Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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Nociceptin
CAS:<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Fórmula:C79H129N27O22Pureza:99.35%Forma y color:SolidPeso molecular:1809.04LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Fórmula:C26H29ClF2N4O8SForma y color:SolidPeso molecular:631.04b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Fórmula:C25H31N3O7Pureza:98.99%Forma y color:SolidPeso molecular:485.53BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Fórmula:C31H34O4Pureza:99.09%Forma y color:SolidPeso molecular:470.6Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Fórmula:C23H28O8Pureza:99.06%Forma y color:SolidPeso molecular:432.46Naloxegol oxalate
CAS:<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Fórmula:C36H55NO15Pureza:99.67% - >99.99%Forma y color:SolidPeso molecular:741.83MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Fórmula:C26H43Cl3N4Pureza:99.89% - 99.91%Forma y color:SolidPeso molecular:518.01BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Fórmula:C132H188N38O33S2Pureza:99.87%Forma y color:SoildPeso molecular:2899.27Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Fórmula:C21H26ClNO3Pureza:98% - 99.85%Forma y color:SolidPeso molecular:375.89AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Fórmula:C23H29ClN2OPureza:98.66%Forma y color:SolidPeso molecular:384.94Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Fórmula:C27H35N5O7SPureza:≥95%Forma y color:White Lyophilised SolidPeso molecular:573.66N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Fórmula:C30H39N5O8Pureza:>99.99%Forma y color:SolidPeso molecular:597.66Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Fórmula:C32H37N5O5Pureza:99.64%Forma y color:SolidPeso molecular:571.67Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Fórmula:C21H26BrNO4Pureza:99.02%Forma y color:SolidPeso molecular:436.35EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Fórmula:C19H27ClF2N2O2Pureza:99.96%Forma y color:SolidPeso molecular:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Fórmula:C26H25N3O2·HClPureza:99.27% - 99.59%Forma y color:SolidPeso molecular:447.96Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Fórmula:C51H79N15O16Pureza:95.54%Forma y color:SolidPeso molecular:1158.26Dermorphin TFA
CAS:<p>Dermorphin TFA is a new class of opioids-like peptides</p>Fórmula:C42H51F3N8O12Pureza:98% - >99.99%Forma y color:SolidPeso molecular:916.89Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Fórmula:C37H52N8O10Pureza:>99.99%Forma y color:SolidPeso molecular:768.86BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Fórmula:C16H15BrClNO3S2Pureza:98.42%Forma y color:SolidPeso molecular:448.78Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Fórmula:C101H159N31O25Pureza:99.69%Forma y color:SolidPeso molecular:2207.58ADL-5859
CAS:<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Fórmula:C24H28N2O3·HClPureza:98.78% - 99.11%Forma y color:SolidPeso molecular:428.95Sec-O-Glucosylhamaudol
CAS:<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Fórmula:C21H26O10Pureza:99.79%Forma y color:SolidPeso molecular:438.43BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Fórmula:C18H25Cl3N2OPureza:99.04%Forma y color:SolidPeso molecular:391.76Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Fórmula:C31H41N7O9Pureza:98.92%Forma y color:SoildPeso molecular:655.7(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Fórmula:C33H46N6O10Pureza:94.17%Forma y color:SoildPeso molecular:686.75Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Fórmula:C77H130N24O17Pureza:99.14%Forma y color:SolidPeso molecular:1664Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Fórmula:C51H73N15O11Pureza:98.59%Forma y color:SolidPeso molecular:1072.22Naloxegol (NKTR-118)
CAS:<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Fórmula:C34H53NO11Forma y color:SolidPeso molecular:651.78Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Fórmula:C19H23NO4Pureza:99.02% - 99.73%Forma y color:White PowderPeso molecular:329.39Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Fórmula:C76H119N21O19Pureza:99.72%Forma y color:SolidPeso molecular:1630.89Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Forma y color:SolidPeso molecular:407.89Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Fórmula:C25H34N2O5Pureza:98%Forma y color:SolidPeso molecular:442.55[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Fórmula:C29H37F3N6O8SPureza:99.81%Forma y color:SolidPeso molecular:686.7GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Fórmula:C25H26ClN3OForma y color:SolidPeso molecular:419.95LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Fórmula:C19H24N2O2Pureza:98%Forma y color:SolidPeso molecular:312.41ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Fórmula:C19H14Cl2N4OSForma y color:SolidPeso molecular:417.31SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Fórmula:C28H31NOPureza:99.54%Forma y color:SolidPeso molecular:397.55μ opioid receptor agonist 2
CAS:<p>μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>Fórmula:C25H34N4OForma y color:SolidPeso molecular:406.56TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Fórmula:C37H38N4O6Pureza:98%Forma y color:SolidPeso molecular:634.72Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Fórmula:C18H23NO2Pureza:98%Forma y color:SolidPeso molecular:285.38LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Fórmula:C24H22F2N2O2Pureza:99.18%Forma y color:SolidPeso molecular:408.44BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Fórmula:C27H37N3O2Forma y color:SolidPeso molecular:435.6ML 190
CAS:<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Fórmula:C27H32N6O3Pureza:99.88%Forma y color:SolidPeso molecular:488.58GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H21ClF2N4Pureza:98%Forma y color:SolidPeso molecular:438.9ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Fórmula:C24H28N2O3Pureza:98%Forma y color:SolidPeso molecular:392.49DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Fórmula:C22H24Cl3N3OSPureza:98%Forma y color:SolidPeso molecular:484.87PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Fórmula:C21H29ClN2O2SPureza:99.59%Forma y color:SolidPeso molecular:408.99CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H28N2O2Pureza:99.56% - >99.99%Forma y color:SoildPeso molecular:376.49
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