molecular:759.81Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Fórmula:C29H45N5O8Pureza:99.39%Forma y color:SolidPeso molecular:591.7Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Fórmula:C36H55NO15Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:741.83Nalmefene hydrochloride
CAS:Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.Fórmula:C21H26ClNO3Pureza:98% - 99.85%Forma y color:SolidPeso molecular:375.89ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFórmula:C24H28N2O3·HClPureza:98.78% - 99.11%Forma y color:SolidPeso molecular:428.95Ref: TM-T6175
1mg49,00€2mg66,00€5mg90,00€10mg166,00€25mg319,00€50mg492,00€100mg710,00€500mg1.468,00€1mL*10mM (DMSO)108,00€Alvimopan monohydrate
CAS:Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.Fórmula:C25H34N2O5Pureza:98%Forma y color:SolidPeso molecular:442.55MCOPPB
CAS:MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.Fórmula:C26H40N4Forma y color:SolidPeso molecular:408.62GR 89696 free base
CAS:GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.Fórmula:C19H25Cl2N3O3Forma y color:SolidPeso molecular:414.33EST73502 hydrochloride
CAS:EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.Fórmula:C19H27ClF2N2O2Forma y color:SolidPeso molecular:388.88LY2940094 tartrate
CAS:LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.Fórmula:C26H29ClF2N4O8SForma y color:SolidPeso molecular:631.04MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Fórmula:C26H43Cl3N4Pureza:99.89% - 99.91%Forma y color:SolidPeso molecular:518.01Ref: TM-T2071
2mg33,00€5mg52,00€10mg82,00€25mg155,00€50mg241,00€100mg355,00€200mg507,00€1mL*10mM (DMSO)55,00€Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Fórmula:C37H52N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:768.86Tyr-Gly-Gly-Phe-Met-OH
CAS:Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.
Fórmula:C27H35N5O7SPureza:≥95%Forma y color:White Lyophilised SolidPeso molecular:573.66Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Fórmula:C32H37N5O5Pureza:99.64%Forma y color:SolidPeso molecular:571.67EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Fórmula:C19H27ClF2N2O2Pureza:99.96%Forma y color:SolidPeso molecular:388.88Ref: TM-T39284
1mg96,00€5mg172,00€10mg244,00€25mg403,00€50mg567,00€100mg750,00€200mg1.018,00€1mL*10mM (DMSO)187,00€JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Fórmula:C26H25N3O2·HClPureza:99.27% - 99.59%Forma y color:SolidPeso molecular:447.96BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Fórmula:C16H15BrClNO3S2Pureza:98.42%Forma y color:SolidPeso molecular:448.78Ref: TM-T26869
1mg48,00€5mg96,00€10mg160,00€25mg311,00€50mg472,00€100mg658,00€200mg929,00€1mL*10mM (DMSO)96,00€Sinomenine
CAS:Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
Fórmula:C19H23NO4Pureza:99.02% - 99.73%Forma y color:White PowderPeso molecular:329.39ADL-5747 (HCl)
CAS:ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.Fórmula:C24H29ClN2O3Forma y color:SolidPeso molecular:428.95PZM21
CAS:PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
Fórmula:C19H27N3O2SPureza:99.93% - >99.99%Forma y color:SolidPeso molecular:361.5BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Fórmula:C31H34O4Pureza:99.09%Forma y color:SolidPeso molecular:470.6GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Fórmula:C23H29Cl2N3O7Pureza:99.75%Forma y color:SolidPeso molecular:530.4Ref: TM-T9459
1mg87,00€2mg143,00€5mg188,00€10mg283,00€25mg509,00€50mg727,00€100mg1.017,00€1mL*10mM (DMSO)250,00€LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Fórmula:C23H22ClN3O2Pureza:97.77%Forma y color:SolidPeso molecular:407.89Ref: TM-TQ0091
1mg52,00€2mg74,00€5mg116,00€10mg180,00€25mg298,00€50mgA consultar1mL*10mM (DMSO)127,00€DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Fórmula:C26H35N5O6Pureza:98.83% - 99.92%Forma y color:SolidPeso molecular:513.59Ref: TM-T4351
