Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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LY2940094
CAS:<p>LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.</p>Fórmula:C22H23ClF2N4O2SPureza:99.4%Forma y color:SolidPeso molecular:480.96Sinomenine hydrochloride
CAS:<p>Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.</p>Fórmula:C19H24ClNO4Pureza:99.43%Forma y color:SolidPeso molecular:365.851Apitegromab
CAS:<p>Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including</p>Pureza:95% - 97.59% (SDS-PAGE); 99.78% (SEC-HPLC)Forma y color:LiquidSamidorphan HCl
CAS:<p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>Fórmula:C21H27ClN2O4Pureza:96.79% - 97.85%Forma y color:SoildPeso molecular:406.9Naltrexone hydrochloride
CAS:<p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>Fórmula:C20H24ClNO4Pureza:98.72% - 99.65%Forma y color:White Crystalline PowderPeso molecular:377.862Meptazinol hydrochloride
CAS:<p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>Fórmula:C15H23NO·HClPureza:99.75%Forma y color:White SolidPeso molecular:269.81BTRX-335140
CAS:<p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>Fórmula:C25H32FN5O2Pureza:98% - 99.89%Forma y color:SolidPeso molecular:453.55Moguisteine
CAS:<p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>Fórmula:C16H21NO5SPureza:99.98%Forma y color:SolidPeso molecular:339.41Matrine
CAS:<p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>Fórmula:C15H24N2OPureza:97.16% - >99.99%Forma y color:SolidPeso molecular:248.36Trimebutine maleate
CAS:<p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>Fórmula:C26H33NO9Pureza:99.76% - 99.98%Forma y color:White SolidPeso molecular:503.55Loperamide hydrochloride
CAS:<p>Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.</p>Fórmula:C29H34Cl2N2O2Pureza:99.91% - >99.99%Forma y color:Crystals Practically Insoluble In WaterPeso molecular:513.50Alvimopan
CAS:<p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>Fórmula:C25H32N2O4Pureza:99.47% - 99.78%Forma y color:SolidPeso molecular:424.53ZT 52656A hydrochloride
CAS:<p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>Fórmula:C19H26ClF3N2OPureza:98.78%Forma y color:SolidPeso molecular:390.87CP 866087
CAS:<p>CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H30N2O3SPureza:99.22% - 99.74%Forma y color:SolidPeso molecular:426.57CSD-CH2(1,8)-NH2
<p>CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.</p>Fórmula:C76H125N25O15S2Pureza:98%Forma y color:SolidPeso molecular:1693.09DPDPE
CAS:<p>DPDPE is selective δ-opioid receptor agonist peptide.</p>Fórmula:C30H39N5O7S2Pureza:98%Forma y color:SolidPeso molecular:645.79UFP-101
CAS:<p>Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>Fórmula:C82H138N32O21Pureza:98%Forma y color:SolidPeso molecular:1908.19Dermorphin
CAS:<p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>Fórmula:C40H50N8O10Pureza:98.82%Forma y color:SolidPeso molecular:802.87SNC 80
CAS:<p>SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.</p>Fórmula:C28H39N3O2Pureza:99.65%Forma y color:SolidPeso molecular:449.63[DPro10] Dynorphin A (1-11)acetate,porcine
<p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>Fórmula:C65H107N21O15Pureza:99.05%Forma y color:SoildPeso molecular:1422.7Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Forma y color:Odour SolidDuP 747 HCl
CAS:<p>DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.</p>Fórmula:C24H29Cl3N2O2Pureza:99.85%Forma y color:SoildPeso molecular:483.86β-Endorphin, equine TFA
<p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>Fórmula:C156H249F3N42O46SForma y color:SolidPeso molecular:3537.96Frakefamide TFA
<p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>Fórmula:C32H35F4N5O7Forma y color:SolidPeso molecular:677.644-Hydroxy-1-(2-phenylethyl)piperidine
CAS:<p>4-Hydroxy-1-(2-phenylethyl)piperidine is a synthetic ligand for muscarinic acetylcholine receptors (mAChR) or non-opioid intracellular sigma-1 receptors (σ1 receptors). It serves as a metabolite of the opioid compounds furanylfentanyl and 4-fluoroisobutyryl fentanyl (FIBF).</p>Fórmula:C13H19NOForma y color:SolidPeso molecular:205.3U-48520
CAS:<p>U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.</p>Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82ICI 174,864
CAS:<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Fórmula:C38H53N5O7Pureza:98%Forma y color:White SolidPeso molecular:691.87DBPR116
