Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Fórmula:C27H35N5O7SPureza:≥95%Forma y color:White Lyophilised SolidPeso molecular:573.66N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:597.66Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Fórmula:C32H37N5O5Pureza:99.64%Forma y color:SolidPeso molecular:571.67Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Fórmula:C21H26BrNO4Pureza:99.02%Forma y color:SolidPeso molecular:436.35EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Fórmula:C19H27ClF2N2O2Pureza:99.96%Forma y color:SolidPeso molecular:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Fórmula:C26H25N3O2·HClPureza:99.27% - 99.59%Forma y color:SolidPeso molecular:447.96Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Fórmula:C51H79N15O16Pureza:95.54%Forma y color:SolidPeso molecular:1158.26Dermorphin TFA
CAS:<p>Dermorphin TFA is a new class of opioids-like peptides</p>Fórmula:C42H51F3N8O12Pureza:98% - >99.99%Forma y color:SolidPeso molecular:916.89Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Fórmula:C37H52N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:768.86BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Fórmula:C16H15BrClNO3S2Pureza:98.42%Forma y color:SolidPeso molecular:448.78Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Fórmula:C101H159N31O25Pureza:99.69%Forma y color:SolidPeso molecular:2207.58ADL-5859
CAS:<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Fórmula:C24H28N2O3·HClPureza:98.78% - 99.11%Forma y color:SolidPeso molecular:428.95Sec-O-Glucosylhamaudol
CAS:<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Fórmula:C21H26O10Pureza:99.79%Forma y color:SolidPeso molecular:438.43BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Fórmula:C18H25Cl3N2OPureza:99.04%Forma y color:SolidPeso molecular:391.76Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Fórmula:C31H41N7O9Pureza:98.92%Forma y color:SoildPeso molecular:655.7(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Fórmula:C33H46N6O10Pureza:94.17%Forma y color:SoildPeso molecular:686.75Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Fórmula:C77H130N24O17Pureza:99.14%Forma y color:SolidPeso molecular:1664Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Forma y color:SolidPeso molecular:1072.22Naloxegol (NKTR-118)
CAS:<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Fórmula:C34H53NO11Forma y color:SolidPeso molecular:651.78Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Forma y color:White PowderPeso molecular:329.39