1mg50,00€2mg60,00€5mg87,00€10mg140,00€25mg283,00€50mg423,00€100mg623,00€1mL*10mM (DMSO)88,00€Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Fórmula:C50H72N15O15SPureza:>99.99%Forma y color:SolidPeso molecular:1326.26[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Fórmula:C29H39N5O7Pureza:98.06%Forma y color:SolidPeso molecular:569.65Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Fórmula:C38H57N7O8Pureza:99.55%Forma y color:SolidPeso molecular:739.9BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.Fórmula:C132H188N38O33S2Pureza:99.87%Forma y color:SoildPeso molecular:2899.27Ref: TM-TP1211L
1mg105,00€5mg398,00€10mg595,00€25mg1.064,00€50mg1.434,00€100mg1.948,00€200mg2.622,00€Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.Fórmula:C101H159N31O25Pureza:99.69%Forma y color:SolidPeso molecular:2207.58(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.Fórmula:C33H46N6O10Pureza:94.17%Forma y color:SoildPeso molecular:686.75Porcine dynorphin A(1-13) acetate
Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.Fórmula:C77H130N24O17Pureza:99.14%Forma y color:SolidPeso molecular:1664Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
Fórmula:C76H119N21O19Pureza:99.72%Forma y color:SolidPeso molecular:1630.89CTAP(TFA) (103429-32-9 free base)
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.Fórmula:C53H70F3N13O13S2Pureza:99.62%Forma y color:SolidPeso molecular:1218.33Nociceptin (1-13) amide TFA
Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).Fórmula:C63H101F3N22O17Pureza:97.64%Forma y color:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.Fórmula:C46H74N14O11Pureza:99.84%Forma y color:SolidPeso molecular:999.17[Met5]-Enkephalin, amide TFA
[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.Fórmula:C29H37F3N6O8SPureza:99.81%Forma y color:SolidPeso molecular:686.7Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Fórmula:C31H40F3N5O9Pureza:98.79%Forma y color:SolidPeso molecular:683.67Ref: TM-T20435L
1mg81,00€2mg105,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Fórmula:C51H79N15O16Pureza:95.54%Forma y color:SolidPeso molecular:1158.26N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Fórmula:C30H39N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:597.66b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Fórmula:C25H31N3O7Pureza:98.99%Forma y color:SolidPeso molecular:485.53Ref: TM-T21660L
5mg42,00€10mg57,00€25mg87,00€50mg131,00€100mg190,00€200mg285,00€1mL*10mM (DMSO)55,00€Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Fórmula:C51H73N15O11Pureza:98.59%Forma y color:SolidPeso molecular:1072.22Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Fórmula:C51H68N12O13Pureza:99.66%Forma y color:SolidPeso molecular:1057.16Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Fórmula:C59H95N19O14Pureza:99.88%Forma y color:SolidPeso molecular:1294.53[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.Fórmula:C30H42N6O8Pureza:99.36%Forma y color:SolidPeso molecular:614.69Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Fórmula:C31H41N7O9Pureza:98.92%Forma y color:SoildPeso molecular:655.7Ref: TM-T23076L
1mg309,00€2mg462,00€5mg697,00€10mg1.054,00€25mg1.549,00€50mg2.110,00€100mg2.840,00€1mL*10mM (DMSO)947,00€AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Fórmula:C23H29ClN2OPureza:98.66%Forma y color:SolidPeso molecular:384.94Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Fórmula:C18H25Cl3N2OPureza:99.04%Forma y color:SolidPeso molecular:391.76Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Fórmula:C26H27FN2O2Pureza:99.9% - 99.97%Forma y color:SolidPeso molecular:418.5Ref: TM-TQ0082
1mg40,00€2mg52,00€5mg88,00€10mg126,00€25mg259,00€50mg406,00€100mg607,00€1mL*10mM (DMSO)87,00€BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Fórmula:C30H31BrO4Pureza:98.76%Forma y color:SolidPeso molecular:535.47BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Fórmula:C29H39N5O7Pureza:>99.99%Forma y color:SolidPeso molecular:569.65Ref: TM-TP1905
2mg39,00€5mg58,00€10mg93,00€25mg145,00€50mg260,00€100mg462,00€200mg655,00€1mL*10mM (DMSO)73,00€
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