CAS:<p>DBPR116 is a prodrug of BPRMU191 that can penetrate the blood-brain barrier. It significantly enhances the delivery efficiency of drugs targeting the central nervous system. When combined with the antagonist Naltrexone, DBPR116 demonstrates superior safety and analgesic effects compared to morphine in various in vivo pharmacological studies, including thermal pain models, cancer pain models, constipation, sedation, psychological dependence, heart rate, and respiratory frequency. As a strategy for peripheral administration, DBPR116 effectively alleviates pain while reducing adverse effects, showing promise as a safer opioid analgesic.</p>Fórmula:C19H18FNO3SForma y color:SolidPeso molecular:359.42AH 7959
CAS:<p>AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.</p>Fórmula:C19H26Cl2N2OForma y color:SolidPeso molecular:369.33Biphalin TFA
CAS:<p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>Fórmula:C46H56N10O10·xC2HF3O2Pureza:98%Forma y color:SolidPeso molecular:909.00 (free base)Ac-RYYRIK-NH2
CAS:<p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>Fórmula:C44H70N14O9Pureza:98%Forma y color:SolidPeso molecular:939.12Orphine
CAS:<p>Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.</p>Fórmula:C20H23N3OForma y color:SolidPeso molecular:321.42AH 7563
CAS:<p>AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.</p>Fórmula:C16H24N2OForma y color:SolidPeso molecular:260.38Corynantheidine
CAS:<p>Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.</p>Fórmula:C22H28N2O3Forma y color:SolidPeso molecular:368.47Axelopran
CAS:<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Fórmula:C26H39N3O4Forma y color:SolidPeso molecular:457.61DAMGO (TFA)
CAS:<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Fórmula:C28H36F3N5O8Pureza:98%Forma y color:SolidPeso molecular:627.61Fluorphine
CAS:<p>Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.</p>Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Fórmula:C38H38N2O5Forma y color:SolidPeso molecular:602.72HINT1-IN-1
<p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>Fórmula:C23H24N8O5Forma y color:SolidPeso molecular:492.49KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Fórmula:C21H25N3Forma y color:SolidPeso molecular:319.44Akuammicine
CAS:<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Fórmula:C20H22N2O2Forma y color:SolidPeso molecular:322.408Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Fórmula:C31H41N7O9Pureza:98%Forma y color:SolidPeso molecular:655.709[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Fórmula:C61H99FN22O15Pureza:98%Forma y color:SolidPeso molecular:1399.6Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Fórmula:C44H59N11O10Pureza:98%Forma y color:SolidPeso molecular:901.43KOR agonist 3
<p>KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.</p>Fórmula:C24H24N2O3Forma y color:SolidPeso molecular:388.46PL-017
CAS:<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Fórmula:C29H37N5O5Pureza:98%Forma y color:SolidPeso molecular:535.64(-)-9-Hydroxycorynantheidine
CAS:<p>(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.</p>Fórmula:C22H28N2O4Forma y color:SolidPeso molecular:384.47Ro 64-6198
CAS:<p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.</p>Fórmula:C26H31N3OPureza:98%Forma y color:SolidPeso molecular:401.54Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Fórmula:C49H75N15O14Pureza:98%Forma y color:SolidPeso molecular:1098.2Piperidylthiambutene hydrochloride
CAS:<p>Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.</p>Fórmula:C17H22ClNS2Forma y color:SolidPeso molecular:339.95[Nphe1]Nociceptin(1-13)NH2
CAS:<p>Competitive nociceptin receptor antagonist with pKi=8.4; no agonist activity; blocks nociceptin effects in vitro/in vivo.</p>Fórmula:C61H100N22O15Pureza:98%Forma y color:SolidPeso molecular:1381.6U-54494A hydrochloride
CAS:<p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>Fórmula:C18H25Cl3N2OForma y color:SolidPeso molecular:391.76AH 8529
CAS:<p>AH 8529 is an orally active opioid compound with analgesic properties.</p>Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82Gluten Exorphin B5
CAS:<p>Gluten exorphin B5 (GE-B5) is a food-derived opioid peptide identified in digests of wheat gluten.</p>Fórmula:C30H38N6O7Pureza:98%Forma y color:SolidPeso molecular:594.66Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Fórmula:C28H30O8Forma y color:SolidPeso molecular:494.53AH 8532
CAS:<p>AH 8532 is an opioid compound with analgesic effects and is effective in inhibiting the quinone-induced writhing response in mice, with an oral ED50 of 16 mg/kg.</p>Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82Dynorphin B (1-13)
CAS:<p>Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.</p>Fórmula:C74H115N21O17Pureza:98%Forma y color:SolidPeso molecular:1570.84Neuropeptide AF (human)
CAS:<p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>Fórmula:C90H132N26O25Pureza:98%Forma y color:SolidPeso molecular:1978.17CTAP
