
Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Forma y color:SolidPeso molecular:683.67Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Forma y color:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Fórmula:C46H74N14O11Pureza:99.84%Forma y color:SolidPeso molecular:999.17BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Fórmula:C30H31BrO4Pureza:98.76%Forma y color:SolidPeso molecular:535.47Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C50H72N15O15SPureza:>99.99%Forma y color:SolidPeso molecular:1326.26Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Fórmula:C22H27NO4Pureza:98.97% - 99.86%Forma y color:SolidPeso molecular:369.45Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Fórmula:C59H95N19O14Pureza:99.88%Forma y color:SolidPeso molecular:1294.53[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Forma y color:SolidPeso molecular:569.65[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Fórmula:C30H42N6O8Pureza:99.36%Forma y color:SolidPeso molecular:614.69Difelikefalin acetate
CAS:<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Fórmula:C38H57N7O8Pureza:99.55%Forma y color:SolidPeso molecular:739.9Nociceptin
CAS:<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Fórmula:C79H129N27O22Pureza:99.35%Forma y color:SolidPeso molecular:1809.04LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Fórmula:C26H29ClF2N4O8SForma y color:SolidPeso molecular:631.04b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Forma y color:SolidPeso molecular:485.53BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Fórmula:C31H34O4Pureza:99.09%Forma y color:SolidPeso molecular:470.6Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Fórmula:C23H28O8Pureza:99.06%Forma y color:SolidPeso molecular:432.46Naloxegol oxalate
CAS:<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Fórmula:C36H55NO15Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:741.83MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Fórmula:C26H43Cl3N4Pureza:99.89% - 99.91%Forma y color:SolidPeso molecular:518.01BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Fórmula:C132H188N38O33S2Pureza:99.87%Forma y color:SoildPeso molecular:2899.27Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Fórmula:C21H26ClNO3Pureza:98% - 99.85%Forma y color:SolidPeso molecular:375.89AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Fórmula:C23H29ClN2OPureza:98.66%Forma y color:SolidPeso molecular:384.94
