Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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Leumorphin, human
CAS:<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Fórmula:C150H224N42O46Pureza:98%Forma y color:SolidPeso molecular:3351.64Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Fórmula:C46H66N10O12S2Pureza:98.93%Forma y color:SolidPeso molecular:1015.21CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Fórmula:C34H35N5O4Forma y color:SolidPeso molecular:577.67N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Fórmula:C36H40N6O6Pureza:98%Forma y color:SolidPeso molecular:652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Fórmula:C32H45N5OForma y color:SolidPeso molecular:515.73Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Pureza:99.89%Forma y color:SoildCTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Fórmula:C52H71N11O13S2Pureza:99.87%Forma y color:SoildPeso molecular:1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Fórmula:C84H142N32O23Pureza:95.92%Forma y color:SolidPeso molecular:1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS:<p>is a ketone and a building block.</p>Fórmula:C38H57N7O8Pureza:96.94%Forma y color:SolidPeso molecular:739.9[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Fórmula:C63H103FN22O17Pureza:98.03%Forma y color:SolidPeso molecular:1459.63[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Fórmula:C31H43N5O9Pureza:98%Forma y color:SolidPeso molecular:629.65β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Fórmula:C141H221N33O42SPureza:96.52%Forma y color:SolidPeso molecular:3082.52β-Endorphin (6-31), human
CAS:<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Fórmula:C131H218N34O40Pureza:98%Forma y color:SolidPeso molecular:2909.38Deltorphin
CAS:<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Fórmula:C44H62N10O10S2Pureza:98.96%Forma y color:SolidPeso molecular:955.15Loperamide phenyl
CAS:<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Fórmula:C35H37ClN2O2Forma y color:SolidPeso molecular:553.14BMS-986121
CAS:<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Fórmula:C15H9Cl2N3O2SPureza:99.67%Forma y color:SolidPeso molecular:366.22[Leu5]-Enkephalin
CAS:<p>[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM</p>Fórmula:C28H37N5O7Pureza:99.87% - 99.88%Forma y color:SolidPeso molecular:555.62Porcine dynorphin A(1-13)
CAS:<p>Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.</p>Fórmula:C75H126N24O15Pureza:98%Forma y color:SolidPeso molecular:1603.95Endomorphin 2 TFA
CAS:<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Fórmula:C34H38F3N5O7Forma y color:SolidPeso molecular:685.69BAN ORL 24 dihydrochloride
CAS:<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Fórmula:C27H37Cl2N3O2Pureza:95.03%Forma y color:SolidPeso molecular:506.51Alvimopan dihydrate (LY246736 dihydrate)
CAS:<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Fórmula:C25H36N2O6Forma y color:SolidPeso molecular:460.56Asimadoline
CAS:<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54GR103545
CAS:<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Fórmula:C23H29Cl2N3O7Pureza:99.75%Forma y color:SolidPeso molecular:530.4Endomorphin 1
CAS:<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Fórmula:C34H38N6O5Pureza:95.92%Forma y color:Solid (Solid Powder )Peso molecular:610.7DPDPE TFA (88373-73-3 free base)
CAS:<p>DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.</p>Fórmula:C32H40F3N5O9S2Pureza:99.39%Forma y color:SolidPeso molecular:759.81CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Fórmula:C53H70F3N13O13S2Pureza:99.62%Forma y color:SolidPeso molecular:1218.33Gluten Exorphin C
CAS:<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Fórmula:C29H45N5O8Pureza:99.39%Forma y color:SolidPeso molecular:591.7ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Fórmula:C24H29ClN2O3Forma y color:SolidPeso molecular:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Fórmula:C19H27N3O2SPureza:99.93% - >99.99%Forma y color:SolidPeso molecular:361.5Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Fórmula:C27H31ClN2O2Pureza:98.94% - 99.32%Forma y color:SolidPeso molecular:451.01Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Fórmula:C51H68N12O13Pureza:99.66%Forma y color:SolidPeso molecular:1057.16DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Fórmula:C26H35N5O6Pureza:98.83% - 99.92%Forma y color:SolidPeso molecular:513.59MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Fórmula:C26H40N4Forma y color:SolidPeso molecular:408.62Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Fórmula:C38H54N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:782.88DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Fórmula:C28H36F3N5O8Pureza:98.67% - 99.76%Forma y color:SolidPeso molecular:627.6BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Fórmula:C29H39N5O7Pureza:>99.99%Forma y color:SolidPeso molecular:569.65N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Fórmula:C17H17ClN4Pureza:97.25% - 99.83%Forma y color:Yellow Crystalline SolidPeso molecular:312.8GR 89696 free base
CAS:<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Fórmula:C19H25Cl2N3O3Forma y color:SolidPeso molecular:414.33Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Fórmula:C26H27FN2O2Pureza:99.53% - 99.93%Forma y color:SolidPeso molecular:418.5EST73502 hydrochloride
CAS:<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Fórmula:C19H27ClF2N2O2Forma y color:SolidPeso molecular:388.88Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Fórmula:C31H40F3N5O9Pureza:98.79%Forma y color:SolidPeso molecular:683.67Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Fórmula:C63H101F3N22O17Pureza:97.64%Forma y color:SolidPeso molecular:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Fórmula:C46H74N14O11Pureza:99.84%Forma y color:SolidPeso molecular:999.17BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Fórmula:C30H31BrO4Pureza:98.76%Forma y color:SolidPeso molecular:535.47Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Fórmula:C50H72N15O15SPureza:>99.99%Forma y color:SolidPeso molecular:1326.26Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Fórmula:C22H27NO4Pureza:98.97% - 99.86%Forma y color:SolidPeso molecular:369.45Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Fórmula:C59H95N19O14Pureza:99.88%Forma y color:SolidPeso molecular:1294.53[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Fórmula:C29H39N5O7Pureza:98.06%Forma y color:SolidPeso molecular:569.65[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Fórmula:C30H42N6O8Pureza:99.36%Forma y color:SolidPeso molecular:614.69Difelikefalin acetate
CAS:<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Fórmula:C38H57N7O8Pureza:99.55%Forma y color:SolidPeso molecular:739.9
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