CAS:<p>Potent μ opioid antagonist, IC50 3.5 nM, 1200x selectivity over δ and somatostatin, brain-penetrant, active in vivo.</p>Fórmula:C51H69N13O11S2Pureza:98%Forma y color:White Solid/PowderPeso molecular:1104.32R-6890
CAS:<p>R-6890 is an opioid compound with analgesic properties.</p>Fórmula:C21H24ClN3OForma y color:SolidPeso molecular:369.89β-Naltrexamine dihydrochloride
CAS:<p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>Fórmula:C20H28Cl2N2O3Pureza:95.98%Forma y color:SoildPeso molecular:415.35N-Phenethylnoroxymorphone
CAS:<p>N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.</p>Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46CTOP
CAS:<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Fórmula:C50H67N11O11S2Pureza:98%Forma y color:SolidPeso molecular:1062.28Cebranopadol hemicitrate
CAS:<p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>Forma y color:SolidAP-238
CAS:<p>AP-238 is a novel synthetic opioid (NSO) that acts as an agonist for the μ-opioid receptor (MOR), with an EC50 of 248 nM. Additionally, AP-238 exhibits analgesic properties.</p>Fórmula:C18H26N2OForma y color:SolidPeso molecular:286.41MT-7716 free base
CAS:<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Fórmula:C27H28N4O2Pureza:98%Forma y color:SolidPeso molecular:440.54LY255582
CAS:<p>LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,</p>Fórmula:C22H35NO2Pureza:98%Forma y color:SolidPeso molecular:345.52BAM-22P
CAS:<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Fórmula:C130H184N38O31S2Pureza:98%Forma y color:SolidPeso molecular:2839.22TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Fórmula:C23H26Br2N2OForma y color:SolidPeso molecular:506.282Boc-ypgflt(O-tbu)
CAS:<p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>Fórmula:C44H64N6O11Forma y color:SolidPeso molecular:853.01Trimebutine
CAS:<p>Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal pain with antimuscarinic and weak mu-opioid</p>Fórmula:C22H29NO5Pureza:98.13% - 99.49%Forma y color:SolidPeso molecular:387.47(Rac)-SNC80
CAS:<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Fórmula:C28H39N3O2Forma y color:SolidPeso molecular:449.63Ac-RYYRWK-NH2
CAS:<p>Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.</p>Fórmula:C49H69N15O9Pureza:98%Forma y color:SolidPeso molecular:1012.17Naldemedine
CAS:<p>Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.</p>Fórmula:C32H34N4O6Forma y color:SolidPeso molecular:570.64AT-121 hydrochloride
CAS:<p>AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.</p>Fórmula:C24H39ClN4O3SPureza:97.28% - >99.99%Forma y color:SolidPeso molecular:499.11[Arg14,Lys15]Nociceptin
CAS:<p>Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>Fórmula:C82H137N31O22Pureza:98%Forma y color:SolidPeso molecular:1909.18N-Desmethyl Loperamide
CAS:<p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>Fórmula:C28H31ClN2O2Forma y color:SolidPeso molecular:463.01β-Endorphin, equine
CAS:<p>Endorphin Beta is A substance produced in the brain, especially in the pituitary gland, Endorphin Beta blocks the sensation of pain.</p>Fórmula:C154H248N42O44SPureza:98%Forma y color:SolidPeso molecular:3423.94MT-7716 hydrochloride
CAS:<p>MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)</p>Fórmula:C27H29ClN4O2Pureza:98%Forma y color:SolidPeso molecular:477(S,S)-J-113397
CAS:<p>(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .</p>Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57Clocinnamox mesylate
CAS:<p>Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).</p>Fórmula:C30H33ClN2O7SForma y color:SolidPeso molecular:601.11Adrenorphin
CAS:<p>Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C44H69N15O9SPureza:98%Forma y color:SolidPeso molecular:984.18[Met5]-Enkephalin, amide
CAS:<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Fórmula:C27H36N6O6SPureza:98%Forma y color:SolidPeso molecular:572.68Valorphin
CAS:<p>Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.</p>Fórmula:C44H61N9O11Pureza:98%Forma y color:SolidPeso molecular:892.01(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS:<p>E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioid</p>Fórmula:C50H81N15O9Forma y color:SolidPeso molecular:1036.27[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Fórmula:C63H101F3N22O17Forma y color:SolidPeso molecular:1495.61Nocistatin
CAS:<p>Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.</p>Fórmula:C32H56N10O12Forma y color:SolidPeso molecular:772.85Helianorphin-19
<p>Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.</p>Forma y color:Liquidβ-Lipotropin (60-65)
CAS:<p>β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.</p>Fórmula:C33H47N9O8SForma y color:SolidPeso molecular:729.85[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS:<p>'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'</p>Fórmula:C76H128N24O15Forma y color:SolidPeso molecular:1617.98β-Endorphin (rat)
