Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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ORL1 antagonist 1
CAS:<p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>Fórmula:C20H22ClN5Pureza:98.92%Forma y color:SolidPeso molecular:367.88ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Fórmula:C34H46N4O6SPureza:98%Forma y color:SolidPeso molecular:638.82JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Fórmula:C26H25N3O2Pureza:98%Forma y color:SolidPeso molecular:411.5LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Fórmula:C28H41N5O4Forma y color:SolidPeso molecular:511.66SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Fórmula:C25H37FN4Pureza:98%Forma y color:SolidPeso molecular:412.59BMS-986124
CAS:<p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>Fórmula:C16H15BrClNO3S2Forma y color:SolidPeso molecular:448.78DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Fórmula:C20H20N2Pureza:98%Forma y color:SolidPeso molecular:288.39Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Fórmula:C21H31ClN2OPureza:98%Forma y color:SolidPeso molecular:362.94Ici 174865
CAS:<p>Ici 174865 is a delta opioid receptor antagonist agent.</p>Fórmula:C38H53N5O7Forma y color:SolidPeso molecular:691.86Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Fórmula:C36H42N6O7Forma y color:SolidPeso molecular:670.75Axomadol
CAS:<p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>Fórmula:C16H25NO3Pureza:98%Forma y color:SolidPeso molecular:279.37LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Fórmula:C32H42N4O6Pureza:98%Forma y color:SolidPeso molecular:578.7Diallyl G
CAS:<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Fórmula:C38H53N5O8Forma y color:SolidPeso molecular:707.86Loperamide oxide
CAS:<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Fórmula:C29H33ClN2O3Forma y color:SolidPeso molecular:493.04CR-665 Acetate
CAS:<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Fórmula:C38H53N9O6Forma y color:SolidPeso molecular:731.899AZD7268
CAS:<p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>Fórmula:C29H30N4O2SForma y color:SolidPeso molecular:498.64AT-076
CAS:<p>AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.</p>Fórmula:C26H35N3O3Forma y color:SolidPeso molecular:437.57GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H23F2N4O4PPureza:98%Forma y color:SolidPeso molecular:500.43Dup 747
CAS:<p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>Fórmula:C24H28Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:447.4σ1 Receptor/μ Opioid receptor modulator 1
CAS:<p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>Fórmula:C24H31FN2O2Forma y color:SolidPeso molecular:398.51Norbinaltorphimine
CAS:<p>nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.</p>Fórmula:C40H43N3O6Forma y color:SolidPeso molecular:661.79GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Fórmula:C24H20F2N4Pureza:99.85%Forma y color:SolidPeso molecular:402.44ADL-5747
CAS:<p>ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal</p>Fórmula:C24H28N2O3Pureza:98.94% - 99.74%Forma y color:SolidPeso molecular:392.49GR 89696 fumarate
CAS:<p>GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.</p>Fórmula:C23H29Cl2N3O7Pureza:99.84%Forma y color:SolidPeso molecular:530.4NNC 63-0532
CAS:<p>NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.</p>Fórmula:C27H29N3O3Pureza:99.53%Forma y color:SolidPeso molecular:443.54SCH-486757
CAS:<p>SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.</p>Fórmula:C24H23Cl2N3OPureza:99.53% - >99.99%Forma y color:SolidPeso molecular:440.37Trimebutine CTB salt
CAS:<p>Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.</p>Fórmula:C29H36N2O8S2Pureza:99.85% - >99.99%Forma y color:SolidPeso molecular:604.74IPAG
CAS:<p>IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.</p>Fórmula:C17H22IN3Pureza:99.65%Forma y color:SolidPeso molecular:395.28ICI 199,441 hydrochloride
CAS:<p>ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.</p>Fórmula:C21H25Cl3N2OPureza:99.57%Forma y color:SolidPeso molecular:427.8ICI 204,448
CAS:<p>ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.</p>Fórmula:C23H27Cl3N2O4Pureza:>99.99%Forma y color:SolidPeso molecular:501.83Bevenopran
CAS:<p>Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.</p>Fórmula:C20H26N4O4Pureza:98.69% - 98.9%Forma y color:SolidPeso molecular:386.44JNJ-20788560
CAS:<p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>Fórmula:C25H28N2O2Pureza:98.02%Forma y color:SolidPeso molecular:388.5ML-335
CAS:<p>ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.</p>Fórmula:C25H32N2O3Pureza:98.52%Forma y color:SolidPeso molecular:408.53AT-121
CAS:<p>AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).</p>Fórmula:C24H38N4O3SPureza:98.49% - 99.73%Forma y color:SolidPeso molecular:462.65SNC 162
CAS:<p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>Fórmula:C27H37N3OPureza:98%Forma y color:SolidPeso molecular:419.6CYT-1010
CAS:<p>CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.</p>Fórmula:C35H40N6O5Pureza:98%Forma y color:SolidPeso molecular:624.73Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Fórmula:C22H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:386.91Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Fórmula:C38H42N4O6Forma y color:SolidPeso molecular:650.76μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Fórmula:C22H28N2O2Pureza:98%Forma y color:SolidPeso molecular:352.47R-84760 hydrochloride
CAS:<p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>Fórmula:C19H25Cl3N2OSForma y color:SolidPeso molecular:435.84DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Fórmula:C30H34FN3O2Pureza:98%Forma y color:SolidPeso molecular:487.61Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Fórmula:C34H48N6O10Pureza:98%Forma y color:SolidPeso molecular:700.78Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Fórmula:C30H34FN5O5Pureza:98%Forma y color:SolidPeso molecular:563.62Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Fórmula:C23H26N4O3Pureza:98%Forma y color:SolidPeso molecular:406.48μ opioid receptor agonist 1
CAS:<p>μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can</p>Fórmula:C26H38N4OForma y color:SolidPeso molecular:422.61Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Fórmula:C38H43ClN4O6Pureza:98%Forma y color:SolidPeso molecular:687.22ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Fórmula:C23H26Cl2N2O4Forma y color:SolidPeso molecular:465.37N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Fórmula:C33H33ClN2O3Pureza:98%Forma y color:SolidPeso molecular:541.08Trap-101 hydrochloride
CAS:<p>nociceptin/orphanin FQ (NOP) receptor antagonist</p>Fórmula:C24H36ClN3O2Pureza:98%Forma y color:SolidPeso molecular:434.02ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.49