CAS:<p>β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.</p>Fórmula:C157H254N42O44SForma y color:SolidPeso molecular:3466.07Dynorphin B (1-13) (TFA)
<p>Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .</p>Fórmula:C76H116N21F3O19Forma y color:SolidPeso molecular:1684.86Ac-RYYRWK-NH2 TFA
CAS:<p>Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.</p>Fórmula:C51H70F3N15O11Forma y color:SolidPeso molecular:1126.21Nociceptin (1-13), amide
CAS:<p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>Fórmula:C61H100N22O15Pureza:98%Forma y color:SolidPeso molecular:1381.59BPR1M97
CAS:<p>BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.</p>Fórmula:C18H18Cl2N2OPureza:98.78% - 99.95%Forma y color:SolidPeso molecular:349.25PIPE-3297
<p>PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.</p>Fórmula:C23H30N2OPeso molecular:350.23581β-Endorphin (1-27) (human)
CAS:<p>β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17,</p>Fórmula:C139H217N33O40SPureza:98%Forma y color:SolidPeso molecular:3022.47SB 205607 dihydrobromide
CAS:<p>non-peptide δ1 opioid receptor agonist</p>Fórmula:C23H24N2OPureza:98%Forma y color:SolidPeso molecular:344.45Dynorphin B (1-9)
CAS:<p>Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selective</p>Fórmula:C54H78N16O12Pureza:98%Forma y color:SolidPeso molecular:1143.3DALDA TFA
<p>DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.</p>Fórmula:C30H45N9O5·xC2HF3O2Pureza:98%Forma y color:SolidPeso molecular:611.74 (free base)Leumorphin, human
CAS:<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Fórmula:C150H224N42O46Pureza:98%Forma y color:SolidPeso molecular:3351.64Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Fórmula:C46H66N10O12S2Pureza:98.93%Forma y color:SolidPeso molecular:1015.21CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Fórmula:C34H35N5O4Forma y color:SolidPeso molecular:577.67N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Fórmula:C36H40N6O6Pureza:98%Forma y color:SolidPeso molecular:652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Fórmula:C32H45N5OForma y color:SolidPeso molecular:515.73Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Pureza:99.89%Forma y color:SoildCTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Fórmula:C52H71N11O13S2Pureza:99.87%Forma y color:SoildPeso molecular:1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Fórmula:C84H142N32O23Pureza:95.92%Forma y color:SolidPeso molecular:1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS:<p>is a ketone and a building block.</p>Fórmula:C38H57N7O8Pureza:96.94%Forma y color:SolidPeso molecular:739.9[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Fórmula:C63H103FN22O17Pureza:98.03%Forma y color:SolidPeso molecular:1459.63[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Fórmula:C31H43N5O9Pureza:98%Forma y color:SolidPeso molecular:629.65β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Fórmula:C141H221N33O42SPureza:96.52%Forma y color:SolidPeso molecular:3082.52β-Endorphin (6-31), human
CAS:<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Fórmula:C131H218N34O40Pureza:98%Forma y color:SolidPeso molecular:2909.38Deltorphin
CAS:<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Fórmula:C44H62N10O10S2Pureza:98.96%Forma y color:SolidPeso molecular:955.15Loperamide phenyl
CAS:<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Fórmula:C35H37ClN2O2Forma y color:SolidPeso molecular:553.14BMS-986121
CAS:<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Fórmula:C15H9Cl2N3O2SPureza:99.67%Forma y color:SolidPeso molecular:366.22[Leu5]-Enkephalin
CAS:<p>[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM</p>Fórmula:C28H37N5O7Pureza:99.87% - 99.88%Forma y color:SolidPeso molecular:555.62Porcine dynorphin A(1-13)
CAS:<p>Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.</p>Fórmula:C75H126N24O15Pureza:98%Forma y color:SolidPeso molecular:1603.95Endomorphin 2 TFA
CAS:<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Fórmula:C34H38F3N5O7Forma y color:SolidPeso molecular:685.69BAN ORL 24 dihydrochloride
CAS:<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Fórmula:C27H37Cl2N3O2Pureza:95.03%Forma y color:SolidPeso molecular:506.51Alvimopan dihydrate (LY246736 dihydrate)
CAS:<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Fórmula:C25H36N2O6Forma y color:SolidPeso molecular:460.56Asimadoline
CAS:<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54GR103545
CAS:<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Fórmula:C23H29Cl2N3O7Pureza:99.75%Forma y color:SolidPeso molecular:530.4Endomorphin 1
CAS:<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Fórmula:C34H38N6O5Pureza:95.92%Forma y color:Solid (Solid Powder )Peso molecular:610.7DPDPE TFA (88373-73-3 free base)
CAS:<p>DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.</p>Fórmula:C32H40F3N5O9S2Pureza:99.39%Forma y color:SolidPeso molecular:759.81CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Fórmula:C53H70F3N13O13S2Pureza:99.62%Forma y color:SolidPeso molecular:1218.33Gluten Exorphin C
CAS:<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Fórmula:C29H45N5O8Pureza:99.39%Forma y color:SolidPeso molecular:591.7ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Fórmula:C24H29ClN2O3Forma y color:SolidPeso molecular:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Fórmula:C19H27N3O2SPureza:99.93% - >99.99%Forma y color:SolidPeso molecular:361.5Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Fórmula:C27H31ClN2O2Pureza:98.94% - 99.32%Forma y color:SolidPeso molecular:451.01Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Fórmula:C51H68N12O13Pureza:99.66%Forma y color:SolidPeso molecular:1057.16DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Fórmula:C26H35N5O6Pureza:98.83% - 99.92%Forma y color:SolidPeso molecular:513.59MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Fórmula:C26H40N4Forma y color:SolidPeso molecular:408.62Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Fórmula:C38H54N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:782.88DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Fórmula:C28H36F3N5O8Pureza:98.67% - 99.76%Forma y color:SolidPeso molecular:627.6BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Fórmula:C29H39N5O7Pureza:>99.99%Forma y color:SolidPeso molecular:569.65N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Forma y color:Yellow Crystalline SolidPeso molecular:312.8GR 89696 free base
CAS:<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Fórmula:C19H25Cl2N3O3Forma y color:SolidPeso molecular:414.33Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Fórmula:C26H27FN2O2Pureza:99.53% - 99.93%Forma y color:SolidPeso molecular:418.5EST73502 hydrochloride
CAS:<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Fórmula:C19H27ClF2N2O2Forma y color:SolidPeso molecular:388.88Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Forma y color:SolidPeso molecular:683.67Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Forma y color:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Fórmula:C46H74N14O11Pureza:99.84%Forma y color:SolidPeso molecular:999.17BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Fórmula:C30H31BrO4Pureza:98.76%Forma y color:SolidPeso molecular:535.47Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C50H72N15O15SPureza:>99.99%Forma y color:SolidPeso molecular:1326.26Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Fórmula:C22H27NO4Pureza:98.97% - 99.86%Forma y color:SolidPeso molecular:369.45Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Fórmula:C59H95N19O14Pureza:99.88%Forma y color:SolidPeso molecular:1294.53[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Forma y color:SolidPeso molecular:569.65[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Fórmula:C30H42N6O8Pureza:99.36%Forma y color:SolidPeso molecular:614.69Difelikefalin acetate
CAS:<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Fórmula:C38H57N7O8Pureza:99.55%Forma y color:SolidPeso molecular:739.9Nociceptin
CAS:<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Fórmula:C79H129N27O22Pureza:99.35%Forma y color:SolidPeso molecular:1809.04LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Fórmula:C26H29ClF2N4O8SForma y color:SolidPeso molecular:631.04b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Forma y color:SolidPeso molecular:485.53BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Fórmula:C31H34O4Pureza:99.09%Forma y color:SolidPeso molecular:470.6Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Fórmula:C23H28O8Pureza:99.06%Forma y color:SolidPeso molecular:432.46Naloxegol oxalate
CAS:<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Fórmula:C36H55NO15Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:741.83MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Fórmula:C26H43Cl3N4Pureza:99.89% - 99.91%Forma y color:SolidPeso molecular:518.01BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Fórmula:C132H188N38O33S2Pureza:99.87%Forma y color:SoildPeso molecular:2899.27Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Fórmula:C21H26ClNO3Pureza:98% - 99.85%Forma y color:SolidPeso molecular:375.89AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Fórmula:C23H29ClN2OPureza:98.66%Forma y color:SolidPeso molecular:384.94Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Fórmula:C27H35N5O7SPureza:≥95%Forma y color:White Lyophilised SolidPeso molecular:573.66N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:597.66Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Fórmula:C32H37N5O5Pureza:99.64%Forma y color:SolidPeso molecular:571.67Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Fórmula:C21H26BrNO4Pureza:99.02%Forma y color:SolidPeso molecular:436.35EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Fórmula:C19H27ClF2N2O2Pureza:99.96%Forma y color:SolidPeso molecular:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Fórmula:C26H25N3O2·HClPureza:99.27% - 99.59%Forma y color:SolidPeso molecular:447.96Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Fórmula:C51H79N15O16Pureza:95.54%Forma y color:SolidPeso molecular:1158.26Dermorphin TFA
CAS:<p>Dermorphin TFA is a new class of opioids-like peptides</p>Fórmula:C42H51F3N8O12Pureza:98% - >99.99%Forma y color:SolidPeso molecular:916.89Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Fórmula:C37H52N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:768.86BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Fórmula:C16H15BrClNO3S2Pureza:98.42%Forma y color:SolidPeso molecular:448.78Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Fórmula:C101H159N31O25Pureza:99.69%Forma y color:SolidPeso molecular:2207.58ADL-5859
CAS:<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Fórmula:C24H28N2O3·HClPureza:98.78% - 99.11%Forma y color:SolidPeso molecular:428.95Sec-O-Glucosylhamaudol
CAS:<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Fórmula:C21H26O10Pureza:99.79%Forma y color:SolidPeso molecular:438.43BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Fórmula:C18H25Cl3N2OPureza:99.04%Forma y color:SolidPeso molecular:391.76Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Fórmula:C31H41N7O9Pureza:98.92%Forma y color:SoildPeso molecular:655.7(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Fórmula:C33H46N6O10Pureza:94.17%Forma y color:SoildPeso molecular:686.75Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Fórmula:C77H130N24O17Pureza:99.14%Forma y color:SolidPeso molecular:1664Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Forma y color:SolidPeso molecular:1072.22Naloxegol (NKTR-118)
CAS:<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Fórmula:C34H53NO11Forma y color:SolidPeso molecular:651.78Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Forma y color:White PowderPeso molecular:329.39Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Fórmula:C76H119N21O19Pureza:99.72%Forma y color:SolidPeso molecular:1630.89Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Forma y color:SolidPeso molecular:407.89Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Fórmula:C25H34N2O5Pureza:98%Forma y color:SolidPeso molecular:442.55[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Fórmula:C29H37F3N6O8SPureza:99.81%Forma y color:SolidPeso molecular:686.7GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Fórmula:C25H26ClN3OForma y color:SolidPeso molecular:419.95LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Fórmula:C19H24N2O2Pureza:98%Forma y color:SolidPeso molecular:312.41ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Fórmula:C19H14Cl2N4OSForma y color:SolidPeso molecular:417.31SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Fórmula:C28H31NOPureza:99.54%Forma y color:SolidPeso molecular:397.55μ opioid receptor agonist 2
CAS:<p>μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>Fórmula:C25H34N4OForma y color:SolidPeso molecular:406.56TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Fórmula:C37H38N4O6Pureza:98%Forma y color:SolidPeso molecular:634.72Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Fórmula:C18H23NO2Pureza:98%Forma y color:SolidPeso molecular:285.38LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Fórmula:C24H22F2N2O2Pureza:99.18%Forma y color:SolidPeso molecular:408.44BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Fórmula:C27H37N3O2Forma y color:SolidPeso molecular:435.6ML 190
CAS:<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Fórmula:C27H32N6O3Pureza:99.88%Forma y color:SolidPeso molecular:488.58GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H21ClF2N4Pureza:98%Forma y color:SolidPeso molecular:438.9ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Fórmula:C24H28N2O3Pureza:98%Forma y color:SolidPeso molecular:392.49DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Fórmula:C22H24Cl3N3OSPureza:98%Forma y color:SolidPeso molecular:484.87PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Fórmula:C21H29ClN2O2SPureza:99.59%Forma y color:SolidPeso molecular:408.99CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H28N2O2Pureza:99.56% - >99.99%Forma y color:SoildPeso molecular:376.49
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